Compile Data Set for Download or QSAR
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Found 9 Enz. Inhib. hit(s) with all data for entry = 50037275
TargetDelta-type opioid receptor(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM21864((21R)-22-(cyclopropylmethyl)-14-oxa-11,22-diazahep...)
Affinity DataKi:  0.0700nMAssay Description:[3H]-Cl-DPDPE competition binding assay using human cloned opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50138632(1-Phenyl-cyclopentanecarboxylic acid [(S)-5-(3-hyd...)
Affinity DataKi:  0.960nMAssay Description:[3H]-Cl-DPDPE competition binding assay using human cloned opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50138633(1-Phenyl-cyclopentanecarboxylic acid [5-(3-hydroxy...)
Affinity DataKi:  2.10nMAssay Description:[3H]-Cl-DPDPE competition binding assay using human cloned opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50138634(1-Phenyl-cyclopentanecarboxylic acid [(R)-5-(3-hyd...)
Affinity DataKi:  9.30nMAssay Description:[3H]-Cl-DPDPE competition binding assay using human cloned opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50006946(2-[2-(2-{2-[2-Diallylamino-3-(4-hydroxy-phenyl)-pr...)
Affinity DataKi:  19nMAssay Description:Binding affinity towards opioid receptor delta 1 expressed in CHO cells was determined by using [3H]DPDPE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50138632(1-Phenyl-cyclopentanecarboxylic acid [(S)-5-(3-hyd...)
Affinity DataIC50:  1.80nMAssay Description:Inverse agonist potency at cloned human delta-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50138633(1-Phenyl-cyclopentanecarboxylic acid [5-(3-hydroxy...)
Affinity DataIC50:  2.40nMAssay Description:Inverse agonist potency at cloned human delta-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50064515(3-[(3R,4R)-3,4-Dimethyl-1-((E)-3-o-tolyl-allyl)-pi...)
Affinity DataIC50:  2.80nMAssay Description:Inverse agonist potency at cloned human opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50138634(1-Phenyl-cyclopentanecarboxylic acid [(R)-5-(3-hyd...)
Affinity DataIC50:  15nMAssay Description:Inverse agonist potency at cloned human opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed