Compile Data Set for Download or QSAR
maximum 50k data
Found 12 Enz. Inhib. hit(s) with all data for entry = 50014288
TargetIntegrase(Human immunodeficiency virus 1)
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM23400((2Z)-4-(3-benzylphenyl)-2-hydroxy-4-oxobut-2-enoic...)
Affinity DataIC50: <100nMAssay Description:Inhibition of Integrase (3'-processing) as measured in an in vitro assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50115572((Z)-4-(3-Benzyloxy-phenyl)-2-hydroxy-4-oxo-but-2-e...)
Affinity DataIC50:  350nMAssay Description:Inhibition of Integrase (3'-processing) as measured in an in vitro assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50140324(4-(3-Benzoyl-phenyl)-2,4-dioxo-butyric acid | CHEM...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of Integrase (3'-processing) as measured in an in vitro assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50140324(4-(3-Benzoyl-phenyl)-2,4-dioxo-butyric acid | CHEM...)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of integrase catalyzed strand transfer (ST) as measured in an in vitro assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50140323(4-(3-Azido-phenyl)-2,4-dioxo-butyric acid | CHEMBL...)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of Integrase catalyzed strand transfer (ST) as measured in an in vitro assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50140323(4-(3-Azido-phenyl)-2,4-dioxo-butyric acid | CHEMBL...)
Affinity DataIC50:  5.30E+3nMAssay Description:Inhibition of Integrase (3'-processing) as measured in an in vitro assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50140322(4-[3-(4-Benzoyl-benzyloxy)-phenyl]-2,4-dioxo-butyr...)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of Integrase catalyzed strand transfer (ST) as measured in an in vitro assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50140322(4-[3-(4-Benzoyl-benzyloxy)-phenyl]-2,4-dioxo-butyr...)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of integrase catalyzed strand transfer (ST) as measured in an in vitro assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50115579((Z)-2-hydroxy-4-oxo-4-phenyl-but-2-enoic acid | 2-...)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of Integrase catalyzed strand transfer (ST) as measured in an in vitro assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50140322(4-[3-(4-Benzoyl-benzyloxy)-phenyl]-2,4-dioxo-butyr...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Integrase (3'-processing) as measured in an in vitro assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50140323(4-(3-Azido-phenyl)-2,4-dioxo-butyric acid | CHEMBL...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Integrase (3'-processing) as measured in an in vitro assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50140324(4-(3-Benzoyl-phenyl)-2,4-dioxo-butyric acid | CHEM...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Integrase catalyzed strand transfer (ST) as measured in an in vitro assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed