Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with all data for entry = 50004688
TargetSolute carrier organic anion transporter family member 4C1(Homo sapiens)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM46356(DIGITOXIN | MLS000069787 | SMR000058529 | US106680...)
Affinity DataIC50:  120nMAssay Description:TP_TRANSPORTER: inhibition of Digoxin uptake in OATP4C1-expressing MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 4C1(Homo sapiens)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM225707(CS337 | Digoxigenin)
Affinity DataIC50:  490nMAssay Description:TP_TRANSPORTER: inhibition of Digoxin uptake in OATP4C1-expressing MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 4C1(Homo sapiens)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50301375(3,3',5,5'-tetraiodo-L-thyronine | 3,5,3',5'-tetrai...)
Affinity DataIC50:  8.00E+3nMAssay Description:TP_TRANSPORTER: inhibition of Triiodothyronine uptake in OATP4C1-expressing MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed