Compile Data Set for Download or QSAR
maximum 50k data
Found 7 Enz. Inhib. hit(s) with all data for entry = 50015094
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Institute

Curated by ChEMBL
LigandPNGBDBM50151228(6-[Cyclopropylidene-(5,5,8,8-tetramethyl-3-propoxy...)
Affinity DataIC50:  6nMAssay Description:Inhibition of [3H]-9-cis-retinoic acid binding to human retinoid X receptor alpha ligand-binding domain expressed in E. coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Institute

Curated by ChEMBL
LigandPNGBDBM50151230(6-[(3-Butoxy-5,5,8,8-tetramethyl-5,6,7,8-tetrahydr...)
Affinity DataIC50:  10nMAssay Description:Inhibition of [3H]-9-cis-retinoic acid binding to human retinoid X receptor alpha ligand-binding domain expressed in E. coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Institute

Curated by ChEMBL
LigandPNGBDBM50151229(4-[Cyclopropylidene-(3,5,5,8,8-pentamethyl-5,6,7,8...)
Affinity DataIC50:  21nMAssay Description:Inhibition of [3H]-9-cis-retinoic acid binding to human retinoid X receptor alpha ligand-binding domain expressed in E. coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Institute

Curated by ChEMBL
LigandPNGBDBM31892(9-cis retinoic acid | 9C-RA | CHEMBL705 | Panretin...)
Affinity DataIC50:  29nMAssay Description:Inhibition of [3H]-9-cis-retinoic acid binding to human retinoid X receptor alpha ligand-binding domain expressed in E. coliMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Institute

Curated by ChEMBL
LigandPNGBDBM50151231(4-[Cyclopropylidene-(5,5,8,8-tetramethyl-3-propoxy...)
Affinity DataIC50:  120nMAssay Description:Inhibition of [3H]-9-cis-retinoic acid binding to human retinoid X receptor alpha ligand-binding domain expressed in E. coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Institute

Curated by ChEMBL
LigandPNGBDBM50151227(4-[(3-Butoxy-5,5,8,8-tetramethyl-5,6,7,8-tetrahydr...)
Affinity DataIC50:  270nMAssay Description:Inhibition of [3H]-9-cis-retinoic acid binding to human retinoid X receptor alpha ligand-binding domain expressed in E. coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Institute

Curated by ChEMBL
LigandPNGBDBM50151226(4-[(3-Butyl-5,5,8,8-tetramethyl-5,6,7,8-tetrahydro...)
Affinity DataIC50:  500nMAssay Description:Inhibition of [3H]-9-cis-retinoic acid binding to human retinoid X receptor alpha ligand-binding domain expressed in E. coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed