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Found 20 Enz. Inhib. hit(s) with all data for entry = 50037338
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
3-Dimensional Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50409948(CHEMBL363098)
Affinity DataIC50:  0.400nMAssay Description:In vitro inhibitory activity against alpha v beta 3 vitronectin protein interaction was measured by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
3-Dimensional Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50150956(CHEMBL186712 | Imidazolyl O-guanidinium analogue)
Affinity DataIC50:  3.40nMAssay Description:In vitro inhibitory activity against alpha v beta 3 vitronectin protein interaction was measured by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
3-Dimensional Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50150958(CHEMBL433785 | Imidazolyl O-guanidinium analogue)
Affinity DataIC50:  6.10nMAssay Description:In vitro inhibitory activity against alpha v beta 3 vitronectin protein interaction was measured by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
3-Dimensional Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50409947(CHEMBL359601)
Affinity DataIC50:  7.20nMAssay Description:In vitro inhibitory activity against alpha v beta 3 vitronectin protein interaction was measured by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
3-Dimensional Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50409940(CHEMBL185580)
Affinity DataIC50:  9nMAssay Description:In vitro inhibitory activity against alpha v beta 3 vitronectin protein interaction was measured by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
3-Dimensional Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50409942(CHEMBL183253)
Affinity DataIC50:  10.5nMAssay Description:In vitro inhibitory activity against alpha v beta 3 vitronectin protein interaction was measured by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
3-Dimensional Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50150956(CHEMBL186712 | Imidazolyl O-guanidinium analogue)
Affinity DataIC50:  13nMAssay Description:In vitro inhibitory activity against alpha IIb beta IIIa fibrinogen protein interaction was measured by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
3-Dimensional Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50409945(CHEMBL426254)
Affinity DataIC50: >20nMAssay Description:In vitro inhibitory activity against alpha v beta 3 vitronectin protein interaction was measured by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
3-Dimensional Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50150958(CHEMBL433785 | Imidazolyl O-guanidinium analogue)
Affinity DataIC50:  25nMAssay Description:In vitro inhibitory activity against alpha IIb beta IIIa fibrinogen protein interaction was measured by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
3-Dimensional Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50150957(2-Benzenesulfonylamino-3-[(5-{2-[N-(4,5-dihydro-1H...)
Affinity DataIC50:  100nMAssay Description:In vitro inhibitory activity against alpha v beta 3 vitronectin protein interaction was measured by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
3-Dimensional Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50409941(CHEMBL185374)
Affinity DataIC50:  130nMAssay Description:In vitro inhibitory activity against alpha v beta 3 vitronectin protein interaction was measured by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
3-Dimensional Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50150957(2-Benzenesulfonylamino-3-[(5-{2-[N-(4,5-dihydro-1H...)
Affinity DataIC50:  170nMAssay Description:In vitro inhibitory activity against alpha IIb beta IIIa fibrinogen protein interaction was measured by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
3-Dimensional Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50409949(CHEMBL185557)
Affinity DataIC50:  310nMAssay Description:In vitro inhibitory activity against alpha v beta 3 vitronectin protein interaction was measured by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
3-Dimensional Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50150958(CHEMBL433785 | Imidazolyl O-guanidinium analogue)
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity against alpha 5 beta 1 fibronectin protein interaction was measured by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
3-Dimensional Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50150956(CHEMBL186712 | Imidazolyl O-guanidinium analogue)
Affinity DataIC50:  1.00E+3nMAssay Description:In vitro inhibitory activity against alpha v beta 5 vitronectin protein interaction was measured by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
3-Dimensional Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50409946(CHEMBL184606)
Affinity DataIC50: >2.00E+4nMAssay Description:In vitro inhibitory activity against alpha v beta 3 vitronectin protein interaction was measured by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
3-Dimensional Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50409944(CHEMBL184638)
Affinity DataIC50: >2.00E+4nMAssay Description:In vitro inhibitory activity against alpha v beta 3 vitronectin protein interaction was measured by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
3-Dimensional Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50150957(2-Benzenesulfonylamino-3-[(5-{2-[N-(4,5-dihydro-1H...)
Affinity DataIC50: >2.00E+4nMAssay Description:In vitro inhibitory activity against alpha v beta 5 vitronectin protein interaction was measured by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
3-Dimensional Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50150957(2-Benzenesulfonylamino-3-[(5-{2-[N-(4,5-dihydro-1H...)
Affinity DataIC50: >2.00E+4nMAssay Description:In vitro inhibitory activity against alpha 5 beta 1 fibronectin protein interaction was measured by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
3-Dimensional Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50409943(CHEMBL367809)
Affinity DataIC50: >2.00E+4nMAssay Description:In vitro inhibitory activity against alpha v beta 3 vitronectin protein interaction was measured by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed