Compile Data Set for Download or QSAR
maximum 50k data
Found 33 Enz. Inhib. hit(s) with all data for entry = 50015299
TargetCathepsin K(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154167(CHEMBL185533 | [1-(1H-Pyrazol-3-ylaminooxalyl)-pen...)
Affinity DataIC50:  1.60nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154170(CHEMBL183788 | [1-(6-Chloro-1H-indazol-3-ylaminoox...)
Affinity DataIC50:  1.60nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154165(CHEMBL424982 | [1-(1H-Pyrazol-3-ylaminooxalyl)-pen...)
Affinity DataIC50:  1.80nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154148(CHEMBL363949 | [1-(1H-Pyrazol-3-ylaminooxalyl)-pen...)
Affinity DataIC50:  1.90nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154174(CHEMBL185090 | [1-(1-Methyl-1H-pyrazol-3-ylaminoox...)
Affinity DataIC50:  3.40nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154149(CHEMBL183632 | [1-(5-Phenyl-1H-pyrazol-3-ylaminoox...)
Affinity DataIC50:  6.20nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154149(CHEMBL183632 | [1-(5-Phenyl-1H-pyrazol-3-ylaminoox...)
Affinity DataIC50:  6.20nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154168(CHEMBL182516 | [1-(5-Phenyl-1H-pyrazol-3-ylaminoox...)
Affinity DataIC50:  10nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154173(CHEMBL360632 | [1-(1H-Pyrazol-3-ylaminooxalyl)-pen...)
Affinity DataIC50:  17nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154156(CHEMBL360863 | [1-(1H-Pyrazol-3-ylaminooxalyl)-pen...)
Affinity DataIC50:  18nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154155(CHEMBL184677 | [1-(Isoxazol-3-ylaminooxalyl)-penty...)
Affinity DataIC50:  20nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154171(CHEMBL184727 | [1-(5-Phenyl-1H-pyrazol-3-ylaminoox...)
Affinity DataIC50:  22nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154147(CHEMBL185211 | [1-(Isoxazol-3-ylaminooxalyl)-penty...)
Affinity DataIC50:  25nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154159(CHEMBL185245 | [1-(1-Phenyl-ethylaminooxalyl)-pent...)
Affinity DataIC50:  36nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154163(CHEMBL186353 | [1-(2-Cyclobutyl-2H-pyrazol-3-ylami...)
Affinity DataIC50:  45nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154160(CHEMBL361911 | [1-(2-Cyclopropylmethyl-2H-pyrazol-...)
Affinity DataIC50:  51nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154175(CHEMBL362393 | [1-(2-Ethyl-2H-pyrazol-3-ylaminooxa...)
Affinity DataIC50:  52nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154172(CHEMBL263181 | [1-(2-Isopropyl-2H-pyrazol-3-ylamin...)
Affinity DataIC50:  54nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154146(CHEMBL362292 | [1-(2-Cyclohexyl-2H-pyrazol-3-ylami...)
Affinity DataIC50:  58nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154169(CHEMBL186352 | [1-(2-Methyl-2H-pyrazol-3-ylaminoox...)
Affinity DataIC50:  62nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154176(CHEMBL183252 | [1-(2-Phenyl-2H-pyrazol-3-ylaminoox...)
Affinity DataIC50:  63nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154162(CHEMBL183959 | [1-(2-Benzyl-2H-pyrazol-3-ylaminoox...)
Affinity DataIC50:  65nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154164(CHEMBL183686 | [1-(1-Phenyl-ethylaminooxalyl)-pent...)
Affinity DataIC50:  68nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154157(CHEMBL359588 | [1-(1-Phenyl-ethylaminooxalyl)-pent...)
Affinity DataIC50:  68nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154150(CHEMBL363950 | {1-[2-(3,3-Dimethyl-butyl)-2H-pyraz...)
Affinity DataIC50:  71nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154151(CHEMBL185062 | [1-(1-Phenyl-ethylaminooxalyl)-pent...)
Affinity DataIC50:  71nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154153(CHEMBL185403 | [1-(2-Isobutyl-2H-pyrazol-3-ylamino...)
Affinity DataIC50:  76nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154152(CHEMBL184212 | [1-(2-Cyclopentyl-2H-pyrazol-3-ylam...)
Affinity DataIC50:  83nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154166(CHEMBL359773 | [1-(Isoxazol-3-ylaminooxalyl)-penty...)
Affinity DataIC50:  120nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154158(CHEMBL425535 | [1-(2-Methyl-2H-pyrazol-3-ylaminoox...)
Affinity DataIC50:  135nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154145(CHEMBL184331 | [1-(1-Phenyl-ethylaminooxalyl)-pent...)
Affinity DataIC50:  140nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154154(CHEMBL184883 | [1-(Isoxazol-3-ylaminooxalyl)-penty...)
Affinity DataIC50:  350nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154161(CHEMBL360630 | [1-(2-Methyl-2H-pyrazol-3-ylaminoox...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed