Compile Data Set for Download or QSAR
maximum 50k data
Found 95 Enz. Inhib. hit(s) with all data for entry = 50037481
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156056(CHEMBL188143 | [4-(4-Chloro-phenyl)-piperidin-3-yl...)
Affinity DataKi:  0.560nMAssay Description:Inhibition of high affinity uptake by the norepinephrine transporter from rat synaptosomal nerve endings by using [3H]NE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156052(2-[4-(4-Chloro-phenyl)-1-methyl-piperidin-3-ylmeth...)
Affinity DataKi:  0.680nMAssay Description:Inhibition of high affinity uptake by the norepinephrine transporter from rat synaptosomal nerve endings by using [3H]NE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156036(2-[4-(4-Chloro-phenyl)-1-methyl-piperidin-3-ylmeth...)
Affinity DataKi:  0.800nMAssay Description:Inhibition of high affinity uptake by the norepinephrine transporter from rat synaptosomal nerve endings by using [3H]NE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156042(2-[4-(4-Chloro-phenyl)-1-methyl-piperidin-3-ylmeth...)
Affinity DataKi:  0.940nMAssay Description:Inhibition of high affinity uptake by the norepinephrine transporter from rat synaptosomal nerve endings by using [3H]NE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156036(2-[4-(4-Chloro-phenyl)-1-methyl-piperidin-3-ylmeth...)
Affinity DataKi:  1nMAssay Description:Inhibition of high affinity uptake by the dopamine transporter from rat synaptosomal nerve endings by using [3H]DA as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156036(2-[4-(4-Chloro-phenyl)-1-methyl-piperidin-3-ylmeth...)
Affinity DataKi:  1.10nMAssay Description:Inhibition of high affinity uptake by the serotonin transporter (5-HT) from rat synaptosomal nerve endings by using [3H]5-HT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156037(Acetic acid 2-[4-(4-chloro-phenyl)-1-methyl-piperi...)
Affinity DataKi:  3.60nMAssay Description:Inhibition of high affinity uptake by the norepinephrine transporter from rat synaptosomal nerve endings by using [3H]NE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156032(Benzoic acid 2-[4-(4-chloro-phenyl)-1-methyl-piper...)
Affinity DataKi:  4.5nMAssay Description:Inhibition of high affinity uptake by the norepinephrine transporter from rat synaptosomal nerve endings by using [3H]NE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156052(2-[4-(4-Chloro-phenyl)-1-methyl-piperidin-3-ylmeth...)
Affinity DataKi:  4.5nMAssay Description:Inhibition of high affinity uptake by the serotonin transporter (5-HT) from rat synaptosomal nerve endings by using [3H]5-HT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156057(4-(4-Chloro-phenyl)-3-(2-methoxy-ethylsulfanylmeth...)
Affinity DataKi:  6nMAssay Description:Inhibition of high affinity uptake by the norepinephrine transporter from rat synaptosomal nerve endings by using [3H]NE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156032(Benzoic acid 2-[4-(4-chloro-phenyl)-1-methyl-piper...)
Affinity DataKi:  6.70nMAssay Description:Inhibition of high affinity uptake by the serotonin transporter (5-HT) from rat synaptosomal nerve endings by using [3H]5-HT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156031(Acetic acid 2-[4-(4-chloro-phenyl)-1-methyl-piperi...)
Affinity DataKi:  9nMAssay Description:Inhibition of high affinity uptake by the dopamine transporter from rat synaptosomal nerve endings by using [3H]DA as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156051(2-[4-(4-Chloro-phenyl)-piperidin-3-ylmethylsulfany...)
Affinity DataKi:  10nMAssay Description:Inhibition of high affinity uptake by the norepinephrine transporter from rat synaptosomal nerve endings by using [3H]NE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156054(2-[4-(4-Chloro-phenyl)-1-methyl-piperidin-3-ylmeth...)
Affinity DataKi:  12nMAssay Description:Inhibition of high affinity uptake by the norepinephrine transporter from rat synaptosomal nerve endings by using [3H]NE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156039(2-[4-(4-Chloro-phenyl)-1-methyl-piperidin-3-ylmeth...)
Affinity DataKi:  12nMAssay Description:Inhibition of high affinity uptake by the dopamine transporter from rat synaptosomal nerve endings by using [3H]DA as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156043(2-[4-(4-Chloro-phenyl)-1-methyl-piperidin-3-ylmeth...)
Affinity DataKi:  13nMAssay Description:Inhibition of high affinity uptake by the dopamine transporter from rat synaptosomal nerve endings by using [3H]DA as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156056(CHEMBL188143 | [4-(4-Chloro-phenyl)-piperidin-3-yl...)
Affinity DataKi:  13nMAssay Description:Inhibition of high affinity uptake by the serotonin transporter (5-HT) from rat synaptosomal nerve endings by using [3H]5-HT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156045(4-(4-Chloro-phenyl)-3-(2-methoxy-ethanesulfinylmet...)
Affinity DataKi:  15nMAssay Description:Inhibition of high affinity uptake by the dopamine transporter from rat synaptosomal nerve endings by using [3H]DA as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156053(2-[4-(4-Chloro-phenyl)-1-methyl-piperidin-3-ylmeth...)
Affinity DataKi:  15nMAssay Description:Inhibition of high affinity uptake by the norepinephrine transporter from rat synaptosomal nerve endings by using [3H]NE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156042(2-[4-(4-Chloro-phenyl)-1-methyl-piperidin-3-ylmeth...)
Affinity DataKi:  16nMAssay Description:Inhibition of high affinity uptake by the dopamine transporter from rat synaptosomal nerve endings by using [3H]DA as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156040(Benzoic acid 2-[4-(4-chloro-phenyl)-1-methyl-piper...)
Affinity DataKi:  18nMAssay Description:Inhibition of high affinity uptake by the norepinephrine transporter from rat synaptosomal nerve endings by using [3H]NE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156048(2-[4-(4-Chloro-phenyl)-1-methyl-piperidin-3-ylmeth...)
Affinity DataKi:  20nMAssay Description:Inhibition of high affinity uptake by the norepinephrine transporter from rat synaptosomal nerve endings by using [3H]NE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156045(4-(4-Chloro-phenyl)-3-(2-methoxy-ethanesulfinylmet...)
Affinity DataKi:  25nMAssay Description:Inhibition of high affinity uptake by the norepinephrine transporter from rat synaptosomal nerve endings by using [3H]NE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156043(2-[4-(4-Chloro-phenyl)-1-methyl-piperidin-3-ylmeth...)
Affinity DataKi:  25nMAssay Description:Inhibition of high affinity uptake by the norepinephrine transporter from rat synaptosomal nerve endings by using [3H]NE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156058(CHEMBL372709 | [4-(4-Chloro-phenyl)-1-methyl-piper...)
Affinity DataKi:  25nMAssay Description:Inhibition of high affinity uptake by the norepinephrine transporter from rat synaptosomal nerve endings by using [3H]NE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156034(2-[4-(4-Chloro-phenyl)-1-methyl-piperidin-3-ylmeth...)
Affinity DataKi:  27nMAssay Description:Inhibition of high affinity uptake by the norepinephrine transporter from rat synaptosomal nerve endings by using [3H]NE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156031(Acetic acid 2-[4-(4-chloro-phenyl)-1-methyl-piperi...)
Affinity DataKi:  29nMAssay Description:Inhibition of high affinity uptake by the norepinephrine transporter from rat synaptosomal nerve endings by using [3H]NE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156038(2-[4-(4-Chloro-phenyl)-piperidin-3-ylmethanesulfin...)
Affinity DataKi:  31nMAssay Description:Inhibition of high affinity uptake by the norepinephrine transporter from rat synaptosomal nerve endings by using [3H]NE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156040(Benzoic acid 2-[4-(4-chloro-phenyl)-1-methyl-piper...)
Affinity DataKi:  32nMAssay Description:Inhibition of high affinity uptake by the dopamine transporter from rat synaptosomal nerve endings by using [3H]DA as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156060(4-(4-Chloro-phenyl)-1-methyl-3-(3-methyl-[1,2,4]ox...)
Affinity DataKi:  32nMAssay Description:Inhibition of high affinity uptake by the norepinephrine transporter from rat synaptosomal nerve endings by using [3H]NE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156037(Acetic acid 2-[4-(4-chloro-phenyl)-1-methyl-piperi...)
Affinity DataKi:  35nMAssay Description:Inhibition of high affinity uptake by the dopamine transporter from rat synaptosomal nerve endings by using [3H]DA as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156047(2-[4-(4-Chloro-phenyl)-1-methyl-piperidin-3-ylmeth...)
Affinity DataKi:  39nMAssay Description:Inhibition of high affinity uptake by the norepinephrine transporter from rat synaptosomal nerve endings by using [3H]NE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156039(2-[4-(4-Chloro-phenyl)-1-methyl-piperidin-3-ylmeth...)
Affinity DataKi:  42nMAssay Description:Inhibition of high affinity uptake by the norepinephrine transporter from rat synaptosomal nerve endings by using [3H]NE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156057(4-(4-Chloro-phenyl)-3-(2-methoxy-ethylsulfanylmeth...)
Affinity DataKi:  50nMAssay Description:Inhibition of high affinity uptake by the dopamine transporter from rat synaptosomal nerve endings by using [3H]DA as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156056(CHEMBL188143 | [4-(4-Chloro-phenyl)-piperidin-3-yl...)
Affinity DataKi:  51nMAssay Description:Inhibition of high affinity uptake by the dopamine transporter from rat synaptosomal nerve endings by using [3H]DA as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156041(CHEMBL188276 | [4-(4-Chloro-phenyl)-1-methyl-piper...)
Affinity DataKi:  53nMAssay Description:Inhibition of high affinity uptake by the norepinephrine transporter from rat synaptosomal nerve endings by using [3H]NE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156054(2-[4-(4-Chloro-phenyl)-1-methyl-piperidin-3-ylmeth...)
Affinity DataKi:  55nMAssay Description:Inhibition of high affinity uptake by the dopamine transporter from rat synaptosomal nerve endings by using [3H]DA as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156037(Acetic acid 2-[4-(4-chloro-phenyl)-1-methyl-piperi...)
Affinity DataKi:  57nMAssay Description:Inhibition of high affinity uptake by the serotonin transporter (5-HT) from rat synaptosomal nerve endings by using [3H]5-HT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156032(Benzoic acid 2-[4-(4-chloro-phenyl)-1-methyl-piper...)
Affinity DataKi:  68nMAssay Description:Inhibition of high affinity uptake by the dopamine transporter from rat synaptosomal nerve endings by using [3H]DA as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156058(CHEMBL372709 | [4-(4-Chloro-phenyl)-1-methyl-piper...)
Affinity DataKi:  80nMAssay Description:Inhibition of high affinity uptake by the dopamine transporter from rat synaptosomal nerve endings by using [3H]DA as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156052(2-[4-(4-Chloro-phenyl)-1-methyl-piperidin-3-ylmeth...)
Affinity DataKi:  83nMAssay Description:Inhibition of high affinity uptake by the dopamine transporter from rat synaptosomal nerve endings by using [3H]DA as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156053(2-[4-(4-Chloro-phenyl)-1-methyl-piperidin-3-ylmeth...)
Affinity DataKi:  85nMAssay Description:Inhibition of high affinity uptake by the dopamine transporter from rat synaptosomal nerve endings by using [3H]DA as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156049(2-[4-(4-Chloro-phenyl)-1-methyl-piperidin-3-ylmeth...)
Affinity DataKi:  86nMAssay Description:Inhibition of high affinity uptake by the norepinephrine transporter from rat synaptosomal nerve endings by using [3H]NE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156031(Acetic acid 2-[4-(4-chloro-phenyl)-1-methyl-piperi...)
Affinity DataKi:  87nMAssay Description:Inhibition of high affinity uptake by the serotonin transporter (5-HT) from rat synaptosomal nerve endings by using [3H]5-HT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156034(2-[4-(4-Chloro-phenyl)-1-methyl-piperidin-3-ylmeth...)
Affinity DataKi:  88nMAssay Description:Inhibition of high affinity uptake by the serotonin transporter (5-HT) from rat synaptosomal nerve endings by using [3H]5-HT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156038(2-[4-(4-Chloro-phenyl)-piperidin-3-ylmethanesulfin...)
Affinity DataKi:  108nMAssay Description:Inhibition of high affinity uptake by the dopamine transporter from rat synaptosomal nerve endings by using [3H]DA as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50084717((+)-(1R,2R,3S,5S)-methyl 3-(benzoyloxy)-8-methyl-8...)
Affinity DataKi:  108nMAssay Description:Inhibition of high affinity uptake by the norepinephrine transporter from rat synaptosomal nerve endings by using [3H]NE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156043(2-[4-(4-Chloro-phenyl)-1-methyl-piperidin-3-ylmeth...)
Affinity DataKi:  110nMAssay Description:Inhibition of high affinity uptake by the serotonin transporter (5-HT) from rat synaptosomal nerve endings by using [3H]5-HT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156051(2-[4-(4-Chloro-phenyl)-piperidin-3-ylmethylsulfany...)
Affinity DataKi:  114nMAssay Description:Inhibition of high affinity uptake by the dopamine transporter from rat synaptosomal nerve endings by using [3H]DA as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50156034(2-[4-(4-Chloro-phenyl)-1-methyl-piperidin-3-ylmeth...)
Affinity DataKi:  116nMAssay Description:Inhibition of high affinity uptake by the dopamine transporter from rat synaptosomal nerve endings by using [3H]DA as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 95 total ) | Next | Last >>
Jump to: