Compile Data Set for Download or QSAR
maximum 50k data
Found 9 Enz. Inhib. hit(s) with all data for entry = 50037486
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50156214(2-(3,4-Dimethoxy-phenyl)-2-isopropyl-5-[4-(2-pheno...)
Affinity DataIC50:  400nMAssay Description:In vitro antagonism of N-type calcium channels expressed in PC12 cells was determined as the increase in intracellular calcium influx in the presence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50156213(CHEMBL439485 | omega-Conotoxin)
Affinity DataIC50:  500nMAssay Description:In vitro antagonism of N-type calcium channels expressed in PC12 cells was determined as the increase in intracellular calcium influx in the presence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50156213(CHEMBL439485 | omega-Conotoxin)
Affinity DataIC50:  600nMAssay Description:In vitro antagonism of N-type calcium channels expressed in PC12 cells was determined as the increase in intracellular calcium influxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50156214(2-(3,4-Dimethoxy-phenyl)-2-isopropyl-5-[4-(2-pheno...)
Affinity DataIC50:  700nMAssay Description:In vitro antagonism of N-type calcium channels expressed in PC12 cells was determined as the increase in intracellular calcium influxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50156215(1-(4-Amino-piperidin-1-yl)-4,4-bis-(4-fluoro-pheny...)
Affinity DataIC50:  1.03E+3nMAssay Description:In vitro antagonism of N-type calcium channels expressed in PC12 cells was determined as the increase in intracellular calcium influxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50156215(1-(4-Amino-piperidin-1-yl)-4,4-bis-(4-fluoro-pheny...)
Affinity DataIC50:  2.40E+3nMAssay Description:In vitro antagonism of N-type calcium channels expressed in PC12 cells was determined as the increase in intracellular calcium influx in the presence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50156216(4-Methyl-2-methylamino-pentanoic acid {1-[4,4-bis-...)
Affinity DataIC50:  3.00E+3nMAssay Description:In vitro antagonism of N-type calcium channels expressed in PC12 cells was determined as the increase in intracellular calcium influxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50156212(2-(3,4-Dimethoxy-phenyl)-2-isopropyl-5-[1-(2-pheno...)
Affinity DataIC50:  3.10E+3nMAssay Description:In vitro antagonism of N-type calcium channels expressed in PC12 cells was determined as the increase in intracellular calcium influx in the presence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50156212(2-(3,4-Dimethoxy-phenyl)-2-isopropyl-5-[1-(2-pheno...)
Affinity DataIC50:  3.80E+3nMAssay Description:In vitro antagonism of N-type calcium channels expressed in PC12 cells was determined as the increase in intracellular calcium influxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed