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Found 11 Enz. Inhib. hit(s) with all data for entry = 50015483
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
Department Of Life Science And National Research Laboratory Of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50062351((R)-N*4*-Hydroxy-N*1*-[(S)-2-(1H-indol-3-yl)-1-met...)
Affinity DataIC50:  1nMAssay Description:In vitro inhibition of A disintegrin and metalloproteinase domain 9 (ADAM9)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 12(Homo sapiens (Human))
Department Of Life Science And National Research Laboratory Of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50062351((R)-N*4*-Hydroxy-N*1*-[(S)-2-(1H-indol-3-yl)-1-met...)
Affinity DataIC50:  5.93nMAssay Description:Inhibition of A disintegrin and metalloproteinase domain 12 (ADAM12) binding in cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Department Of Life Science And National Research Laboratory Of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50062351((R)-N*4*-Hydroxy-N*1*-[(S)-2-(1H-indol-3-yl)-1-met...)
Affinity DataIC50:  7.5nMAssay Description:In vitro inhibition of A disintegrin and metalloproteinase domain 17 (ADAM17, TACE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 10(Homo sapiens (Human))
Department Of Life Science And National Research Laboratory Of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50062351((R)-N*4*-Hydroxy-N*1*-[(S)-2-(1H-indol-3-yl)-1-met...)
Affinity DataIC50:  8.10nMAssay Description:In vitro inhibition of A disintegrin and metalloproteinase domain 10 (ADAM10)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 12(Homo sapiens (Human))
Department Of Life Science And National Research Laboratory Of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50156477(CHEMBL366034 | {3-(3-Bromo-phenyl)-2-[(furan-2-car...)
Affinity DataIC50:  16.7nMAssay Description:Inhibition of A disintegrin and metalloproteinase domain 12 (ADAM12) binding in cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 12(Homo sapiens (Human))
Department Of Life Science And National Research Laboratory Of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50156475(2-[2-[(5-Bromo-furan-2-carbonyl)-amino]-3-(4-bromo...)
Affinity DataIC50:  24.8nMAssay Description:Inhibition of A disintegrin and metalloproteinase domain 12 (ADAM12) binding in cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 12(Homo sapiens (Human))
Department Of Life Science And National Research Laboratory Of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50156476(2-[2-Benzoylamino-3-(2-fluoro-phenyl)-acryloylamin...)
Affinity DataIC50:  40.5nMAssay Description:Inhibition of A disintegrin and metalloproteinase domain 12 (ADAM12) binding in cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 12(Homo sapiens (Human))
Department Of Life Science And National Research Laboratory Of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50156478(2-{2-[(Furan-2-carbonyl)-amino]-3-furan-2-yl-acryl...)
Affinity DataIC50:  42.3nMAssay Description:Inhibition of A disintegrin and metalloproteinase domain 12 (ADAM12) binding in cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 10(Homo sapiens (Human))
Department Of Life Science And National Research Laboratory Of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50156477(CHEMBL366034 | {3-(3-Bromo-phenyl)-2-[(furan-2-car...)
Affinity DataIC50: >1.05E+4nMAssay Description:In vitro inhibition of A disintegrin and metalloproteinase domain 10 (ADAM10)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 10(Homo sapiens (Human))
Department Of Life Science And National Research Laboratory Of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50156478(2-{2-[(Furan-2-carbonyl)-amino]-3-furan-2-yl-acryl...)
Affinity DataIC50:  1.05E+4nMAssay Description:In vitro inhibition of A disintegrin and metalloproteinase domain 10 (ADAM10)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 10(Homo sapiens (Human))
Department Of Life Science And National Research Laboratory Of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50156476(2-[2-Benzoylamino-3-(2-fluoro-phenyl)-acryloylamin...)
Affinity DataIC50: >1.05E+4nMAssay Description:In vitro inhibition of A disintegrin and metalloproteinase domain 10 (ADAM10)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed