TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
University Of Newcastle
Curated by ChEMBL
University Of Newcastle
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against DNA-dependent protein kinase (DNA-PK)More data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
University Of Newcastle
Curated by ChEMBL
University Of Newcastle
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against DNA-dependent protein kinase (DNA-PK) at 0.5 uMMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
University Of Newcastle
Curated by ChEMBL
University Of Newcastle
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibitory activity against DNA-dependent protein kinase (DNA-PK) at 0.5 uMMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
University Of Newcastle
Curated by ChEMBL
University Of Newcastle
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Inhibitory activity against DNA-dependent protein kinase (DNA-PK) at 0.5 uMMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
University Of Newcastle
Curated by ChEMBL
University Of Newcastle
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Inhibitory activity against DNA-dependent protein kinase (DNA-PK)More data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
University Of Newcastle
Curated by ChEMBL
University Of Newcastle
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibitory activity against DNA-dependent protein kinase (DNA-PK) at 0.5 uMMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
University Of Newcastle
Curated by ChEMBL
University Of Newcastle
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Inhibitory activity against DNA-dependent protein kinase (DNA-PK) at 0.5 uMMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
University Of Newcastle
Curated by ChEMBL
University Of Newcastle
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Inhibitory activity against DNA-dependent protein kinase (DNA-PK) at 0.5 uMMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
University Of Newcastle
Curated by ChEMBL
University Of Newcastle
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibitory activity against DNA-dependent protein kinase (DNA-PK) at 0.5 uMMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
University Of Newcastle
Curated by ChEMBL
University Of Newcastle
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibitory activity against DNA-dependent protein kinase (DNA-PK) at 0.5 uMMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
University Of Newcastle
Curated by ChEMBL
University Of Newcastle
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:Inhibitory activity against DNA-dependent protein kinase (DNA-PK) at 0.5 uMMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
University Of Newcastle
Curated by ChEMBL
University Of Newcastle
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibitory activity against DNA-dependent protein kinase (DNA-PK)More data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
University Of Newcastle
Curated by ChEMBL
University Of Newcastle
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibitory activity against DNA-dependent protein kinase (DNA-PK) at 0.5 uMMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
University Of Newcastle
Curated by ChEMBL
University Of Newcastle
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of Mammalian target of Rapamycin mTORMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
University Of Newcastle
Curated by ChEMBL
University Of Newcastle
Curated by ChEMBL
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of Phosphatidylinositol 3-kinase p110 alpha subunitMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
University Of Newcastle
Curated by ChEMBL
University Of Newcastle
Curated by ChEMBL
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of Mammalian target of Rapamycin mTORMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
University Of Newcastle
Curated by ChEMBL
University Of Newcastle
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of Phosphatidylinositol 3-kinase p110 alpha subunitMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
University Of Newcastle
Curated by ChEMBL
University Of Newcastle
Curated by ChEMBL
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibition of Mammalian target of Rapamycin mTORMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
University Of Newcastle
Curated by ChEMBL
University Of Newcastle
Curated by ChEMBL
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of Phosphatidylinositol 3-kinase p110 alpha subunitMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Mutated in ataxia telangiectasia protein ATM kinaseMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ATR(Homo sapiens (Human))
University Of Newcastle
Curated by ChEMBL
University Of Newcastle
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Ataxia telangiectasia related protein ATR kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Mutated in ataxia telangiectasia protein ATM kinaseMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ATR(Homo sapiens (Human))
University Of Newcastle
Curated by ChEMBL
University Of Newcastle
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Ataxia telangiectasia related protein ATR kinaseMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ATR(Homo sapiens (Human))
University Of Newcastle
Curated by ChEMBL
University Of Newcastle
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Ataxia telangiectasia related protein ATR kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Mutated in ataxia telangiectasia protein ATM kinaseMore data for this Ligand-Target Pair