Compile Data Set for Download or QSAR
maximum 50k data
Found 59 Enz. Inhib. hit(s) with all data for entry = 851
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6683(aminoimidazo[1,2-a]pyridine deriv. 18 | {2-amino-6...)
Affinity DataIC50:  26nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6684(aminoimidazo[1,2-a]pyridine deriv. 20 | {2-amino-6...)
Affinity DataIC50:  29nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6687(6-[(2-chloro-6-fluorophenyl)carbonyl]-3-[(2,6-difl...)
Affinity DataIC50:  33nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6686(4-({2-amino-6-[(2,6-dichlorophenyl)carbonyl]imidaz...)
Affinity DataIC50:  46nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6702(4-({2-amino-6-[(2,6-dichlorophenyl)carbonyl]imidaz...)
Affinity DataIC50:  52nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6689((2E)-3-{2-amino-3-[(2,6-difluorophenyl)carbonyl]im...)
Affinity DataIC50:  53nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6697(6-[(2,6-dichlorophenyl)carbonyl]-3-[(2,6-difluorop...)
Affinity DataIC50:  53nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6677(3,6-bis[(2,6-difluorophenyl)carbonyl]imidazo[1,2-a...)
Affinity DataIC50:  57nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6688(3-[(2,6-difluorophenyl)carbonyl]-6-[1-(2,6-difluor...)
Affinity DataIC50:  63nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6680(6-[(2,6-difluorophenyl)carbonyl]-3-[(2-methoxyphen...)
Affinity DataIC50:  68nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6679(3-[(2,6-difluoro-4-methoxyphenyl)carbonyl]-6-[(2,6...)
Affinity DataIC50:  91nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6688(3-[(2,6-difluorophenyl)carbonyl]-6-[1-(2,6-difluor...)
Affinity DataIC50:  93nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6685(4-({2-amino-6-[(2,6-dichlorophenyl)carbonyl]imidaz...)
Affinity DataIC50:  95nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6690(6-[(Z)-1-(2,6-difluorophenyl)-2-(1H-1,2,3,4-tetraz...)
Affinity DataIC50:  96nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6678(3-[(2-chloro-6-fluorophenyl)carbonyl]-6-[(2,6-difl...)
Affinity DataIC50:  102nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6687(6-[(2-chloro-6-fluorophenyl)carbonyl]-3-[(2,6-difl...)
Affinity DataIC50:  104nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6683(aminoimidazo[1,2-a]pyridine deriv. 18 | {2-amino-6...)
Affinity DataIC50:  105nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6681(3-[(2,6-dichlorophenyl)carbonyl]-6-[(2,6-difluorop...)
Affinity DataIC50:  121nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6677(3,6-bis[(2,6-difluorophenyl)carbonyl]imidazo[1,2-a...)
Affinity DataIC50:  122nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6679(3-[(2,6-difluoro-4-methoxyphenyl)carbonyl]-6-[(2,6...)
Affinity DataIC50:  132nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6684(aminoimidazo[1,2-a]pyridine deriv. 20 | {2-amino-6...)
Affinity DataIC50:  143nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6686(4-({2-amino-6-[(2,6-dichlorophenyl)carbonyl]imidaz...)
Affinity DataIC50:  154nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6689((2E)-3-{2-amino-3-[(2,6-difluorophenyl)carbonyl]im...)
Affinity DataIC50:  160nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6682(aminoimidazo[1,2-a]pyridine deriv. 17 | {2-amino-6...)
Affinity DataIC50:  165nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6681(3-[(2,6-dichlorophenyl)carbonyl]-6-[(2,6-difluorop...)
Affinity DataIC50:  209nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6682(aminoimidazo[1,2-a]pyridine deriv. 17 | {2-amino-6...)
Affinity DataIC50:  214nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6678(3-[(2-chloro-6-fluorophenyl)carbonyl]-6-[(2,6-difl...)
Affinity DataIC50:  239nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6676(3-benzoyl-6-[(2,6-difluorophenyl)carbonyl]imidazo[...)
Affinity DataIC50:  324nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6676(3-benzoyl-6-[(2,6-difluorophenyl)carbonyl]imidazo[...)
Affinity DataIC50:  326nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6685(4-({2-amino-6-[(2,6-dichlorophenyl)carbonyl]imidaz...)
Affinity DataIC50:  328nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6681(3-[(2,6-dichlorophenyl)carbonyl]-6-[(2,6-difluorop...)
Affinity DataIC50:  359nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6692(6-[(2-chlorophenyl)carbonyl]-3-[(2,6-difluoropheny...)
Affinity DataIC50:  428nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6684(aminoimidazo[1,2-a]pyridine deriv. 20 | {2-amino-6...)
Affinity DataIC50:  464nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6680(6-[(2,6-difluorophenyl)carbonyl]-3-[(2-methoxyphen...)
Affinity DataIC50:  475nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6699(6-[(2,6-difluorophenyl)carbonyl]-3-(thiophen-2-ylc...)
Affinity DataIC50:  547nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6695(3-[(2,6-difluorophenyl)carbonyl]-6-[(2-methoxyphen...)
Affinity DataIC50:  603nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6683(aminoimidazo[1,2-a]pyridine deriv. 18 | {2-amino-6...)
Affinity DataIC50:  786nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6687(6-[(2-chloro-6-fluorophenyl)carbonyl]-3-[(2,6-difl...)
Affinity DataIC50:  810nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6704(6-[(2,6-dichlorophenyl)carbonyl]-3-({2,6-difluoro-...)
Affinity DataIC50:  812nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6678(3-[(2-chloro-6-fluorophenyl)carbonyl]-6-[(2,6-difl...)
Affinity DataIC50:  827nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6679(3-[(2,6-difluoro-4-methoxyphenyl)carbonyl]-6-[(2,6...)
Affinity DataIC50:  838nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6705((2Z)-3-{2-amino-3-[(2,6-difluorophenyl)carbonyl]im...)
Affinity DataIC50:  896nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6703(6-[(2,6-dichlorophenyl)carbonyl]-3-({4-[2-(diethyl...)
Affinity DataIC50:  984nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6688(3-[(2,6-difluorophenyl)carbonyl]-6-[1-(2,6-difluor...)
Affinity DataIC50:  1.03E+3nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6693(3-[(2,6-difluorophenyl)carbonyl]-6-{[2-(trifluorom...)
Affinity DataIC50:  1.07E+3nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6677(3,6-bis[(2,6-difluorophenyl)carbonyl]imidazo[1,2-a...)
Affinity DataIC50:  1.08E+3nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6686(4-({2-amino-6-[(2,6-dichlorophenyl)carbonyl]imidaz...)
Affinity DataIC50:  1.14E+3nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6694(3-[(2,6-difluorophenyl)carbonyl]-6-[(2-methylpheny...)
Affinity DataIC50:  1.29E+3nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6689((2E)-3-{2-amino-3-[(2,6-difluorophenyl)carbonyl]im...)
Affinity DataIC50:  1.55E+3nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6690(6-[(Z)-1-(2,6-difluorophenyl)-2-(1H-1,2,3,4-tetraz...)
Affinity DataIC50:  1.69E+3nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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