Affinity DataIC50: 7nMAssay Description:Concentration for 50% inhibition of human melanocortin-4 receptor expressed in CHO cells using [125I]NDP-alpha-MSH as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Concentration for 50% inhibition of human melanocortin-4 receptor expressed in CHO cells using [125I]NDP-alpha-MSH as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Concentration for 50% inhibition of human melanocortin-4 receptor expressed in CHO cells using [125I]NDP-alpha-MSH as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Concentration for 50% inhibition of human melanocortin-4 receptor expressed in CHO cells using [125I]NDP-alpha-MSH as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Concentration for 50% inhibition of human melanocortin-4 receptor expressed in CHO cells using [125I]NDP-alpha-MSH as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Concentration for 50% inhibition of human melanocortin-4 receptor expressed in CHO cells using [125I]NDP-alpha-MSH as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Concentration for 50% inhibition of human melanocortin-4 receptor expressed in CHO cells using [125I]NDP-alpha-MSH as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Concentration for 50% inhibition of human melanocortin-4 receptor expressed in CHO cells using [125I]NDP-alpha-MSH as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 52nMAssay Description:Concentration for 50% inhibition of human melanocortin-4 receptor expressed in CHO cells using [125I]NDP-alpha-MSH as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 87nMAssay Description:Concentration for 50% inhibition of human melanocortin-4 receptor expressed in CHO cells using [125I]NDP-alpha-MSH as radioligandMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Concentration for 50% inhibition of human melanocortin-1 receptor expressed in CHO cells using [125I]-NDP-alpha-MSH as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30E+3nMAssay Description:Concentration for 50% inhibition of human melanocortin-3 receptor expressed in CHO cells using [125I]NDP-alpha-MSH as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+3nMAssay Description:Concentration for 50% inhibition of human melanocortin-5 receptor expressed in CHO cells using [125I]NDP-alpha-MSH as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+3nMAssay Description:Concentration for 50% inhibition of human melanocortin-5 receptor expressed in CHO cells using [125I]NDP-alpha-MSH as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 6.50E+3nMAssay Description:Concentration for 50% inhibition of human melanocortin-4 receptor expressed in CHO cells using [125I]NDP-alpha-MSH as radioligandMore data for this Ligand-Target Pair
Affinity DataEC50: 990nMAssay Description:Effective concentration towards human melanocortin-3 receptor mediated cAMP accumulation in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 11nMAssay Description:Effective concentration towards human melanocortin-4 receptor mediated cAMP accumulation in CHO cellsMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: 350nMAssay Description:Effective concentration towards human melanocortin-1 receptor mediated cAMP accumulation in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.80E+3nMAssay Description:Effective concentration towards human melanocortin-5 receptor mediated cAMP accumulation in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 2.90E+3nMAssay Description:Effective concentration towards human melanocortin-3 receptor mediated cAMP accumulation in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 29nMAssay Description:Effective concentration towards human melanocortin-4 receptor mediated cAMP accumulation in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 13nMAssay Description:Effective concentration towards human melanocortin-4 receptor mediated cAMP accumulation in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.90E+3nMAssay Description:Effective concentration towards human melanocortin-5 receptor mediated cAMP accumulation in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.90nMAssay Description:Effective concentration towards human melanocortin-4 receptor mediated cAMP accumulation in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 3.30E+3nMAssay Description:Effective concentration towards human melanocortin-5 receptor mediated cAMP accumulation in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 82nMAssay Description:Effective concentration towards human melanocortin-4 receptor mediated cAMP accumulation in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 2.70E+3nMAssay Description:Effective concentration towards human melanocortin-5 receptor mediated cAMP accumulation in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 52nMAssay Description:Effective concentration towards human melanocortin-4 receptor mediated cAMP accumulation in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 52nMAssay Description:Effective concentration towards human melanocortin-4 receptor mediated cAMP accumulation in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 34nMAssay Description:Effective concentration towards human melanocortin-4 receptor mediated cAMP accumulation in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 270nMAssay Description:Effective concentration towards human melanocortin-4 receptor mediated cAMP accumulation in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 510nMAssay Description:Effective concentration towards human melanocortin-5 receptor mediated cAMP accumulation in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 17nMAssay Description:Effective concentration towards human melanocortin-5 receptor mediated cAMP accumulation in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.10nMAssay Description:Effective concentration towards human melanocortin-3 receptor mediated cAMP accumulation in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 340nMAssay Description:Effective concentration towards human melanocortin-5 receptor mediated cAMP accumulation in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 840nMAssay Description:Effective concentration towards human melanocortin-5 receptor mediated cAMP accumulation in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 2.00E+3nMAssay Description:Effective concentration towards human melanocortin-5 receptor mediated cAMP accumulation in CHO cellsMore data for this Ligand-Target Pair