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Found 62 Enz. Inhib. hit(s) with all data for entry = 50015592
LigandPNGBDBM50157959(5-Chloro-thiophene-2-sulfonic acid [5-((E)-3-morph...)
Affinity DataIC50:  1nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158012(CHEMBL183351 | N-[13-(5-Chloro-thiophene-2-sulfony...)
Affinity DataIC50:  5nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157998(5-Chloro-thiophene-2-sulfonic acid [5-(2-morpholin...)
Affinity DataIC50:  5nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157959(5-Chloro-thiophene-2-sulfonic acid [5-((E)-3-morph...)
Affinity DataIC50:  5nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157959(5-Chloro-thiophene-2-sulfonic acid [5-((E)-3-morph...)
Affinity DataIC50:  5nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158017(CHEMBL180384 | N-[13-(5-Chloro-thiophene-2-sulfony...)
Affinity DataIC50:  6nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158000(CHEMBL183774 | N-[13-(5-Chloro-thiophene-2-sulfony...)
Affinity DataIC50:  7nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157983(CHEMBL183558 | N-[13-(5-Chloro-thiophene-2-sulfony...)
Affinity DataIC50:  7nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157994(CHEMBL183764 | Pyridine-2-carboxylic acid [13-(5-c...)
Affinity DataIC50:  12nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158009(5-Chloro-thiophene-2-sulfonic acid [5-((E)-3-imida...)
Affinity DataIC50:  15nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158018((13-Benzenesulfonylamino-tricyclo[8.2.1.0*3,8*]tri...)
Affinity DataIC50:  16nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157975(5-Chloro-thiophene-2-sulfonic acid {5-[(E)-3-(4-ph...)
Affinity DataIC50:  21nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157966(CHEMBL180784 | [13-(5-Chloro-thiophene-2-sulfonyla...)
Affinity DataIC50:  23nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158010(5-Chloro-thiophene-2-sulfonic acid (5-fluoro-tricy...)
Affinity DataIC50:  29nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157965(5-Chloro-thiophene-2-sulfonic acid (4-fluoro-tricy...)
Affinity DataIC50:  34nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158008(5-Chloro-thiophene-2-sulfonic acid {5-[(E)-3-(4-me...)
Affinity DataIC50:  39nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157984(CHEMBL182349 | N-[13-(5-Chloro-thiophene-2-sulfony...)
Affinity DataIC50:  41nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157977(CHEMBL183654 | Thiophene-2-sulfonic acid tricyclo[...)
Affinity DataIC50:  50nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157973(5-chloro-thiophene-2-sulfonic acid tricyclo[8.2.1....)
Affinity DataIC50:  62nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157960(CHEMBL362644 | N-[13-(5-Chloro-thiophene-2-sulfony...)
Affinity DataIC50:  69nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157991(CHEMBL183449 | N-(5-Fluoro-tricyclo[8.2.1.0*3,8*]t...)
Affinity DataIC50:  70nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158003(5-Chloro-thiophene-2-sulfonic acid [5-(2-piperidin...)
Affinity DataIC50:  73nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158007((13-Benzenesulfonylamino-tricyclo[8.2.1.0*3,8*]tri...)
Affinity DataIC50:  74nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157972(CHEMBL183585 | Pyridine-2-carboxylic acid (13-benz...)
Affinity DataIC50:  75nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157978(4-Fluoro-N-tricyclo[8.2.1.0*3,8*]trideca-3(8),4,6-...)
Affinity DataIC50:  129nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157988(5-Chloro-thiophene-2-sulfonic acid (5-chloro-tricy...)
Affinity DataIC50:  146nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158016(5-Chloro-thiophene-2-sulfonic acid [5-((E)-3-piper...)
Affinity DataIC50:  152nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157968((13-Benzenesulfonylamino-tricyclo[8.2.1.0*3,8*]tri...)
Affinity DataIC50:  153nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157995(5-Chloro-thiophene-2-sulfonic acid (4-chloro-tricy...)
Affinity DataIC50:  175nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158004(CHEMBL183326 | N-Tricyclo[8.2.1.0*3,8*]trideca-3(8...)
Affinity DataIC50:  190nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157969(5-Chloro-thiophene-2-sulfonic acid {5-[2-(3-hydrox...)
Affinity DataIC50:  209nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158002(2-(Benzyl-methyl-amino)-N-[13-(5-chloro-thiophene-...)
Affinity DataIC50:  226nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157963(5-Chloro-thiophene-2-sulfonic acid {5-[2-(2-methyl...)
Affinity DataIC50:  227nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157967(2-Fluoro-N-tricyclo[8.2.1.0*3,8*]trideca-3(8),4,6-...)
Affinity DataIC50:  239nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157976(5-Chloro-thiophene-2-sulfonic acid (5-hydroxy-tric...)
Affinity DataIC50:  269nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157964(3-Fluoro-N-tricyclo[8.2.1.0*3,8*]trideca-3(8),4,6-...)
Affinity DataIC50:  324nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157981(5-Chloro-thiophene-2-sulfonic acid {5-[2-(2-methyl...)
Affinity DataIC50:  335nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157970((13-Benzenesulfonylamino-tricyclo[8.2.1.0*3,8*]tri...)
Affinity DataIC50:  412nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157979(4-Chloro-N-tricyclo[8.2.1.0*3,8*]trideca-3(8),4,6-...)
Affinity DataIC50:  467nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158006(5-Chloro-thiophene-2-sulfonic acid (5-methoxy-tric...)
Affinity DataIC50:  490nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158014(5-Methyl-hexanoic acid (13-benzenesulfonylamino-tr...)
Affinity DataIC50:  535nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157997(Butane-1-sulfonic acid tricyclo[8.2.1.0*3,8*]tride...)
Affinity DataIC50:  610nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157989(5-Chloro-thiophene-2-sulfonic acid {5-[2-(4-hydrox...)
Affinity DataIC50:  623nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157999(4-Methyl-N-tricyclo[8.2.1.0*3,8*]trideca-3(8),4,6-...)
Affinity DataIC50:  651nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157986(CHEMBL360239 | Propane-1-sulfonic acid tricyclo[8....)
Affinity DataIC50:  721nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157987(CHEMBL181152 | N-(13-Benzenesulfonylamino-tricyclo...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157985(4-tert-Butyl-N-tricyclo[8.2.1.0*3,8*]trideca-3(8),...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158011(CHEMBL183165 | N-(13-Benzenesulfonylamino-tricyclo...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50158001(CHEMBL361113 | Ethanesulfonic acid tricyclo[8.2.1....)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50157996(4-Ethyl-N-tricyclo[8.2.1.0*3,8*]trideca-3(8),4,6-t...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory concentration against Gamma-secretase in whole cell inhibition assay using SH-SY5Y cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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