Compile Data Set for Download or QSAR
maximum 50k data
Found 5 Enz. Inhib. hit(s) with all data for entry = 50015659
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50069792((2S)-2-[(2S)-2-acetamido-4-methylpentanamido]-N-[(...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory concentration against Calpain I activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50159158(CHEMBL433563 | Peptidyl boronic acid derivative)
Affinity DataIC50: >1.00E+6nMAssay Description:In vitro inhibitory activity against Factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50159158(CHEMBL433563 | Peptidyl boronic acid derivative)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory concentration against Calpain I activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50159149(CHEMBL179042 | Peptidyl boronic acid derivative)
Affinity DataIC50: >1.00E+6nMAssay Description:In vitro inhibitory activity against Factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50159149(CHEMBL179042 | Peptidyl boronic acid derivative)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory concentration against Calpain I activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed