Compile Data Set for Download or QSAR
maximum 50k data
Found 44 Enz. Inhib. hit(s) with all data for entry = 50015731
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160488(1-Benzyl-2-(2-pyridin-3-yl-ethylsulfanyl)-1H-benzo...)
Affinity DataIC50:  120nMAssay Description:Inhibitory concentration towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160488(1-Benzyl-2-(2-pyridin-3-yl-ethylsulfanyl)-1H-benzo...)
Affinity DataIC50:  140nMAssay Description:Inhibitory concentration towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160501(1-Benzyl-2-(2-morpholin-4-yl-ethylsulfanyl)-1H-ben...)
Affinity DataIC50:  160nMAssay Description:Inhibitory concentration towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160501(1-Benzyl-2-(2-morpholin-4-yl-ethylsulfanyl)-1H-ben...)
Affinity DataIC50:  170nMAssay Description:Inhibitory concentration towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160496(1-Benzyl-2-ethylsulfanyl-1H-benzoimidazole-5-sulfo...)
Affinity DataIC50:  200nMAssay Description:Inhibitory concentration towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160483(1-Benzyl-2-methylsulfanyl-1H-benzoimidazole-5-sulf...)
Affinity DataIC50:  210nMAssay Description:Inhibitory concentration towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160483(1-Benzyl-2-methylsulfanyl-1H-benzoimidazole-5-sulf...)
Affinity DataIC50:  220nMAssay Description:Inhibitory concentration towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160485(1-Benzyl-2-(2-pyridin-2-yl-ethylsulfanyl)-1H-benzo...)
Affinity DataIC50:  230nMAssay Description:Inhibitory concentration towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160489(1-Benzyl-2-(pyridin-4-ylmethylsulfanyl)-1H-benzoim...)
Affinity DataIC50:  240nMAssay Description:Inhibitory concentration towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160496(1-Benzyl-2-ethylsulfanyl-1H-benzoimidazole-5-sulfo...)
Affinity DataIC50:  250nMAssay Description:Inhibitory concentration towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160487(1-Benzyl-2-(2-hydroxy-ethylsulfanyl)-1H-benzoimida...)
Affinity DataIC50:  270nMAssay Description:Inhibitory concentration towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160485(1-Benzyl-2-(2-pyridin-2-yl-ethylsulfanyl)-1H-benzo...)
Affinity DataIC50:  280nMAssay Description:Inhibitory concentration towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160490(1-Benzyl-2-ethylsulfanyl-1H-benzoimidazole-5-sulfo...)
Affinity DataIC50:  280nMAssay Description:Inhibitory concentration towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160491(1-Benzyl-2-ethoxy-1H-benzoimidazole-5-sulfonic aci...)
Affinity DataIC50:  300nMAssay Description:Inhibitory concentration towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160489(1-Benzyl-2-(pyridin-4-ylmethylsulfanyl)-1H-benzoim...)
Affinity DataIC50:  320nMAssay Description:Inhibitory concentration towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160490(1-Benzyl-2-ethylsulfanyl-1H-benzoimidazole-5-sulfo...)
Affinity DataIC50:  330nMAssay Description:Inhibitory concentration towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160491(1-Benzyl-2-ethoxy-1H-benzoimidazole-5-sulfonic aci...)
Affinity DataIC50:  470nMAssay Description:Inhibitory concentration towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160492(CHEMBL183572 | [1-Benzyl-5-(4-fluoro-benzylsulfamo...)
Affinity DataIC50:  490nMAssay Description:Inhibitory concentration towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160484(1-Benzyl-2-(2-benzylamino-ethylsulfanyl)-1H-benzoi...)
Affinity DataIC50:  530nMAssay Description:Inhibitory concentration towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160487(1-Benzyl-2-(2-hydroxy-ethylsulfanyl)-1H-benzoimida...)
Affinity DataIC50:  600nMAssay Description:Inhibitory concentration towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160484(1-Benzyl-2-(2-benzylamino-ethylsulfanyl)-1H-benzoi...)
Affinity DataIC50:  670nMAssay Description:Inhibitory concentration towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160492(CHEMBL183572 | [1-Benzyl-5-(4-fluoro-benzylsulfamo...)
Affinity DataIC50:  810nMAssay Description:Inhibitory concentration towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160486(1-Benzyl-2-(pyridin-2-ylmethylsulfanyl)-1H-benzoim...)
Affinity DataIC50:  820nMAssay Description:Inhibitory concentration towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160503(1-(3-Chloro-benzyl)-2-ethoxy-1H-benzoimidazole-5-s...)
Affinity DataIC50:  880nMAssay Description:Inhibitory concentration towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160494(1-Benzyl-2-ethylsulfanyl-1H-benzoimidazole-5-sulfo...)
Affinity DataIC50:  940nMAssay Description:Inhibitory concentration towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160486(1-Benzyl-2-(pyridin-2-ylmethylsulfanyl)-1H-benzoim...)
Affinity DataIC50:  960nMAssay Description:Inhibitory concentration towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160502(1-Benzyl-2-ethylsulfanyl-1H-benzoimidazole-5-sulfo...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibitory concentration towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160494(1-Benzyl-2-ethylsulfanyl-1H-benzoimidazole-5-sulfo...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibitory concentration towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160502(1-Benzyl-2-ethylsulfanyl-1H-benzoimidazole-5-sulfo...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibitory concentration towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160493(2-Ethoxy-1-thiophen-3-ylmethyl-1H-benzoimidazole-5...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibitory concentration towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160503(1-(3-Chloro-benzyl)-2-ethoxy-1H-benzoimidazole-5-s...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibitory concentration towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160493(2-Ethoxy-1-thiophen-3-ylmethyl-1H-benzoimidazole-5...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibitory concentration towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160504(2-Ethoxy-1-(2-morpholin-4-yl-ethyl)-1H-benzoimidaz...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibitory concentration towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160498(1-Benzyl-2-(2-morpholin-4-yl-ethoxy)-1H-benzoimida...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibitory concentration towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160497(1-Benzyl-2-ethylsulfanyl-1H-benzoimidazole-5-sulfo...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibitory concentration towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160497(1-Benzyl-2-ethylsulfanyl-1H-benzoimidazole-5-sulfo...)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibitory concentration towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160498(1-Benzyl-2-(2-morpholin-4-yl-ethoxy)-1H-benzoimida...)
Affinity DataIC50:  5.80E+3nMAssay Description:Inhibitory concentration towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160504(2-Ethoxy-1-(2-morpholin-4-yl-ethyl)-1H-benzoimidaz...)
Affinity DataIC50:  7.20E+3nMAssay Description:Inhibitory concentration towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160500(2-Ethylsulfanyl-1-phenethyl-1H-benzoimidazole-5-su...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory concentration towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160495(1-Benzyl-2-(2-morpholin-4-yl-ethylamino)-1H-benzoi...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory concentration towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160495(1-Benzyl-2-(2-morpholin-4-yl-ethylamino)-1H-benzoi...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory concentration towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160500(2-Ethylsulfanyl-1-phenethyl-1H-benzoimidazole-5-su...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory concentration towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160499(1-Benzyl-2-ethylsulfanyl-1H-benzoimidazole-5-sulfo...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory concentration towards human leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50160499(1-Benzyl-2-ethylsulfanyl-1H-benzoimidazole-5-sulfo...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory concentration towards rat leutinizing releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed