TargetCytochrome P450 2D6(Homo sapiens (Human))
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 82nMAssay Description:Inhibition of human liver microsome CYP2D6 in assessed as [14C]formaldehyde formationMore data for this Ligand-Target Pair
TargetCytochrome P450 3A4(Homo sapiens (Human))
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 440nMAssay Description:Inhibition of human liver microsome CYP3A4 in assessed as [14C]formaldehyde formationMore data for this Ligand-Target Pair
TargetCytochrome P450 3A4(Homo sapiens (Human))
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of human liver microsome CYP3A4 in assessed as [14C]formaldehyde formationMore data for this Ligand-Target Pair
TargetCytochrome P450 3A4(Homo sapiens (Human))
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 830nMAssay Description:Inhibition of human liver microsome CYP3A4 in assessed as [14C]formaldehyde formationMore data for this Ligand-Target Pair
TargetCytochrome P450 3A4(Homo sapiens (Human))
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 830nMAssay Description:Inhibition of human liver microsome CYP3A4 in assessed as [14C]formaldehyde formationMore data for this Ligand-Target Pair
TargetCytochrome P450 3A4(Homo sapiens (Human))
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human liver microsome CYP3A4 in assessed as [14C]formaldehyde formationMore data for this Ligand-Target Pair
TargetCytochrome P450 3A4(Homo sapiens (Human))
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human liver microsome CYP3A4 in assessed as [14C]formaldehyde formationMore data for this Ligand-Target Pair
TargetCytochrome P450 3A4(Homo sapiens (Human))
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibition of human liver microsome CYP3A4 in assessed as [14C]formaldehyde formationMore data for this Ligand-Target Pair
TargetCytochrome P450 3A4(Homo sapiens (Human))
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 7.70E+3nMAssay Description:Inhibition of human liver microsome CYP3A4 in assessed as [14C]formaldehyde formationMore data for this Ligand-Target Pair
TargetCytochrome P450 3A4(Homo sapiens (Human))
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of human liver microsome CYP3A4 in assessed as [14C]formaldehyde formationMore data for this Ligand-Target Pair
TargetCytochrome P450 3A4(Homo sapiens (Human))
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 8.80E+3nMAssay Description:Inhibition of human liver microsome CYP3A4 in assessed as [14C]formaldehyde formationMore data for this Ligand-Target Pair
TargetCytochrome P450 3A4(Homo sapiens (Human))
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of human liver microsome CYP3A4 in assessed as [14C]formaldehyde formationMore data for this Ligand-Target Pair
TargetCytochrome P450 3A4(Homo sapiens (Human))
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 9.50E+3nMAssay Description:Inhibition of human liver microsome CYP3A4 in assessed as [14C]formaldehyde formationMore data for this Ligand-Target Pair
TargetCytochrome P450 3A4(Homo sapiens (Human))
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 1.37E+4nMAssay Description:Inhibition of human liver microsome CYP3A4 in assessed as [14C]formaldehyde formationMore data for this Ligand-Target Pair
TargetCytochrome P450 3A4(Homo sapiens (Human))
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 1.49E+4nMAssay Description:Inhibition of human liver microsome CYP3A4 in assessed as [14C]formaldehyde formationMore data for this Ligand-Target Pair
TargetCytochrome P450 3A4(Homo sapiens (Human))
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of human liver microsome CYP3A4 in assessed as [14C]formaldehyde formationMore data for this Ligand-Target Pair
TargetCytochrome P450 2D6(Homo sapiens (Human))
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 1.75E+4nMAssay Description:Inhibition of human liver microsome CYP2D6 in assessed as [14C]formaldehyde formationMore data for this Ligand-Target Pair
TargetCytochrome P450 2D6(Homo sapiens (Human))
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 2.65E+4nMAssay Description:Inhibition of human liver microsome CYP2D6 in assessed as [14C]formaldehyde formationMore data for this Ligand-Target Pair
TargetCytochrome P450 3A4(Homo sapiens (Human))
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 2.87E+4nMAssay Description:Inhibition of human liver microsome CYP3A4 in assessed as [14C]formaldehyde formationMore data for this Ligand-Target Pair
TargetCytochrome P450 2D6(Homo sapiens (Human))
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 3.55E+4nMAssay Description:Inhibition of human liver microsome CYP2D6 in assessed as [14C]formaldehyde formationMore data for this Ligand-Target Pair
TargetCytochrome P450 3A4(Homo sapiens (Human))
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 7.40E+4nMAssay Description:Inhibition of human liver microsome CYP3A4 in assessed as [14C]formaldehyde formationMore data for this Ligand-Target Pair
TargetCytochrome P450 3A4(Homo sapiens (Human))
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 8.54E+4nMAssay Description:Inhibition of human liver microsome CYP3A4 in assessed as [14C]formaldehyde formationMore data for this Ligand-Target Pair
TargetCytochrome P450 2D6(Homo sapiens (Human))
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 8.79E+4nMAssay Description:Inhibition of human liver microsome CYP2D6 in assessed as [14C]formaldehyde formationMore data for this Ligand-Target Pair
TargetCytochrome P450 2D6(Homo sapiens (Human))
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 9.57E+4nMAssay Description:Inhibition of human liver microsome CYP2D6 in assessed as [14C]formaldehyde formationMore data for this Ligand-Target Pair
TargetCytochrome P450 3A4(Homo sapiens (Human))
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 9.82E+4nMAssay Description:Inhibition of human liver microsome CYP3A4 in assessed as [14C]formaldehyde formationMore data for this Ligand-Target Pair
TargetCytochrome P450 2D6(Homo sapiens (Human))
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human liver microsome CYP2D6 in assessed as [14C]formaldehyde formationMore data for this Ligand-Target Pair
TargetCytochrome P450 2D6(Homo sapiens (Human))
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human liver microsome CYP2D6 in assessed as [14C]formaldehyde formationMore data for this Ligand-Target Pair
TargetCytochrome P450 2D6(Homo sapiens (Human))
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human liver microsome CYP2D6 in assessed as [14C]formaldehyde formationMore data for this Ligand-Target Pair
TargetCytochrome P450 2D6(Homo sapiens (Human))
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human liver microsome CYP2D6 in assessed as [14C]formaldehyde formationMore data for this Ligand-Target Pair
TargetCytochrome P450 2D6(Homo sapiens (Human))
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human liver microsome CYP2D6 in assessed as [14C]formaldehyde formationMore data for this Ligand-Target Pair
TargetCytochrome P450 2D6(Homo sapiens (Human))
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human liver microsome CYP2D6 in assessed as [14C]formaldehyde formationMore data for this Ligand-Target Pair
TargetCytochrome P450 2D6(Homo sapiens (Human))
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human liver microsome CYP2D6 in assessed as [14C]formaldehyde formationMore data for this Ligand-Target Pair
TargetCytochrome P450 2D6(Homo sapiens (Human))
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human liver microsome CYP2D6 in assessed as [14C]formaldehyde formationMore data for this Ligand-Target Pair
TargetCytochrome P450 2D6(Homo sapiens (Human))
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human liver microsome CYP2D6 in assessed as [14C]formaldehyde formationMore data for this Ligand-Target Pair
TargetCytochrome P450 2D6(Homo sapiens (Human))
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human liver microsome CYP2D6 in assessed as [14C]formaldehyde formationMore data for this Ligand-Target Pair
TargetCytochrome P450 2D6(Homo sapiens (Human))
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human liver microsome CYP2D6 in assessed as [14C]formaldehyde formationMore data for this Ligand-Target Pair
TargetCytochrome P450 2D6(Homo sapiens (Human))
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human liver microsome CYP2D6 in assessed as [14C]formaldehyde formationMore data for this Ligand-Target Pair
TargetCytochrome P450 2D6(Homo sapiens (Human))
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human liver microsome CYP2D6 in assessed as [14C]formaldehyde formationMore data for this Ligand-Target Pair
TargetCytochrome P450 2D6(Homo sapiens (Human))
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human liver microsome CYP2D6 in assessed as [14C]formaldehyde formationMore data for this Ligand-Target Pair
TargetCytochrome P450 2D6(Homo sapiens (Human))
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human liver microsome CYP2D6 in assessed as [14C]formaldehyde formationMore data for this Ligand-Target Pair