Compile Data Set for Download or QSAR
maximum 50k data
Found 45 Enz. Inhib. hit(s) with all data for entry = 50015916
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162325(5-ethyl-3-{2-[1-(5-ethyl-2-sulfanyl-3-thienyl)-(E)...)
Affinity DataIC50:  6.00E+3nMAssay Description:Concentration to inhibit strand transfer of soluble mutant (F185K, C280S) of wild type Human immunodeficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162324(Benzene-1,3,5-tricarboxylic acid tris-[(furan-2-yl...)
Affinity DataIC50:  8.00E+3nMAssay Description:Concentration to inhibit strand transfer of wild type Human immuno deficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162334(5-[3-carboxy-4-(3-nitrophenylcarboxamido)benzyl]-2...)
Affinity DataIC50:  1.30E+4nMAssay Description:Concentration of the compound to inhibit strand transfer of wild type Human immunodeficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162334(5-[3-carboxy-4-(3-nitrophenylcarboxamido)benzyl]-2...)
Affinity DataIC50:  1.50E+4nMAssay Description:Concentration to inhibit 3' processing of wild type Human immunodeficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162325(5-ethyl-3-{2-[1-(5-ethyl-2-sulfanyl-3-thienyl)-(E)...)
Affinity DataIC50:  2.10E+4nMAssay Description:Concentration to inhibit strand transfer of wild type Human immuno deficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162323(1-(2-fluorophenylcarboxamido)-4-[3-(2-fluorophenyl...)
Affinity DataIC50:  3.30E+4nMAssay Description:Concentration to inhibit strand transfer of soluble mutant (F185K, C280S) of wild type Human immunodeficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162324(Benzene-1,3,5-tricarboxylic acid tris-[(furan-2-yl...)
Affinity DataIC50:  3.70E+4nMAssay Description:Concentration to inhibit 3' processing of wild type Human immuno deficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162333(5-[3-carboxy-4-(2-thienylcarboxamido)benzyl]-2-(2-...)
Affinity DataIC50:  3.80E+4nMAssay Description:Concentration of the compound to inhibit strand transfer of wild type Human immunodeficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162328(CHEMBL195166 | N-Furan-2-ylmethyl-N''-(3-{[(furan-...)
Affinity DataIC50:  4.00E+4nMAssay Description:Concentration to inhibit strand transfer of soluble mutant (F185K, C280S) of wild type Human immunodeficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162335(5-Cyclopropyl-2H-pyrazole-3-carboxylic acid [1-(2,...)
Affinity DataIC50:  4.30E+4nMAssay Description:Concentration to inhibit strand transfer of wild type Human immuno deficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162333(5-[3-carboxy-4-(2-thienylcarboxamido)benzyl]-2-(2-...)
Affinity DataIC50:  6.30E+4nMAssay Description:Concentration to inhibit 3' processing of wild type Human immunodeficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162332(5-(4-Benzylamino-3-nitro-benzenesulfonylamino)-iso...)
Affinity DataIC50:  6.60E+4nMAssay Description:Concentration of the compound to inhibit strand transfer of wild type Human immunodeficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162327(CHEMBL191854 | N-{5-[(5-Chloro-2-methyl-phenylamin...)
Affinity DataIC50:  7.00E+4nMAssay Description:Concentration to inhibit strand transfer of soluble mutant (F185K, C280S) of wild type Human immunodeficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162341(2-Methyl-4-oxo-5-[1-{5-[(p-tolylaminooxalyl-amino)...)
Affinity DataIC50:  8.10E+4nMAssay Description:Concentration to inhibit strand transfer of wild type Human immunodeficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162329(3-[4-(2-methyloxycarbonyl-3-thienylcarbamoyl)pheny...)
Affinity DataIC50:  9.70E+4nMAssay Description:Concentration of the compound to inhibit strand transfer of wild type Human immunodeficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162327(CHEMBL191854 | N-{5-[(5-Chloro-2-methyl-phenylamin...)
Affinity DataIC50: >1.00E+5nMAssay Description:Concentration to inhibit strand transfer of wild type Human immuno deficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162328(CHEMBL195166 | N-Furan-2-ylmethyl-N''-(3-{[(furan-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Concentration to inhibit 3' processing of wild type Human immuno deficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162323(1-(2-fluorophenylcarboxamido)-4-[3-(2-fluorophenyl...)
Affinity DataIC50: >1.00E+5nMAssay Description:Concentration to inhibit 3' processing of wild type Human immunodeficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162328(CHEMBL195166 | N-Furan-2-ylmethyl-N''-(3-{[(furan-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Concentration to inhibit strand transfer of wild type Human immuno deficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162322(2-hydroxy-4-[3-hydroxy-4-(4-methoxyphenylcarboxami...)
Affinity DataIC50: >1.00E+5nMAssay Description:Concentration to inhibit 3' processing of wild type Human immuno deficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162336(5-Cyclopropyl-2H-pyrazole-3-carboxylic acid [1-(4-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Concentration to inhibit 3' processing of wild type Human immuno deficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162339(5-{3-Amino-4-[(pyridin-3-ylmethyl)-amino]-benzenes...)
Affinity DataIC50: >1.00E+5nMAssay Description:Concentration to inhibit strand transfer of wild type Human immuno deficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162331(2-[(4-Bromo-phenylcarbamoyl)-methylsulfanyl]-6-hyd...)
Affinity DataIC50: >1.00E+5nMAssay Description:Concentration to inhibit strand transfer of wild type Human immuno deficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162323(1-(2-fluorophenylcarboxamido)-4-[3-(2-fluorophenyl...)
Affinity DataIC50: >1.00E+5nMAssay Description:Concentration of the compound to inhibit strand transfer of wild type Human immunodeficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162322(2-hydroxy-4-[3-hydroxy-4-(4-methoxyphenylcarboxami...)
Affinity DataIC50: >1.00E+5nMAssay Description:Concentration to inhibit strand transfer of wild type Human immuno deficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162340(CHEMBL179185 | {4-[3-(4-Benzoyl-3-hydroxy-phenoxy)...)
Affinity DataIC50: >1.00E+5nMAssay Description:Concentration to inhibit strand transfer of wild type Human immuno deficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162326(2-Hydroxy-5-[2-(5-methoxy-1H-benzoimidazol-2-ylsul...)
Affinity DataIC50: >1.00E+5nMAssay Description:Concentration to inhibit 3' processing of wild type Human immuno deficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162326(2-Hydroxy-5-[2-(5-methoxy-1H-benzoimidazol-2-ylsul...)
Affinity DataIC50: >1.00E+5nMAssay Description:Concentration to inhibit strand transfer of wild type Human immuno deficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162338(5-[4-(3-Morpholin-4-yl-propylamino)-3-nitro-benzen...)
Affinity DataIC50:  1.00E+5nMAssay Description:Concentration to inhibit strand transfer of wild type Human immuno deficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162331(2-[(4-Bromo-phenylcarbamoyl)-methylsulfanyl]-6-hyd...)
Affinity DataIC50: >1.00E+5nMAssay Description:Concentration to inhibit 3' processing of wild type Human immuno deficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162325(5-ethyl-3-{2-[1-(5-ethyl-2-sulfanyl-3-thienyl)-(E)...)
Affinity DataIC50: >1.00E+5nMAssay Description:Concentration to inhibit 3' processing of wild type Human immuno deficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162325(5-ethyl-3-{2-[1-(5-ethyl-2-sulfanyl-3-thienyl)-(E)...)
Affinity DataIC50: >1.00E+5nMAssay Description:Concentration to inhibit 3' processing of soluble mutant (F185K, C280S) of wild type Human immunodeficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162339(5-{3-Amino-4-[(pyridin-3-ylmethyl)-amino]-benzenes...)
Affinity DataIC50: >1.00E+5nMAssay Description:Concentration to inhibit 3' processing of wild type Human immuno deficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162336(5-Cyclopropyl-2H-pyrazole-3-carboxylic acid [1-(4-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Concentration to inhibit strand transfer of wild type Human immuno deficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162327(CHEMBL191854 | N-{5-[(5-Chloro-2-methyl-phenylamin...)
Affinity DataIC50: >1.00E+5nMAssay Description:Concentration to inhibit 3' processing of wild type Human immuno deficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162340(CHEMBL179185 | {4-[3-(4-Benzoyl-3-hydroxy-phenoxy)...)
Affinity DataIC50: >1.00E+5nMAssay Description:Concentration to inhibit 3' processing of wild type Human immuno deficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162338(5-[4-(3-Morpholin-4-yl-propylamino)-3-nitro-benzen...)
Affinity DataIC50:  1.40E+5nMAssay Description:Concentration to inhibit 3' processing of wild type Human immuno deficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162337(3-[(2,4-Dihydroxy-benzoyl)-hydrazono]-N-(2,4,6-tri...)
Affinity DataIC50:  1.50E+5nMAssay Description:Concentration of the compound to inhibit strand transfer of wild type Human immunodeficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162335(5-Cyclopropyl-2H-pyrazole-3-carboxylic acid [1-(2,...)
Affinity DataIC50:  1.77E+5nMAssay Description:Concentration to inhibit 3' processing of wild type Human immuno deficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162323(1-(2-fluorophenylcarboxamido)-4-[3-(2-fluorophenyl...)
Affinity DataIC50:  2.05E+5nMAssay Description:Concentration to inhibit 3' processing of soluble mutant (F185K, C280S) of wild type Human immunodeficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162330(2-[3-(4-Methoxy-phenylsulfamoyl)-benzoylamino]-ben...)
Affinity DataIC50:  3.00E+5nMAssay Description:Concentration to inhibit strand transfer of wild type Human immuno deficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162330(2-[3-(4-Methoxy-phenylsulfamoyl)-benzoylamino]-ben...)
Affinity DataIC50:  3.55E+5nMAssay Description:Concentration to inhibit 3' processing of wild type Human immuno deficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162327(CHEMBL191854 | N-{5-[(5-Chloro-2-methyl-phenylamin...)
Affinity DataIC50:  5.10E+5nMAssay Description:Concentration to inhibit 3' processing of soluble mutant (F185K, C280S) of wild type Human immunodeficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162337(3-[(2,4-Dihydroxy-benzoyl)-hydrazono]-N-(2,4,6-tri...)
Affinity DataIC50: >1.00E+6nMAssay Description:Concentration to inhibit 3' processing of wild type Human immunodeficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50162328(CHEMBL195166 | N-Furan-2-ylmethyl-N''-(3-{[(furan-...)
Affinity DataIC50:  1.00E+6nMAssay Description:Concentration to inhibit 3' processing of soluble mutant (F185K, C280S) of wild type Human immunodeficiency virus-1 integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed