Compile Data Set for Download or QSAR
maximum 50k data
Found 98 Enz. Inhib. hit(s) with all data for entry = 1591
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12466((2S)-1-[2-(adamantan-1-ylamino)acetyl]pyrrolidine-...)
Affinity DataIC50:  350nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12437(1-Benzyl-N-(2-cyclohexylidene-2-fluoroethyl)-4-pip...)
Affinity DataIC50:  1.04E+3nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12425(1-Benzyl-N-(2-cyclopentylidene-2-fluoroethyl)-4-pi...)
Affinity DataIC50:  1.30E+3nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12465((2S)-1-{2-[(2-phenylethyl)amino]acetyl}pyrrolidine...)
Affinity DataIC50:  2.13E+3nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12455(1-Benzyl-N-[2-oxo-2-(1-piperidinyl)ethyl]-4-piperi...)
Affinity DataIC50:  3.10E+3nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12467((2S)-1-(2-{[(4-fluorophenyl)methyl]amino}acetyl)py...)
Affinity DataIC50:  3.70E+3nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12436(9.8j | Fluoro-Olefin Analogue 18 | N-(2-Cyclohexyl...)
Affinity DataIC50:  4.20E+3nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12442((2H-1,3-benzodioxol-5-ylmethyl)(2-cyclopentylidene...)
Affinity DataIC50:  7.50E+3nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12434((2-cyclohexylidene-2-fluoroethyl)({[3-(trifluorome...)
Affinity DataIC50:  9.60E+3nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12422((2-cyclopentylidene-2-fluoroethyl)[(4-fluorophenyl...)
Affinity DataIC50:  1.08E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12435((2-cyclohexylidene-2-fluoroethyl)(2-phenylethyl)am...)
Affinity DataIC50:  1.10E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12460((1R,S)-(2Z)-2-[2-(1-Adamantylamino)-1-fluoroethyli...)
Affinity DataIC50:  1.20E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12438(9.8l | Benzyl 4-[(2-cyclohexylidene-2-fluoroethyl)...)
Affinity DataIC50:  1.28E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12432((2H-1,3-benzodioxol-5-ylmethyl)(2-cyclohexylidene-...)
Affinity DataIC50:  1.29E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12431((2-cyclohexylidene-2-fluoroethyl)[(4-methoxyphenyl...)
Affinity DataIC50:  1.34E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12451((2H-1,3-benzodioxol-5-ylmethyl)(2-cyclohexylidenee...)
Affinity DataIC50:  1.44E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12463((1R,S)-(2E)-2-[2-(1-Adamantylamino)-1-fluoroethyli...)
Affinity DataIC50:  1.50E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12421((2-cyclopentylidene-2-fluoroethyl)[(4-methoxypheny...)
Affinity DataIC50:  1.55E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12423((2-cyclopentylidene-2-fluoroethyl)[2-(pyridin-2-yl...)
Affinity DataIC50:  1.57E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12465((2S)-1-{2-[(2-phenylethyl)amino]acetyl}pyrrolidine...)
Affinity DataIC50:  1.63E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12433((2-cyclohexylidene-2-fluoroethyl)[(4-fluorophenyl)...)
Affinity DataIC50:  2.19E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12467((2S)-1-(2-{[(4-fluorophenyl)methyl]amino}acetyl)py...)
Affinity DataIC50:  2.55E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12441(10.7b | Olefin Analogue 23 | benzyl(2-cyclopentyli...)
Affinity DataIC50:  2.60E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12424((2-cyclopentylidene-2-fluoroethyl)(2-phenylethyl)a...)
Affinity DataIC50:  2.72E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12459((1R,S)-(2Z)-2-{1-Fluoro-2-[(2-phenylethyl)amino]et...)
Affinity DataIC50:  3.29E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12430(9.8d | Fluoro-Olefin Analogue 12 | N-Benzyl-2-cycl...)
Affinity DataIC50:  3.40E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12462((1R,S)-(2E)-2-{1-Fluoro-2-[(2-phenylethyl)amino]et...)
Affinity DataIC50:  3.61E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12420(9.7b | Fluoro-Olefin Analogue 2 | N-Benzyl-2-cyclo...)
Affinity DataIC50:  3.78E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12464((1R,S)-(2E)-2-{1-Fluoro-2-[(4-fluorobenzyl)amino]e...)
Affinity DataIC50:  4.04E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12458((2H-1,3-benzodioxol-5-ylmethyl)[2-(piperidin-1-yl)...)
Affinity DataIC50:  4.20E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12457(16.2b | N-Benzyl-2-thioxo-2-(1-piperidinyl)ethanea...)
Affinity DataIC50:  4.84E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12454(15.2c | 2-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-1...)
Affinity DataIC50:  5.20E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12426((2-cyclopentylidene-2-fluoroethyl)[3-(dimethylamin...)
Affinity DataIC50:  5.37E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12439((2-cyclohexylidene-2-fluoroethyl)[3-(dimethylamino...)
Affinity DataIC50:  5.46E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12450(10.8b | Olefin Analogue 32 | benzyl(2-cyclohexylid...)
Affinity DataIC50:  5.53E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12440(10.7a | N-(2-cyclopentylideneethyl)cyclohexanamine...)
Affinity DataIC50:  6.20E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12445(15.1c | 2-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-1...)
Affinity DataIC50:  6.30E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12448((2H-1,3-benzodioxol-5-ylmethyl)[2-(pyrrolidin-1-yl...)
Affinity DataIC50:  6.70E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12456(16.2a | N-Cyclohexyl-2-thioxo-2-(1-piperidinyl)eth...)
Affinity DataIC50:  6.90E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12461((1R,S)-(2Z)-2-{1-Fluoro-2-[(4-fluorobenzyl)amino]e...)
Affinity DataIC50:  8.73E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12419(9.7a | Fluoro-Olefin Analogue 1 | N-(2-Cyclopentyl...)
Affinity DataIC50:  9.00E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12428(9.8b | Fluoro-Olefin Analogue 10 | N-(2-Cyclohexyl...)
Affinity DataIC50:  9.13E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12446(16.1a | N-Cyclohexyl-2-thioxo-2-(1-pyrrolidinyl)et...)
Affinity DataIC50:  9.20E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12429(9.8c | Fluoro-Olefin Analogue 11 | N-(2-Cyclohexyl...)
Affinity DataIC50:  1.00E+5nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12463((1R,S)-(2E)-2-[2-(1-Adamantylamino)-1-fluoroethyli...)
Affinity DataIC50: >1.00E+5nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12460((1R,S)-(2Z)-2-[2-(1-Adamantylamino)-1-fluoroethyli...)
Affinity DataIC50: >1.00E+5nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12434((2-cyclohexylidene-2-fluoroethyl)({[3-(trifluorome...)
Affinity DataIC50: >1.25E+5nMpH: 8.3 T: 2°CAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12438(9.8l | Benzyl 4-[(2-cyclohexylidene-2-fluoroethyl)...)
Affinity DataIC50: >1.25E+5nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12466((2S)-1-[2-(adamantan-1-ylamino)acetyl]pyrrolidine-...)
Affinity DataIC50:  1.34E+5nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

LigandPNGBDBM12449(10.8a | N-(2-cyclohexylideneethyl)cyclohexanamine ...)
Affinity DataIC50:  1.36E+5nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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