Compile Data Set for Download or QSAR
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Found 19 Enz. Inhib. hit(s) with all data for entry = 50016057
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  5.40nMAssay Description:Inhibition of [3H]-SR-141,716A binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50067498((6aS,10aS)-3-(1,1-Dimethyl-heptyl)-9-hydroxymethyl...)
Affinity DataKi:  18.6nMAssay Description:Inhibition of [3H]-SR-141,716A binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50164429(3-Allyl-5,5-bis-(4-iodo-phenyl)-2-thioxo-imidazoli...)
Affinity DataKi:  589nMAssay Description:Inhibition of [3H]-SR-141,716A binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50164432(3-Butyl-5,5-bis-(4-iodo-phenyl)-2-thioxo-imidazoli...)
Affinity DataKi:  724nMAssay Description:Inhibition of [3H]-SR-141,716A binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50164431(3-Allyl-5,5-bis-(4-bromo-phenyl)-2-thioxo-imidazol...)
Affinity DataKi:  871nMAssay Description:Inhibition of [3H]-SR-141,716A binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50164441(3-Benzyl-5,5-bis-(4-bromo-phenyl)-2-thioxo-imidazo...)
Affinity DataKi:  993nMAssay Description:Inhibition of [3H]-SR-141,716A binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50164442(5,5-Bis-(4-bromo-phenyl)-3-butyl-2-thioxo-imidazol...)
Affinity DataKi:  1.41E+3nMAssay Description:Inhibition of [3H]-SR-141,716A binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50164439(3-Allyl-5,5-bis-(4-iodo-phenyl)-imidazolidine-2,4-...)
Affinity DataKi:  1.74E+3nMAssay Description:Inhibition of [3H]-SR-141,716A binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50164433(5,5-Bis-(4-bromo-phenyl)-3-isobutyl-2-thioxo-imida...)
Affinity DataKi:  1.78E+3nMAssay Description:Inhibition of [3H]-SR-141,716A binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50164430(3-Butyl-5,5-bis-(4-iodo-phenyl)-imidazolidine-2,4-...)
Affinity DataKi:  1.82E+3nMAssay Description:Inhibition of [3H]-SR-141,716A binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50164438(5,5-Bis-(4-chloro-phenyl)-3-isobutyl-2-thioxo-imid...)
Affinity DataKi:  2.09E+3nMAssay Description:Inhibition of [3H]-SR-141,716A binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50164440(3-Benzyl-5,5-bis-(4-chloro-phenyl)-2-thioxo-imidaz...)
Affinity DataKi:  2.19E+3nMAssay Description:Inhibition of [3H]-SR-141,716A binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50164428(5,5-Bis-(4-bromo-phenyl)-3-ethyl-2-thioxo-imidazol...)
Affinity DataKi:  2.19E+3nMAssay Description:Inhibition of [3H]-SR-141,716A binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50164443(3-Benzyl-5,5-bis-(4-bromo-phenyl)-imidazolidine-2,...)
Affinity DataKi:  3.47E+3nMAssay Description:Inhibition of [3H]-SR-141,716A binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50164437(5,5-Bis-(4-bromo-phenyl)-3-isopropyl-2-thioxo-imid...)
Affinity DataKi:  3.63E+3nMAssay Description:Inhibition of [3H]-SR-141,716A binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50164435(5,5-Bis-(4-chloro-phenyl)-3-phenethyl-2-thioxo-imi...)
Affinity DataKi:  3.80E+3nMAssay Description:Inhibition of [3H]-SR-141,716A binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM21281((11R)-2-methyl-11-(morpholin-4-ylmethyl)-3-(naphth...)
Affinity DataKi:  3.80E+3nMAssay Description:Inhibition of [3H]-SR-141,716A binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50164436(5,5-Bis-(4-bromo-phenyl)-3-butyl-imidazolidine-2,4...)
Affinity DataKi:  5.50E+3nMAssay Description:Inhibition of [3H]-SR-141,716A binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50164434(5,5-Bis-(4-bromo-phenyl)-3-phenethyl-2-thioxo-imid...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [3H]-SR-141,716A binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed