Compile Data Set for Download or QSAR
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Found 4 Enz. Inhib. hit(s) with all data for entry = 50016133
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Homo sapiens (Human))
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50165369(12-(4-Amino-4-carboxy-butyrylamino)-dodecanoic aci...)
Affinity DataIC50:  1.20nMAssay Description:Inhibitory activity against sarco- endoplasmic reticulum calcium-ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Homo sapiens (Human))
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50165368(CHEMBL191633 | Dodecanedioic acid mono-((2S,3aR,4S...)
Affinity DataIC50:  2.08nMAssay Description:Inhibitory activity against sarco- endoplasmic reticulum calcium-ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Homo sapiens (Human))
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50165366(CHEMBL191927 | Pentanedioic acid mono-((2S,3aR,4S,...)
Affinity DataIC50:  19.8nMAssay Description:Inhibitory activity against sarco- endoplasmic reticulum calcium-ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Homo sapiens (Human))
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50165367(CHEMBL362947 | Octanoic acid (2S,3aR,4S,6S,6aR,7S,...)
Affinity DataIC50:  9.04E+3nMAssay Description:Inhibitory activity against sarco- endoplasmic reticulum calcium-ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed