Compile Data Set for Download or QSAR
maximum 50k data
Found 57 Enz. Inhib. hit(s) with all data for entry = 50016207
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166332(9-[1-(3'-Fluoro-biphenyl-4-yl)-meth-(Z)-ylidene]-7...)
Affinity DataKi:  5nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166328(9-[3-(2,6-Difluoro-phenyl)-prop-2-yn-(Z)-ylidene]-...)
Affinity DataKi:  5.30nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166336(9-[1-[2,3']Bithiophenyl-5-yl-meth-(Z)-ylidene]-7-a...)
Affinity DataKi:  5.90nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166339(9-[1-(2'-Methoxy-biphenyl-4-yl)-meth-(Z)-ylidene]-...)
Affinity DataKi:  6.5nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM35229(3-(10,11-dihydro-5H-dibenzo[b,f]azepin-5-yl)-N-met...)
Affinity DataKi:  7.36nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166333(9-[1-(3'-Trifluoromethyl-biphenyl-4-yl)-meth-(Z)-y...)
Affinity DataKi:  8.80nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166334(9-[1-(3'-Methoxy-biphenyl-4-yl)-meth-(Z)-ylidene]-...)
Affinity DataKi:  9.40nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166341(9-[3-(4-Fluoro-phenyl)-prop-2-yn-(Z)-ylidene]-7-az...)
Affinity DataKi:  17nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166329(9-[3-Thiophen-3-yl-prop-2-yn-(Z)-ylidene]-7-aza-tr...)
Affinity DataKi:  22nMAssay Description:Inhibitory constant for [3H]-NE reuptake at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166328(9-[3-(2,6-Difluoro-phenyl)-prop-2-yn-(Z)-ylidene]-...)
Affinity DataKi:  32nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166336(9-[1-[2,3']Bithiophenyl-5-yl-meth-(Z)-ylidene]-7-a...)
Affinity DataKi:  32nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166330(9-[3-(3-Fluoro-4-methyl-phenyl)-prop-2-yn-(Z)-ylid...)
Affinity DataKi:  52nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166326(9-[1-(4'-Fluoro-biphenyl-4-yl)-meth-(Z)-ylidene]-7...)
Affinity DataKi:  53nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166327(9-[1-(4'-Methylsulfanyl-biphenyl-4-yl)-meth-(Z)-yl...)
Affinity DataKi:  62nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166337(9-[3-(3,4-Difluoro-phenyl)-prop-2-yn-(Z)-ylidene]-...)
Affinity DataKi:  69nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166329(9-[3-Thiophen-3-yl-prop-2-yn-(Z)-ylidene]-7-aza-tr...)
Affinity DataKi:  86nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166341(9-[3-(4-Fluoro-phenyl)-prop-2-yn-(Z)-ylidene]-7-az...)
Affinity DataKi:  104nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166337(9-[3-(3,4-Difluoro-phenyl)-prop-2-yn-(Z)-ylidene]-...)
Affinity DataKi:  110nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166336(9-[1-[2,3']Bithiophenyl-5-yl-meth-(Z)-ylidene]-7-a...)
Affinity DataKi:  114nMAssay Description:Inhibitory constant against reuptake of [3H]-DA at dopamine transporter of rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166334(9-[1-(3'-Methoxy-biphenyl-4-yl)-meth-(Z)-ylidene]-...)
Affinity DataKi:  114nMAssay Description:Inhibitory constant against reuptake of [3H]-DA at dopamine transporter of rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166332(9-[1-(3'-Fluoro-biphenyl-4-yl)-meth-(Z)-ylidene]-7...)
Affinity DataKi:  138nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166323(9-[3-Thiophen-2-yl-prop-2-yn-(Z)-ylidene]-7-aza-tr...)
Affinity DataKi:  142nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166326(9-[1-(4'-Fluoro-biphenyl-4-yl)-meth-(Z)-ylidene]-7...)
Affinity DataKi:  161nMAssay Description:Inhibitory constant against reuptake of [3H]-DA at dopamine transporter of rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM35229(3-(10,11-dihydro-5H-dibenzo[b,f]azepin-5-yl)-N-met...)
Affinity DataKi:  163nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166325(9-[3-Phenyl-prop-2-yn-(Z)-ylidene]-7-aza-tricyclo[...)
Affinity DataKi:  207nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166338(9-[3-(2,5-Difluoro-phenyl)-prop-2-yn-(Z)-ylidene]-...)
Affinity DataKi:  215nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50133750(9-[1-[5-(4-Methylsulfanyl-phenyl)-thiophen-2-yl]-m...)
Affinity DataKi:  273nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166335(9-[3-(3-Fluoro-phenyl)-prop-2-yn-(Z)-ylidene]-7-az...)
Affinity DataKi:  317nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166334(9-[1-(3'-Methoxy-biphenyl-4-yl)-meth-(Z)-ylidene]-...)
Affinity DataKi:  346nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166340(9-[1-(2'-Fluoro-biphenyl-4-yl)-meth-(Z)-ylidene]-7...)
Affinity DataKi:  393nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166340(9-[1-(2'-Fluoro-biphenyl-4-yl)-meth-(Z)-ylidene]-7...)
Affinity DataKi:  466nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166333(9-[1-(3'-Trifluoromethyl-biphenyl-4-yl)-meth-(Z)-y...)
Affinity DataKi:  556nMAssay Description:Inhibitory constant against reuptake of [3H]-DA at dopamine transporter of rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166332(9-[1-(3'-Fluoro-biphenyl-4-yl)-meth-(Z)-ylidene]-7...)
Affinity DataKi:  646nMAssay Description:Inhibitory constant against reuptake of [3H]-DA at dopamine transporter of rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166339(9-[1-(2'-Methoxy-biphenyl-4-yl)-meth-(Z)-ylidene]-...)
Affinity DataKi:  787nMAssay Description:Inhibitory constant against reuptake of [3H]-DA at dopamine transporter of rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166330(9-[3-(3-Fluoro-4-methyl-phenyl)-prop-2-yn-(Z)-ylid...)
Affinity DataKi:  914nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166327(9-[1-(4'-Methylsulfanyl-biphenyl-4-yl)-meth-(Z)-yl...)
Affinity DataKi:  1.05E+3nMAssay Description:Inhibitory constant against reuptake of [3H]-DA at dopamine transporter of rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166327(9-[1-(4'-Methylsulfanyl-biphenyl-4-yl)-meth-(Z)-yl...)
Affinity DataKi:  1.08E+3nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166333(9-[1-(3'-Trifluoromethyl-biphenyl-4-yl)-meth-(Z)-y...)
Affinity DataKi:  1.17E+3nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166339(9-[1-(2'-Methoxy-biphenyl-4-yl)-meth-(Z)-ylidene]-...)
Affinity DataKi:  1.34E+3nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166326(9-[1-(4'-Fluoro-biphenyl-4-yl)-meth-(Z)-ylidene]-7...)
Affinity DataKi:  1.39E+3nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166323(9-[3-Thiophen-2-yl-prop-2-yn-(Z)-ylidene]-7-aza-tr...)
Affinity DataKi:  1.57E+3nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50133750(9-[1-[5-(4-Methylsulfanyl-phenyl)-thiophen-2-yl]-m...)
Affinity DataKi:  1.65E+3nMAssay Description:Inhibitory constant against reuptake of [3H]-DA at dopamine transporter of rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166338(9-[3-(2,5-Difluoro-phenyl)-prop-2-yn-(Z)-ylidene]-...)
Affinity DataKi:  1.72E+3nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166335(9-[3-(3-Fluoro-phenyl)-prop-2-yn-(Z)-ylidene]-7-az...)
Affinity DataKi:  2.11E+3nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166337(9-[3-(3,4-Difluoro-phenyl)-prop-2-yn-(Z)-ylidene]-...)
Affinity DataKi:  3.15E+3nMAssay Description:Inhibitory constant against reuptake of [3H]-DA at dopamine transporter of rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50133750(9-[1-[5-(4-Methylsulfanyl-phenyl)-thiophen-2-yl]-m...)
Affinity DataKi:  3.32E+3nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166340(9-[1-(2'-Fluoro-biphenyl-4-yl)-meth-(Z)-ylidene]-7...)
Affinity DataKi:  3.40E+3nMAssay Description:Inhibitory constant against reuptake of [3H]-DA at dopamine transporter of rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166330(9-[3-(3-Fluoro-4-methyl-phenyl)-prop-2-yn-(Z)-ylid...)
Affinity DataKi:  7.07E+3nMAssay Description:Inhibitory constant against reuptake of [3H]-DA at dopamine transporter of rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166341(9-[3-(4-Fluoro-phenyl)-prop-2-yn-(Z)-ylidene]-7-az...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibitory constant against reuptake of [3H]-DA at dopamine transporter of rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery

Curated by ChEMBL
LigandPNGBDBM50166338(9-[3-(2,5-Difluoro-phenyl)-prop-2-yn-(Z)-ylidene]-...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibitory constant against reuptake of [3H]-DA at dopamine transporter of rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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