Affinity DataKi: 5nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
Affinity DataKi: 5.30nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
Affinity DataKi: 5.90nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
Affinity DataKi: 6.5nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
Affinity DataKi: 7.36nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
Affinity DataKi: 8.80nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
Affinity DataKi: 9.40nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery
Curated by ChEMBL
Acenta Discovery
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Inhibitory constant for [3H]-NE reuptake at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery
Curated by ChEMBL
Acenta Discovery
Curated by ChEMBL
Affinity DataKi: 32nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery
Curated by ChEMBL
Acenta Discovery
Curated by ChEMBL
Affinity DataKi: 32nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
Affinity DataKi: 52nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
Affinity DataKi: 53nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
Affinity DataKi: 62nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery
Curated by ChEMBL
Acenta Discovery
Curated by ChEMBL
Affinity DataKi: 69nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery
Curated by ChEMBL
Acenta Discovery
Curated by ChEMBL
Affinity DataKi: 86nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
Affinity DataKi: 104nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery
Curated by ChEMBL
Acenta Discovery
Curated by ChEMBL
Affinity DataKi: 114nMAssay Description:Inhibitory constant against reuptake of [3H]-DA at dopamine transporter of rat striatal membranesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery
Curated by ChEMBL
Acenta Discovery
Curated by ChEMBL
Affinity DataKi: 114nMAssay Description:Inhibitory constant against reuptake of [3H]-DA at dopamine transporter of rat striatal membranesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery
Curated by ChEMBL
Acenta Discovery
Curated by ChEMBL
Affinity DataKi: 138nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery
Curated by ChEMBL
Acenta Discovery
Curated by ChEMBL
Affinity DataKi: 142nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery
Curated by ChEMBL
Acenta Discovery
Curated by ChEMBL
Affinity DataKi: 161nMAssay Description:Inhibitory constant against reuptake of [3H]-DA at dopamine transporter of rat striatal membranesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery
Curated by ChEMBL
Acenta Discovery
Curated by ChEMBL
Affinity DataKi: 163nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery
Curated by ChEMBL
Acenta Discovery
Curated by ChEMBL
Affinity DataKi: 207nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery
Curated by ChEMBL
Acenta Discovery
Curated by ChEMBL
Affinity DataKi: 215nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
Affinity DataKi: 273nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery
Curated by ChEMBL
Acenta Discovery
Curated by ChEMBL
Affinity DataKi: 317nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery
Curated by ChEMBL
Acenta Discovery
Curated by ChEMBL
Affinity DataKi: 346nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
Affinity DataKi: 393nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery
Curated by ChEMBL
Acenta Discovery
Curated by ChEMBL
Affinity DataKi: 466nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery
Curated by ChEMBL
Acenta Discovery
Curated by ChEMBL
Affinity DataKi: 556nMAssay Description:Inhibitory constant against reuptake of [3H]-DA at dopamine transporter of rat striatal membranesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery
Curated by ChEMBL
Acenta Discovery
Curated by ChEMBL
Affinity DataKi: 646nMAssay Description:Inhibitory constant against reuptake of [3H]-DA at dopamine transporter of rat striatal membranesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery
Curated by ChEMBL
Acenta Discovery
Curated by ChEMBL
Affinity DataKi: 787nMAssay Description:Inhibitory constant against reuptake of [3H]-DA at dopamine transporter of rat striatal membranesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery
Curated by ChEMBL
Acenta Discovery
Curated by ChEMBL
Affinity DataKi: 914nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery
Curated by ChEMBL
Acenta Discovery
Curated by ChEMBL
Affinity DataKi: 1.05E+3nMAssay Description:Inhibitory constant against reuptake of [3H]-DA at dopamine transporter of rat striatal membranesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery
Curated by ChEMBL
Acenta Discovery
Curated by ChEMBL
Affinity DataKi: 1.08E+3nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery
Curated by ChEMBL
Acenta Discovery
Curated by ChEMBL
Affinity DataKi: 1.17E+3nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery
Curated by ChEMBL
Acenta Discovery
Curated by ChEMBL
Affinity DataKi: 1.34E+3nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery
Curated by ChEMBL
Acenta Discovery
Curated by ChEMBL
Affinity DataKi: 1.39E+3nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
Affinity DataKi: 1.57E+3nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery
Curated by ChEMBL
Acenta Discovery
Curated by ChEMBL
Affinity DataKi: 1.65E+3nMAssay Description:Inhibitory constant against reuptake of [3H]-DA at dopamine transporter of rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.72E+3nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
Affinity DataKi: 2.11E+3nMAssay Description:Inhibitory constant against reuptake of [3H]-NE at norepinephrine transporter of rat parietal-occipital cortexMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery
Curated by ChEMBL
Acenta Discovery
Curated by ChEMBL
Affinity DataKi: 3.15E+3nMAssay Description:Inhibitory constant against reuptake of [3H]-DA at dopamine transporter of rat striatal membranesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Acenta Discovery
Curated by ChEMBL
Acenta Discovery
Curated by ChEMBL
Affinity DataKi: 3.32E+3nMAssay Description:Inhibitory constant against reuptake of [3H]-5-HT at serotonin transporter of rat midbrain cortexMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery
Curated by ChEMBL
Acenta Discovery
Curated by ChEMBL
Affinity DataKi: 3.40E+3nMAssay Description:Inhibitory constant against reuptake of [3H]-DA at dopamine transporter of rat striatal membranesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery
Curated by ChEMBL
Acenta Discovery
Curated by ChEMBL
Affinity DataKi: 7.07E+3nMAssay Description:Inhibitory constant against reuptake of [3H]-DA at dopamine transporter of rat striatal membranesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery
Curated by ChEMBL
Acenta Discovery
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibitory constant against reuptake of [3H]-DA at dopamine transporter of rat striatal membranesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Acenta Discovery
Curated by ChEMBL
Acenta Discovery
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibitory constant against reuptake of [3H]-DA at dopamine transporter of rat striatal membranesMore data for this Ligand-Target Pair