Compile Data Set for Download or QSAR
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Found 7 Enz. Inhib. hit(s) with all data for entry = 50041592
TargetHistidine-rich protein PFHRP-II(Plasmodium falciparum)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50412201(CRYPTOLEPINE HYDROCHLORIDE | Cryptolepine)
Affinity DataIC50:  1.72E+9nMAssay Description:Inhibition of beta-hematin formation by BHIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine-rich protein PFHRP-II(Plasmodium falciparum)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM22985(Aralen | CHEMBL76 | CHLOROQUINE PHOSPHATE | Chloro...)
Affinity DataIC50:  2.56E+9nMAssay Description:Inhibition of beta-hematin formation by BHIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine-rich protein PFHRP-II(Plasmodium falciparum)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50412205(CHEMBL512770)
Affinity DataIC50:  5.24E+9nMAssay Description:Inhibition of beta-hematin formation by BHIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine-rich protein PFHRP-II(Plasmodium falciparum)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50412204(CHEMBL465591)
Affinity DataIC50:  5.97E+9nMAssay Description:Inhibition of beta-hematin formation by BHIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine-rich protein PFHRP-II(Plasmodium falciparum)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50367247(QUININE | Quinamm | Quinsan | cid_3034034)
Affinity DataIC50:  7.40E+9nMAssay Description:Inhibition of beta-hematin formation by BHIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine-rich protein PFHRP-II(Plasmodium falciparum)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50412203(CHEMBL502768)
Affinity DataIC50:  7.59E+9nMAssay Description:Inhibition of beta-hematin formation by BHIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine-rich protein PFHRP-II(Plasmodium falciparum)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50412202(CHEMBL463913)
Affinity DataIC50: >1.30E+10nMAssay Description:Inhibition of beta-hematin formation by BHIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed