Compile Data Set for Download or QSAR
maximum 50k data
Found 68 Enz. Inhib. hit(s) with all data for entry = 50016454
TargetPlasmepsin I(Plasmodium falciparum)
LinköPing University

Curated by ChEMBL
LigandPNGBDBM50169098(CHEMBL264770 | Pyridine-2-carboxylic acid {(S)-1-[...)
Affinity DataKi:  0.300nMAssay Description:Inhibitory concentration against the Plasmepsin I of Plasmodium falciparumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
LinköPing University

Curated by ChEMBL
LigandPNGBDBM50169100(CHEMBL191260 | Pyridine-2-carboxylic acid {(S)-1-[...)
Affinity DataKi:  0.300nMAssay Description:Inhibitory concentration against the Plasmepsin I of Plasmodium falciparumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
LinköPing University

Curated by ChEMBL
LigandPNGBDBM50169103(CHEMBL191130 | Pyridine-2-carboxylic acid {(S)-1-[...)
Affinity DataKi:  0.400nMAssay Description:Inhibitory concentration against the Plasmepsin I of Plasmodium falciparumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
LinköPing University

Curated by ChEMBL
LigandPNGBDBM50169104(CHEMBL371417 | Pyridine-2-carboxylic acid {(S)-1-[...)
Affinity DataKi:  0.400nMAssay Description:Inhibitory concentration against the Plasmepsin I of Plasmodium falciparumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
LinköPing University

Curated by ChEMBL
LigandPNGBDBM7977((3S,4S)-5-[(4-bromophenyl)methoxy]-N-[(1S)-1-{[(1S...)
Affinity DataKi:  0.5nMAssay Description:Inhibitory concentration against the Plasmepsin I of Plasmodium falciparumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
LinköPing University

Curated by ChEMBL
LigandPNGBDBM7974((3S,4S)-N-[(1S)-1-{[(1S)-1-carbamoyl-3-methylbutyl...)
Affinity DataKi:  0.560nMAssay Description:Inhibitory concentration against the Plasmepsin II of Plasmodium falciparumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
LinköPing University

Curated by ChEMBL
LigandPNGBDBM50169106(CHEMBL363286 | Pyridine-2-carboxylic acid ((S)-1-{...)
Affinity DataKi:  0.700nMAssay Description:Inhibitory concentration against the Plasmepsin I of Plasmodium falciparumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
LinköPing University

Curated by ChEMBL
LigandPNGBDBM50169103(CHEMBL191130 | Pyridine-2-carboxylic acid {(S)-1-[...)
Affinity DataKi:  0.700nMAssay Description:Inhibitory concentration against the human Cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
LinköPing University

Curated by ChEMBL
LigandPNGBDBM50169098(CHEMBL264770 | Pyridine-2-carboxylic acid {(S)-1-[...)
Affinity DataKi:  0.900nMAssay Description:Inhibitory concentration against the Plasmepsin II of Plasmodium falciparumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
LinköPing University

Curated by ChEMBL
LigandPNGBDBM50169109(CHEMBL190290 | Pyridine-2-carboxylic acid ((S)-1-{...)
Affinity DataKi:  1nMAssay Description:Inhibitory concentration against the Plasmepsin I of Plasmodium falciparumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
LinköPing University

Curated by ChEMBL
LigandPNGBDBM50169105(CHEMBL370086 | Pyridine-2-carboxylic acid {(S)-1-[...)
Affinity DataKi:  1nMAssay Description:Inhibitory concentration against the Plasmepsin I of Plasmodium falciparumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
LinköPing University

Curated by ChEMBL
LigandPNGBDBM50169103(CHEMBL191130 | Pyridine-2-carboxylic acid {(S)-1-[...)
Affinity DataKi:  1.10nMAssay Description:Inhibitory concentration against the Plasmepsin II of Plasmodium falciparumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
LinköPing University

Curated by ChEMBL
LigandPNGBDBM50169100(CHEMBL191260 | Pyridine-2-carboxylic acid {(S)-1-[...)
Affinity DataKi:  1.10nMAssay Description:Inhibitory concentration against the Plasmepsin II of Plasmodium falciparumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
LinköPing University

Curated by ChEMBL
LigandPNGBDBM50169104(CHEMBL371417 | Pyridine-2-carboxylic acid {(S)-1-[...)
Affinity DataKi:  1.60nMAssay Description:Inhibitory concentration against the human Cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
LinköPing University

Curated by ChEMBL
LigandPNGBDBM50169110(CHEMBL364630 | Pyridine-2-carboxylic acid {(S)-1-[...)
Affinity DataKi:  1.90nMAssay Description:Inhibitory concentration against the Plasmepsin I of Plasmodium falciparumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
LinköPing University

Curated by ChEMBL
LigandPNGBDBM50169104(CHEMBL371417 | Pyridine-2-carboxylic acid {(S)-1-[...)
Affinity DataKi:  1.90nMAssay Description:Inhibitory concentration against the Plasmepsin II of Plasmodium falciparumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
LinköPing University

Curated by ChEMBL
LigandPNGBDBM50169112(CHEMBL371082 | N-[(1S,2S)-3-[(S)-1-((S)-1-Carbamoy...)
Affinity DataKi:  2.10nMAssay Description:Inhibitory concentration against the Plasmepsin I of Plasmodium falciparumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
LinköPing University

Curated by ChEMBL
LigandPNGBDBM7977((3S,4S)-5-[(4-bromophenyl)methoxy]-N-[(1S)-1-{[(1S...)
Affinity DataKi:  2.20nMAssay Description:Inhibitory concentration against the Plasmepsin II of Plasmodium falciparumMore data for this Ligand-Target Pair
TargetCathepsin D(Homo sapiens (Human))
LinköPing University

Curated by ChEMBL
LigandPNGBDBM50169098(CHEMBL264770 | Pyridine-2-carboxylic acid {(S)-1-[...)
Affinity DataKi:  2.5nMAssay Description:Inhibitory concentration against the human Cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
LinköPing University

Curated by ChEMBL
LigandPNGBDBM50169113(CHEMBL371182 | Pyridine-2-carboxylic acid {(S)-1-[...)
Affinity DataKi:  2.70nMAssay Description:Inhibitory concentration against the Plasmepsin I of Plasmodium falciparumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
LinköPing University

Curated by ChEMBL
LigandPNGBDBM50169100(CHEMBL191260 | Pyridine-2-carboxylic acid {(S)-1-[...)
Affinity DataKi:  3.20nMAssay Description:Inhibitory concentration against the human Cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
LinköPing University

Curated by ChEMBL
LigandPNGBDBM50169102(CHEMBL189976 | N-{(1S,2S)-1-(4-Benzo[1,3]dioxol-5-...)
Affinity DataKi:  3.30nMAssay Description:Inhibitory concentration against the Plasmepsin I of Plasmodium falciparumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
LinköPing University

Curated by ChEMBL
LigandPNGBDBM7988((3S,4S)-5-[(4-bromophenyl)methoxy]-N-[(1S)-1-{[(1S...)
Affinity DataKi:  3.40nMAssay Description:Inhibitory concentration against the Plasmepsin I of Plasmodium falciparumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
LinköPing University

Curated by ChEMBL
LigandPNGBDBM50169106(CHEMBL363286 | Pyridine-2-carboxylic acid ((S)-1-{...)
Affinity DataKi:  3.90nMAssay Description:Inhibitory concentration against the human Cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
LinköPing University

Curated by ChEMBL
LigandPNGBDBM8019(2-(3-chlorophenoxy)-N-[(2S,3S)-3-hydroxy-4-{N-[2-(...)
Affinity DataKi:  4.30nMAssay Description:Inhibitory concentration against the Plasmepsin II of Plasmodium falciparumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
LinköPing University

Curated by ChEMBL
LigandPNGBDBM50169106(CHEMBL363286 | Pyridine-2-carboxylic acid ((S)-1-{...)
Affinity DataKi:  4.40nMAssay Description:Inhibitory concentration against the Plasmepsin II of Plasmodium falciparumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
LinköPing University

Curated by ChEMBL
LigandPNGBDBM7977((3S,4S)-5-[(4-bromophenyl)methoxy]-N-[(1S)-1-{[(1S...)
Affinity DataKi:  4.90nMAssay Description:Inhibitory concentration against the human Cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
LinköPing University

Curated by ChEMBL
LigandPNGBDBM50169109(CHEMBL190290 | Pyridine-2-carboxylic acid ((S)-1-{...)
Affinity DataKi:  5.70nMAssay Description:Inhibitory concentration against the Plasmepsin II of Plasmodium falciparumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
LinköPing University

Curated by ChEMBL
LigandPNGBDBM50169111(CHEMBL365935 | N-{(1S,2S)-1-(Biphenyl-4-ylmethoxym...)
Affinity DataKi:  5.90nMAssay Description:Inhibitory concentration against the Plasmepsin I of Plasmodium falciparumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
LinköPing University

Curated by ChEMBL
LigandPNGBDBM7985((3S,4S)-5-[(4-bromophenyl)methoxy]-N-butyl-3-hydro...)
Affinity DataKi:  8.10nMAssay Description:Inhibitory concentration against the Plasmepsin I of Plasmodium falciparumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
LinköPing University

Curated by ChEMBL
LigandPNGBDBM7988((3S,4S)-5-[(4-bromophenyl)methoxy]-N-[(1S)-1-{[(1S...)
Affinity DataKi:  10nMAssay Description:Inhibitory concentration against the Plasmepsin II of Plasmodium falciparumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
LinköPing University

Curated by ChEMBL
LigandPNGBDBM50169105(CHEMBL370086 | Pyridine-2-carboxylic acid {(S)-1-[...)
Affinity DataKi:  13nMAssay Description:Inhibitory concentration against the Plasmepsin II of Plasmodium falciparumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
LinköPing University

Curated by ChEMBL
LigandPNGBDBM50169110(CHEMBL364630 | Pyridine-2-carboxylic acid {(S)-1-[...)
Affinity DataKi:  16nMAssay Description:Inhibitory concentration against the Plasmepsin II of Plasmodium falciparumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
LinköPing University

Curated by ChEMBL
LigandPNGBDBM7974((3S,4S)-N-[(1S)-1-{[(1S)-1-carbamoyl-3-methylbutyl...)
Affinity DataKi:  16nMAssay Description:Inhibitory concentration against the Plasmepsin I of Plasmodium falciparumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
LinköPing University

Curated by ChEMBL
LigandPNGBDBM50169102(CHEMBL189976 | N-{(1S,2S)-1-(4-Benzo[1,3]dioxol-5-...)
Affinity DataKi:  19nMAssay Description:Inhibitory concentration against the Plasmepsin II of Plasmodium falciparumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
LinköPing University

Curated by ChEMBL
LigandPNGBDBM7974((3S,4S)-N-[(1S)-1-{[(1S)-1-carbamoyl-3-methylbutyl...)
Affinity DataKi:  21nMAssay Description:Inhibitory concentration against the human Cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
LinköPing University

Curated by ChEMBL
LigandPNGBDBM50169109(CHEMBL190290 | Pyridine-2-carboxylic acid ((S)-1-{...)
Affinity DataKi:  32nMAssay Description:Inhibitory concentration against the human Cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
LinköPing University

Curated by ChEMBL
LigandPNGBDBM50169113(CHEMBL371182 | Pyridine-2-carboxylic acid {(S)-1-[...)
Affinity DataKi:  45nMAssay Description:Inhibitory concentration against the Plasmepsin II of Plasmodium falciparumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
LinköPing University

Curated by ChEMBL
LigandPNGBDBM50169111(CHEMBL365935 | N-{(1S,2S)-1-(Biphenyl-4-ylmethoxym...)
Affinity DataKi:  48nMAssay Description:Inhibitory concentration against the Plasmepsin II of Plasmodium falciparumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
LinköPing University

Curated by ChEMBL
LigandPNGBDBM50169112(CHEMBL371082 | N-[(1S,2S)-3-[(S)-1-((S)-1-Carbamoy...)
Affinity DataKi:  55nMAssay Description:Inhibitory concentration against the Plasmepsin II of Plasmodium falciparumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
LinköPing University

Curated by ChEMBL
LigandPNGBDBM8019(2-(3-chlorophenoxy)-N-[(2S,3S)-3-hydroxy-4-{N-[2-(...)
Affinity DataKi:  63nMAssay Description:Inhibitory concentration against the human Cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
LinköPing University

Curated by ChEMBL
LigandPNGBDBM7985((3S,4S)-5-[(4-bromophenyl)methoxy]-N-butyl-3-hydro...)
Affinity DataKi:  68nMAssay Description:Inhibitory concentration against the Plasmepsin II of Plasmodium falciparumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
LinköPing University

Curated by ChEMBL
LigandPNGBDBM50169107(CHEMBL190348 | N-{(1S,2S)-1-(Biphenyl-4-ylmethoxym...)
Affinity DataKi:  116nMAssay Description:Inhibitory concentration against the Plasmepsin I of Plasmodium falciparumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
LinköPing University

Curated by ChEMBL
LigandPNGBDBM50169099(CHEMBL363692 | N-[(1S,2S)-1-(Biphenyl-4-ylmethoxym...)
Affinity DataKi:  188nMAssay Description:Inhibitory concentration against the Plasmepsin I of Plasmodium falciparumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
LinköPing University

Curated by ChEMBL
LigandPNGBDBM50169099(CHEMBL363692 | N-[(1S,2S)-1-(Biphenyl-4-ylmethoxym...)
Affinity DataKi:  214nMAssay Description:Inhibitory concentration against the Plasmepsin II of Plasmodium falciparumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
LinköPing University

Curated by ChEMBL
LigandPNGBDBM50169108(2,4,6-Trifluoro-N-[(1S,2S)-2-hydroxy-3-[2-(3-metho...)
Affinity DataKi:  221nMAssay Description:Inhibitory concentration against the Plasmepsin I of Plasmodium falciparumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
LinköPing University

Curated by ChEMBL
LigandPNGBDBM7995((3S,4S)-5-[(4-bromophenyl)methoxy]-N-cyclohexyl-3-...)
Affinity DataKi:  230nMAssay Description:Inhibitory concentration against the Plasmepsin II of Plasmodium falciparumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
LinköPing University

Curated by ChEMBL
LigandPNGBDBM50169105(CHEMBL370086 | Pyridine-2-carboxylic acid {(S)-1-[...)
Affinity DataKi:  241nMAssay Description:Inhibitory concentration against the human Cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
LinköPing University

Curated by ChEMBL
LigandPNGBDBM50169101(CHEMBL191487 | N-[(1S,2S)-3-Cyclohexylcarbamoyl-2-...)
Affinity DataKi:  260nMAssay Description:Inhibitory concentration against the Plasmepsin II of Plasmodium falciparumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin I(Plasmodium falciparum)
LinköPing University

Curated by ChEMBL
LigandPNGBDBM50169101(CHEMBL191487 | N-[(1S,2S)-3-Cyclohexylcarbamoyl-2-...)
Affinity DataKi:  278nMAssay Description:Inhibitory concentration against the Plasmepsin I of Plasmodium falciparumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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