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Found 22 Enz. Inhib. hit(s) with all data for entry = 50016525
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50170047((4-Hydroxy-3-iodo-5-methoxy-phenyl)-acetic acid (2...)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of 100 nM capsaicin effect on intracellular [Ca2+] concentration in HEK293 cells expressing human TRPV1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50170053(CHEMBL177809 | N-(4-hydroxy-2-iodo-5-methoxybenzyl...)
Affinity DataIC50:  10nMAssay Description:Inhibition of 100 nM capsaicin effect on intracellular [Ca2+] concentration in HEK293 cells expressing human TRPV1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50170062(CHEMBL190554 | Nonanoic acid 2-bromo-4-hydroxy-5-m...)
Affinity DataIC50:  16nMAssay Description:Inhibition of 100 nM capsaicin effect on intracellular [Ca2+] concentration in HEK293 cells expressing human TRPV1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50170061((E)-Octadec-9-enal | CHEMBL190707)
Affinity DataIC50:  35nMAssay Description:Inhibition of 100 nM capsaicin effect on intracellular [Ca2+] concentration in HEK293 cells expressing human TRPV1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50170054(CHEMBL187993 | Nonanoic acid 2-chloro-4-hydroxy-5-...)
Affinity DataIC50:  50nMAssay Description:Inhibition of 100 nM capsaicin effect on intracellular [Ca2+] concentration in HEK293 cells expressing human TRPV1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50170065((5E,8E,11E,14E)-Icosa-5,8,11,14-tetraenal | CHEMBL...)
Affinity DataIC50:  51nMAssay Description:Inhibition of 100 nM capsaicin effect on intracellular [Ca2+] concentration in HEK293 cells expressing human TRPV1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM20284(CHEMBL391997 | CPZ | Capsazepine | N-[2-(4-chlorop...)
Affinity DataIC50:  56nMAssay Description:Inhibition of 100 nM capsaicin effect on intracellular [Ca2+] concentration in HEK293 cells expressing human TRPV1More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50170066(CHEMBL365972 | Nonanoic acid 4-hydroxy-3-iodo-5-me...)
Affinity DataIC50:  126nMAssay Description:Inhibition of 100 nM capsaicin effect on intracellular [Ca2+] concentration in HEK293 cells expressing human TRPV1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50170063(CHEMBL414663 | Nonanoic acid 3-bromo-4-hydroxy-5-m...)
Affinity DataIC50:  252nMAssay Description:Inhibition of 100 nM capsaicin effect on intracellular [Ca2+] concentration in HEK293 cells expressing human TRPV1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50170049(CHEMBL190452 | Nonanoic acid 3-ethyl-4-hydroxy-5-m...)
Affinity DataIC50:  355nMAssay Description:Inhibition of 100 nM capsaicin effect on intracellular [Ca2+] concentration in HEK293 cells expressing human TRPV1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50170059(CHEMBL190051 | Nonanoic acid 4-hydroxy-3-methoxy-5...)
Affinity DataIC50:  390nMAssay Description:Inhibition of 100 nM capsaicin effect on intracellular [Ca2+] concentration in HEK293 cells expressing human TRPV1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50170050(CHEMBL191184 | Nonanoic acid 3-chloro-4-hydroxy-5-...)
Affinity DataIC50:  631nMAssay Description:Inhibition of 100 nM capsaicin effect on intracellular [Ca2+] concentration in HEK293 cells expressing human TRPV1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50170048(CHEMBL193046 | Nonanoic acid 3-ethynyl-4-hydroxy-5...)
Affinity DataIC50:  2.74E+3nMAssay Description:Inhibition of 100 nM capsaicin effect on intracellular [Ca2+] concentration in HEK293 cells expressing human TRPV1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50170056(CHEMBL191117 | Nonanoic acid 4-hydroxy-2-iodo-3-me...)
Affinity DataIC50:  3.38E+3nMAssay Description:Inhibition of 100 nM capsaicin effect on intracellular [Ca2+] concentration in HEK293 cells expressing human TRPV1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50170058(7-Hydroxy-8-methoxy-3-nonanoyl-3,4-dihydro-1H-quin...)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of 100 nM capsaicin effect on intracellular [Ca2+] concentration in HEK293 cells expressing human TRPV1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50170055(3-[5-Hydroxy-4-methoxy-2-(nonanoylamino-methyl)-ph...)
Affinity DataIC50:  3.93E+3nMAssay Description:Inhibition of 100 nM capsaicin effect on intracellular [Ca2+] concentration in HEK293 cells expressing human TRPV1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50170052(CHEMBL189913 | Nonanoic acid 2-acetylamino-4-hydro...)
Affinity DataIC50:  9.54E+3nMAssay Description:Inhibition of 100 nM capsaicin effect on intracellular [Ca2+] concentration in HEK293 cells expressing human TRPV1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50170060(CHEMBL426272 | Nonanoic acid 3-acetyl-4-hydroxy-5-...)
Affinity DataIC50:  1.04E+4nMAssay Description:Inhibition of 100 nM capsaicin effect on intracellular [Ca2+] concentration in HEK293 cells expressing human TRPV1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50170057(CHEMBL190663 | Nonanoic acid 4-hydroxy-3-methoxy-2...)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of 100 nM capsaicin effect on intracellular [Ca2+] concentration in HEK293 cells expressing human TRPV1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50170067((2E,4E,6E,8E)-9-(6,6-Dimethyl-cyclohex-1-enyl)-3,7...)
Affinity DataIC50:  1.75E+4nMAssay Description:Inhibition of 100 nM capsaicin effect on intracellular [Ca2+] concentration in HEK293 cells expressing human TRPV1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50170064(CHEMBL191343 | Nonanoic acid [6,2'-dihydroxy-5,3'-...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of 100 nM capsaicin effect on intracellular [Ca2+] concentration in HEK293 cells expressing human TRPV1; (weak agonist activity)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50170051(CHEMBL189961 | Nonanoic acid (6-hydroxy-5-methoxy-...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of 100 nM capsaicin effect on intracellular [Ca2+] concentration in HEK293 cells expressing human TRPV1; (weak agonist activity)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed