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Found 4 Enz. Inhib. hit(s) with all data for entry = 50016960
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50175776(1-ALLYL-5-(2-PHENYLPYRAZOLO[1,5-A]PYRIDIN-3-YL)-1H...)
Affinity DataIC50:  560nMAssay Description:Inhibitory activity against human ERK2More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50175778(1-methyl-5-(2-phenylH-pyrazolo[1,5-a]pyridin-3-yl)...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibitory activity against human ERK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50229978(5-(2-PHENYLPYRAZOLO[1,5-A]PYRIDIN-3-YL)-1H-PYRAZOL...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibitory activity against human ERK2More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50175777(2-(3-amino-5-(2-phenylH-pyrazolo[1,5-a]pyridin-3-y...)
Affinity DataIC50:  5.10E+3nMAssay Description:Inhibitory activity against human ERK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed