Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with all data for entry = 50016987
TargetGlucagon receptor(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50075780(4-[5-(4-Chloro-phenyl)-3-isopropyl-1H-pyrrol-2-yl]...)
Affinity DataIC50:  32nMAssay Description:Antagonist activity against glucagon receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50075782(4-[4-(4-Fluoro-phenyl)-5-pyridin-4-yl-1H-pyrrol-2-...)
Affinity DataIC50:  90nMAssay Description:Inhibitiory activity against Mitogen-activated protein kinase 14, p38-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50071899(4-[5-(4-Chloro-phenyl)-3-(4-fluoro-phenyl)-1H-pyrr...)
Affinity DataIC50:  800nMAssay Description:Antagonist activity against glucagon receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50071899(4-[5-(4-Chloro-phenyl)-3-(4-fluoro-phenyl)-1H-pyrr...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibitiory activity against Mitogen-activated protein kinase 14, p38-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed