Compile Data Set for Download or QSAR
maximum 50k data
Found 68 Enz. Inhib. hit(s) with all data for entry = 50017248
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179600(5-(2-fluorobenzylthio)-1-(5-(methylsulfonyl)pyridi...)
Affinity DataIC50:  40nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179598(1-(5-(methylsulfonyl)pyridin-2-yl)-5-(propylthio)-...)
Affinity DataIC50: <50nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179631(5-(sec-butylthio)-1-(5-(methylsulfonyl)pyridin-2-y...)
Affinity DataIC50: <50nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179609(1-(5-(methylsulfonyl)pyridin-2-yl)-5-(phenylthio)-...)
Affinity DataIC50:  60nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179596(5-(cyclopentylmethoxy)-1-(5-(methylsulfonyl)pyridi...)
Affinity DataIC50:  60nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179611(5-(cycloheptyloxy)-1-(5-(methylsulfonyl)pyridin-2-...)
Affinity DataIC50:  70nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179616(5-(benzylthio)-1-(5-(methylsulfonyl)pyridin-2-yl)-...)
Affinity DataIC50:  80nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179606(5-(cyclobutylmethoxy)-1-(5-(methylsulfonyl)pyridin...)
Affinity DataIC50:  80nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179620(5-((4-methylenecyclohexyl)methoxy)-1-(5-(methylsul...)
Affinity DataIC50: <90nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179591(5-(3-methylbutan-2-yloxy)-1-(5-(methylsulfonyl)pyr...)
Affinity DataIC50:  90nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179602(1-(5-(methylsulfonyl)pyridin-2-yl)-5-(5,6,7,8-tetr...)
Affinity DataIC50:  100nMAssay Description:Inhibition of COX1 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179624(5-(2,3-dimethylphenoxy)-1-(5-(methylsulfonyl)pyrid...)
Affinity DataIC50:  100nMAssay Description:Inhibition of COX1 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179621(5-(cyclohexylthio)-1-(5-(methylsulfonyl)pyridin-2-...)
Affinity DataIC50:  100nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179592(5-isobutoxy-1-(5-(methylsulfonyl)pyridin-2-yl)-3-(...)
Affinity DataIC50:  110nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50176545(3-(difluoromethyl)-5-((2R,6S)-2,6-dimethylmorpholi...)
Affinity DataIC50:  140nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179601(5-(cyclohex-3-enylmethoxy)-1-(5-(methylsulfonyl)py...)
Affinity DataIC50:  140nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179595(5-(3-methylcyclopentyloxy)-1-(5-(methylsulfonyl)py...)
Affinity DataIC50:  160nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179608(5-(2-ethoxyethylthio)-1-(5-(methylsulfonyl)pyridin...)
Affinity DataIC50:  170nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179610(5-(2-methylpentan-3-yloxy)-1-(5-(methylsulfonyl)py...)
Affinity DataIC50:  170nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179624(5-(2,3-dimethylphenoxy)-1-(5-(methylsulfonyl)pyrid...)
Affinity DataIC50:  170nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179609(1-(5-(methylsulfonyl)pyridin-2-yl)-5-(phenylthio)-...)
Affinity DataIC50:  200nMAssay Description:Inhibition of COX1 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179598(1-(5-(methylsulfonyl)pyridin-2-yl)-5-(propylthio)-...)
Affinity DataIC50:  200nMAssay Description:Inhibition of COX1 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179593(5-(2-methylcyclohexyloxy)-1-(5-(methylsulfonyl)pyr...)
Affinity DataIC50:  200nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179625(5-(cyclopentyloxy)-1-(5-(methylsulfonyl)pyridin-2-...)
Affinity DataIC50:  210nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179628(1-(5-(methylsulfonyl)pyridin-2-yl)-5-(pentylthio)-...)
Affinity DataIC50:  300nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50137425(2-(3-(difluoromethyl)-5-phenyl-1H-pyrazol-1-yl)-5-...)
Affinity DataIC50:  310nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179596(5-(cyclopentylmethoxy)-1-(5-(methylsulfonyl)pyridi...)
Affinity DataIC50:  400nMAssay Description:Inhibition of COX1 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179613(5-(4-methylpentylthio)-1-(5-(methylsulfonyl)pyridi...)
Affinity DataIC50:  400nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50024426(CHEMBL204252)
Affinity DataIC50: <500nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179594(5-(methylsulfonyl)-2-(5-(naphthalen-1-ylmethoxy)-3...)
Affinity DataIC50: >500nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179597(2-(5-(cyclopropylmethoxy)-3-(trifluoromethyl)-1H-p...)
Affinity DataIC50: >500nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179599(2-(4-methyl-5-(pentan-3-yloxy)-3-(trifluoromethyl)...)
Affinity DataIC50: >500nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179603(2-(5-(cyclopentyloxy)-3-(trifluoromethyl)-1H-pyraz...)
Affinity DataIC50: >500nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179605(1-(5-(methylsulfonyl)pyridin-2-yl)-5-(pentan-2-ylo...)
Affinity DataIC50: >500nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179607(2-(5-(benzyloxy)-3-(trifluoromethyl)-1H-pyrazol-1-...)
Affinity DataIC50: >500nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179612(2-(5-butoxy-3-(trifluoromethyl)-1H-pyrazol-1-yl)-5...)
Affinity DataIC50: >500nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179614(5-(methylsulfonyl)-2-(5-(pyridin-4-ylmethoxy)-3-(t...)
Affinity DataIC50: >500nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179617(1-(5-(methylsulfonyl)pyridin-2-yl)-5-(tetrahydrofu...)
Affinity DataIC50: >500nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179618(2-(5-isobutoxy-4-methyl-3-(trifluoromethyl)-1H-pyr...)
Affinity DataIC50: >500nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179619(2-(5-isopropoxy-4-methyl-3-(trifluoromethyl)-1H-py...)
Affinity DataIC50: >500nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179623(5-(1-methoxybutan-2-yloxy)-1-(5-(methylsulfonyl)py...)
Affinity DataIC50: >500nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179626(2-(5-(cyclohexyloxy)-3-(trifluoromethyl)-1H-pyrazo...)
Affinity DataIC50: >500nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179629(1-(5-(methylsulfonyl)pyridin-2-yl)-5-phenoxy-3-(tr...)
Affinity DataIC50: >500nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179630(2-(5-(3-fluorobenzyloxy)-3-(trifluoromethyl)-1H-py...)
Affinity DataIC50: >500nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179633(2-(4-chloro-5-isopropoxy-3-(trifluoromethyl)-1H-py...)
Affinity DataIC50: >500nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179632(2-(5-methoxy-3-(trifluoromethyl)-1H-pyrazol-1-yl)-...)
Affinity DataIC50: >500nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179634(2-(5-isopropoxy-3-(trifluoromethyl)-1H-pyrazol-1-y...)
Affinity DataIC50: >500nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179622(5-cyclobutoxy-1-(5-(methylsulfonyl)pyridin-2-yl)-3...)
Affinity DataIC50:  550nMAssay Description:Inhibition of COX2 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179600(5-(2-fluorobenzylthio)-1-(5-(methylsulfonyl)pyridi...)
Affinity DataIC50:  600nMAssay Description:Inhibition of COX1 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Canis familiaris)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179616(5-(benzylthio)-1-(5-(methylsulfonyl)pyridin-2-yl)-...)
Affinity DataIC50:  900nMAssay Description:Inhibition of COX1 by canine whole blood assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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