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Found 18 Enz. Inhib. hit(s) with all data for entry = 50035975
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Rattus norvegicus (Rat))
Laboratoire De Pharmacie Chimique, Facult�

Curated by ChEMBL
LigandPNGBDBM24183(4-amino-n-[2,3-3H]butyric acid | 4-aminobutanoic a...)
Affinity DataIC50:  40nMAssay Description:Inhibition of [3H]baclofen binding to rat gamma-aminobutyric acid type B receptor.More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Rattus norvegicus (Rat))
Laboratoire De Pharmacie Chimique, Facult�

Curated by ChEMBL
LigandPNGBDBM24182(4-amino-3-(4-chlorophenyl)butanoic acid | Baclofen...)
Affinity DataIC50:  330nMAssay Description:Inhibition of [3H]baclofen binding to rat gamma-aminobutyric acid type B receptor.More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Rattus norvegicus (Rat))
Laboratoire De Pharmacie Chimique, Facult�

Curated by ChEMBL
LigandPNGBDBM24182(4-amino-3-(4-chlorophenyl)butanoic acid | Baclofen...)
Affinity DataIC50:  330nMAssay Description:Inhibition of [3H]baclofen binding to rat gamma-aminobutyric acid type B receptor.More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Rattus norvegicus (Rat))
Laboratoire De Pharmacie Chimique, Facult�

Curated by ChEMBL
LigandPNGBDBM50007118(4-Amino-3-(5-chloro-thiophen-2-yl)-butyric acid | ...)
Affinity DataIC50:  610nMAssay Description:Inhibition of [3H]baclofen binding to rat gamma-aminobutyric acid type B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Rattus norvegicus (Rat))
Laboratoire De Pharmacie Chimique, Facult�

Curated by ChEMBL
LigandPNGBDBM50007121(4-Amino-3-(2-chloro-phenyl)-butyric acid | CHEMBL8...)
Affinity DataIC50:  800nMAssay Description:Inhibition of [3H]baclofen binding to rat gamma-aminobutyric acid type B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Rattus norvegicus (Rat))
Laboratoire De Pharmacie Chimique, Facult�

Curated by ChEMBL
LigandPNGBDBM50368295(CHEMBL301492)
Affinity DataIC50:  1.33E+3nMAssay Description:Inhibition of [3H]baclofen binding to rat gamma-aminobutyric acid type B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Rattus norvegicus (Rat))
Laboratoire De Pharmacie Chimique, Facult�

Curated by ChEMBL
LigandPNGBDBM50007107(4-Amino-3-(5-methyl-thiophen-2-yl)-butyric acid | ...)
Affinity DataIC50:  1.34E+3nMAssay Description:Inhibition of [3H]baclofen binding to rat gamma-aminobutyric acid type B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Rattus norvegicus (Rat))
Laboratoire De Pharmacie Chimique, Facult�

Curated by ChEMBL
LigandPNGBDBM50007108(4-Amino-3-(5-bromo-thiophen-2-yl)-butyric acid | C...)
Affinity DataIC50:  1.86E+3nMAssay Description:Inhibition of [3H]baclofen binding to rat gamma-aminobutyric acid type B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Rattus norvegicus (Rat))
Laboratoire De Pharmacie Chimique, Facult�

Curated by ChEMBL
LigandPNGBDBM50007117(4-Amino-3-thiophen-2-yl-butyric acid | CHEMBL31547...)
Affinity DataIC50:  9.72E+3nMAssay Description:Inhibition of [3H]baclofen binding to rat gamma-aminobutyric acid type B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Rattus norvegicus (Rat))
Laboratoire De Pharmacie Chimique, Facult�

Curated by ChEMBL
LigandPNGBDBM50007109(4-Amino-3-(3-chloro-phenyl)-butyric acid | CHEMBL3...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of [3H]baclofen binding to rat gamma-aminobutyric acid type B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Rattus norvegicus (Rat))
Laboratoire De Pharmacie Chimique, Facult�

Curated by ChEMBL
LigandPNGBDBM50007113(4-Amino-3-thiophen-3-yl-butyric acid | CHEMBL87856)
Affinity DataIC50:  2.09E+4nMAssay Description:Inhibition of [3H]baclofen binding to rat gamma-aminobutyric acid type B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Rattus norvegicus (Rat))
Laboratoire De Pharmacie Chimique, Facult�

Curated by ChEMBL
LigandPNGBDBM50007110(4-Amino-3-(4-bromo-thiophen-2-yl)-butyric acid | C...)
Affinity DataIC50:  3.91E+4nMAssay Description:Inhibition of [3H]baclofen binding to rat gamma-aminobutyric acid type B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Rattus norvegicus (Rat))
Laboratoire De Pharmacie Chimique, Facult�

Curated by ChEMBL
LigandPNGBDBM50007111(4-Amino-3-(4-chloro-thiophen-2-yl)-butyric acid | ...)
Affinity DataIC50:  4.53E+4nMAssay Description:Inhibition of [3H]baclofen binding to rat gamma-aminobutyric acid type B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Rattus norvegicus (Rat))
Laboratoire De Pharmacie Chimique, Facult�

Curated by ChEMBL
LigandPNGBDBM50007114(4-Amino-3-furan-2-yl-butyric acid | CHEMBL85880)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of [3H]baclofen binding to rat gamma-aminobutyric acid type B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Rattus norvegicus (Rat))
Laboratoire De Pharmacie Chimique, Facult�

Curated by ChEMBL
LigandPNGBDBM50007119(4-Amino-3-phenyl-butyric acid | CHEMBL53073)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of [3H]baclofen binding to rat gamma-aminobutyric acid type B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Rattus norvegicus (Rat))
Laboratoire De Pharmacie Chimique, Facult�

Curated by ChEMBL
LigandPNGBDBM50007112(4-Amino-3-(5-methyl-furan-2-yl)-butyric acid | CHE...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of [3H]baclofen binding to rat gamma-aminobutyric acid type B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Rattus norvegicus (Rat))
Laboratoire De Pharmacie Chimique, Facult�

Curated by ChEMBL
LigandPNGBDBM50007120(4-Amino-3-(4-hydroxy-phenyl)-butyric acid | CHEMBL...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of [3H]baclofen binding to rat gamma-aminobutyric acid type B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Rattus norvegicus (Rat))
Laboratoire De Pharmacie Chimique, Facult�

Curated by ChEMBL
LigandPNGBDBM50007116(4-Amino-3-(3-methyl-thiophen-2-yl)-butyric acid | ...)
Affinity DataIC50:  1.24E+5nMAssay Description:Inhibition of [3H]baclofen binding to rat gamma-aminobutyric acid type B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed