Compile Data Set for Download or QSAR
maximum 50k data
Found 81 Enz. Inhib. hit(s) with all data for entry = 50017618
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184650(CHEMBL381066 | [4-(4,4''-bis-trifluoromethoxy-[1,1...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effect on human PPARdelta transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184651(CHEMBL377093 | {4-[4,6-bis-(4-trifluoromethyl-phen...)
Affinity DataEC50:  40nMAssay Description:Effect on human PPARdelta transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184652(CHEMBL210469 | [4-(4,4''-Bis-trifluoromethyl-[1,1'...)
Affinity DataEC50:  3.33E+3nMAssay Description:Effect on human PPARalpha transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184653(CHEMBL210873 | [4-(4,4''-bis-dimethylamino-[1,1';3...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effect on human PPARgamma transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184650(CHEMBL381066 | [4-(4,4''-bis-trifluoromethoxy-[1,1...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effect on human PPARgamma transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184654(CHEMBL383313 | {4-[2,6-bis-(4-trifluoromethyl-phen...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effect on human PPARalpha transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184655(CHEMBL207887 | [4-(3,4''-bis-trifluoromethyl-[1,1'...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effect on human PPARgamma transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184654(CHEMBL383313 | {4-[2,6-bis-(4-trifluoromethyl-phen...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effect on human PPARgamma transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184656(CHEMBL208755 | {4-[5,6-bis-(4-trifluoromethyl-phen...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effect on human PPARdelta transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184657(CHEMBL207198 | [4-(4,4''-bis-trifluoromethyl-[1,1'...)
Affinity DataEC50:  110nMAssay Description:Effect on human PPARdelta transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184658(CHEMBL208202 | [2-methyl-4-(4'''-trifluoromethyl-[...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effect on human PPARgamma transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184659(CHEMBL208203 | {4-[4,6-bis-(4-trifluoromethoxy-phe...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effect on human PPARalpha transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184657(CHEMBL207198 | [4-(4,4''-bis-trifluoromethyl-[1,1'...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effect on human PPARgamma transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184660(2-[4-(4,4''-bis-trifluoromethyl-[1,1';3',1'']terph...)
Affinity DataEC50:  370nMAssay Description:Effect on human PPARgamma transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184656(CHEMBL208755 | {4-[5,6-bis-(4-trifluoromethyl-phen...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effect on human PPARalpha transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184661(CHEMBL207811 | {4-[2,6-bis-(4-trifluoromethoxy-phe...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effect on human PPARalpha transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184659(CHEMBL208203 | {4-[4,6-bis-(4-trifluoromethoxy-phe...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effect on human PPARgamma transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184664(CHEMBL425945 | [2-methyl-4-(4-methyl-4''-trifluoro...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effect on human PPARgamma transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184665(CHEMBL377883 | [2-methyl-4-(4-trifluoromethoxy-4''...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effect on human PPARgamma transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184662(CHEMBL206578 | {4-[4,6-bis-(4-methoxy-phenyl)-pyri...)
Affinity DataEC50:  110nMAssay Description:Effect on human PPARdelta transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184663(CHEMBL206895 | [4-(4,4''-bis-trifluoromethyl-[1,1'...)
Affinity DataEC50:  540nMAssay Description:Effect on human PPARdelta transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184666(CHEMBL379123 | [4-([1,1';3',1'']terphenyl-5'-ylmet...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effect on human PPARalpha transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184658(CHEMBL208202 | [2-methyl-4-(4'''-trifluoromethyl-[...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effect on human PPARalpha transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184667(CHEMBL207957 | [4-(4,4''-dimethoxy-[1,1';2',1'']te...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effect on human PPARalpha transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184668(CHEMBL377695 | [4-(4,4''-dichloro-[1,1';3',1'']ter...)
Affinity DataEC50:  110nMAssay Description:Effect on human PPARdelta transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184655(CHEMBL207887 | [4-(3,4''-bis-trifluoromethyl-[1,1'...)
Affinity DataEC50:  560nMAssay Description:Effect on human PPARdelta transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184663(CHEMBL206895 | [4-(4,4''-bis-trifluoromethyl-[1,1'...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effect on human PPARalpha transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184660(2-[4-(4,4''-bis-trifluoromethyl-[1,1';3',1'']terph...)
Affinity DataEC50:  730nMAssay Description:Effect on human PPARalpha transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184659(CHEMBL208203 | {4-[4,6-bis-(4-trifluoromethoxy-phe...)
Affinity DataEC50:  90nMAssay Description:Effect on human PPARdelta transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184670(CHEMBL379851 | [4-(4,4''-bis-trifluoromethyl-[1,1'...)
Affinity DataEC50:  70nMAssay Description:Effect on human PPARdelta transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184669(CHEMBL379145 | [4-(4,4''-bis-trifluoromethyl-[1,1'...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effect on human PPARalpha transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184655(CHEMBL207887 | [4-(3,4''-bis-trifluoromethyl-[1,1'...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effect on human PPARalpha transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184651(CHEMBL377093 | {4-[4,6-bis-(4-trifluoromethyl-phen...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effect on human PPARgamma transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184670(CHEMBL379851 | [4-(4,4''-bis-trifluoromethyl-[1,1'...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effect on human PPARalpha transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184660(2-[4-(4,4''-bis-trifluoromethyl-[1,1';3',1'']terph...)
Affinity DataEC50:  50nMAssay Description:Effect on human PPARdelta transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184673(CHEMBL207449 | [4-(4,4''-bis-trifluoromethyl-[1,1'...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effect on human PPARalpha transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184665(CHEMBL377883 | [2-methyl-4-(4-trifluoromethoxy-4''...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effect on human PPARalpha transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184672(CHEMBL208318 | [4-(4,4''-bis-trifluoromethoxy-[1,1...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effect on human PPARalpha transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184656(CHEMBL208755 | {4-[5,6-bis-(4-trifluoromethyl-phen...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effect on human PPARgamma transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184674(CHEMBL383404 | [4-(4-methoxy-4''-trifluoromethyl-[...)
Affinity DataEC50:  70nMAssay Description:Effect on human PPARdelta transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184668(CHEMBL377695 | [4-(4,4''-dichloro-[1,1';3',1'']ter...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effect on human PPARgamma transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184661(CHEMBL207811 | {4-[2,6-bis-(4-trifluoromethoxy-phe...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effect on human PPARgamma transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184650(CHEMBL381066 | [4-(4,4''-bis-trifluoromethoxy-[1,1...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effect on human PPARalpha transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184671(CHEMBL211047 | [4-(4,4''-dimethoxy-[1,1';3',1'']te...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effect on human PPARalpha transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184673(CHEMBL207449 | [4-(4,4''-bis-trifluoromethyl-[1,1'...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effect on human PPARgamma transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184664(CHEMBL425945 | [2-methyl-4-(4-methyl-4''-trifluoro...)
Affinity DataEC50:  70nMAssay Description:Effect on human PPARdelta transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184669(CHEMBL379145 | [4-(4,4''-bis-trifluoromethyl-[1,1'...)
Affinity DataEC50:  160nMAssay Description:Effect on human PPARdelta transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184666(CHEMBL379123 | [4-([1,1';3',1'']terphenyl-5'-ylmet...)
Affinity DataEC50:  970nMAssay Description:Effect on human PPARdelta transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184665(CHEMBL377883 | [2-methyl-4-(4-trifluoromethoxy-4''...)
Affinity DataEC50:  60nMAssay Description:Effect on human PPARdelta transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184668(CHEMBL377695 | [4-(4,4''-dichloro-[1,1';3',1'']ter...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effect on human PPARalpha transactivation in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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