Compile Data Set for Download or QSAR
maximum 50k data
Found 21 Enz. Inhib. hit(s) with all data for entry = 2431
LigandPNGBDBM20490(1-(2-bromophenyl)-3-[2-(2,3-dihydro-1H-indol-1-yl)...)
Affinity DataEC50:  158nMpH: 7.2 T: 2°CAssay Description:One day before the assay was performed, human TRPV1 expressed in 1321N1 astrocytoma cells were plated onto 96-well assay plates and grown until 2.5 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM20509(1-(2-bromophenyl)-3-[(3R)-1-(5-methylpyridin-2-yl)...)
Affinity DataEC50: >200nMpH: 7.2 T: 2°CAssay Description:One day before the assay was performed, human TRPV1 expressed in 1321N1 astrocytoma cells were plated onto 96-well assay plates and grown until 2.5 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM20492(1-(2-bromophenyl)-3-[2-(5-methyl-2,3-dihydro-1H-in...)
Affinity DataEC50:  50nMpH: 7.2 T: 2°CAssay Description:One day before the assay was performed, human TRPV1 expressed in 1321N1 astrocytoma cells were plated onto 96-well assay plates and grown until 2.5 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM20493(1-(2-bromophenyl)-3-[2-(4-fluoro-2,3-dihydro-1H-in...)
Affinity DataEC50:  40nMpH: 7.2 T: 2°CAssay Description:One day before the assay was performed, human TRPV1 expressed in 1321N1 astrocytoma cells were plated onto 96-well assay plates and grown until 2.5 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM20494(1-(2-bromophenyl)-3-[2-(5-fluoro-2,3-dihydro-1H-in...)
Affinity DataEC50:  79nMpH: 7.2 T: 2°CAssay Description:One day before the assay was performed, human TRPV1 expressed in 1321N1 astrocytoma cells were plated onto 96-well assay plates and grown until 2.5 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM20495(3-(2-bromophenyl)-1-[2-(6-methyl-1,2,3,4-tetrahydr...)
Affinity DataEC50:  40nMpH: 7.2 T: 2°CAssay Description:One day before the assay was performed, human TRPV1 expressed in 1321N1 astrocytoma cells were plated onto 96-well assay plates and grown until 2.5 h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM20468(3-(2-bromophenyl)-1-{2-[ethyl(3-methylphenyl)amino...)
Affinity DataEC50:  16nMpH: 7.2 T: 2°CAssay Description:One day before the assay was performed, human TRPV1 expressed in 1321N1 astrocytoma cells were plated onto 96-well assay plates and grown until 2.5 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM20496(1-(2-bromophenyl)-3-[(3S)-1-(3-methylphenyl)pyrrol...)
Affinity DataEC50: >158nMpH: 7.2 T: 2°CAssay Description:One day before the assay was performed, human TRPV1 expressed in 1321N1 astrocytoma cells were plated onto 96-well assay plates and grown until 2.5 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM20497(1-(2-bromophenyl)-3-[(3R)-1-(3-methylphenyl)pyrrol...)
Affinity DataEC50:  20nMpH: 7.2 T: 2°CAssay Description:One day before the assay was performed, human TRPV1 expressed in 1321N1 astrocytoma cells were plated onto 96-well assay plates and grown until 2.5 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM20498(1-(2-bromophenyl)-3-[(3R)-1-(3-fluorophenyl)pyrrol...)
Affinity DataEC50:  16nMpH: 7.2 T: 2°CAssay Description:One day before the assay was performed, human TRPV1 expressed in 1321N1 astrocytoma cells were plated onto 96-well assay plates and grown until 2.5 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM20499(1-(2-bromophenyl)-3-[(3R)-1-(3,4-difluorophenyl)py...)
Affinity DataEC50:  8nMpH: 7.2 T: 2°CAssay Description:One day before the assay was performed, human TRPV1 expressed in 1321N1 astrocytoma cells were plated onto 96-well assay plates and grown until 2.5 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM20500(1-(2-bromophenyl)-3-[(3R)-1-(3-fluoro-4-methylphen...)
Affinity DataEC50:  5nMpH: 7.2 T: 2°CAssay Description:One day before the assay was performed, human TRPV1 expressed in 1321N1 astrocytoma cells were plated onto 96-well assay plates and grown until 2.5 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM20501(1-(2-bromophenyl)-3-[(3R)-1-(pyridin-2-yl)pyrrolid...)
Affinity DataEC50: >251nMpH: 7.2 T: 2°CAssay Description:One day before the assay was performed, human TRPV1 expressed in 1321N1 astrocytoma cells were plated onto 96-well assay plates and grown until 2.5 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM20502(1-(2-bromophenyl)-3-[(3R)-1-[3-(trifluoromethyl)py...)
Affinity DataEC50:  79nMpH: 7.2 T: 2°CAssay Description:One day before the assay was performed, human TRPV1 expressed in 1321N1 astrocytoma cells were plated onto 96-well assay plates and grown until 2.5 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM20503(1-(2-bromophenyl)-3-[(3R)-1-[4-(trifluoromethyl)py...)
Affinity DataEC50:  126nMpH: 7.2 T: 2°CAssay Description:One day before the assay was performed, human TRPV1 expressed in 1321N1 astrocytoma cells were plated onto 96-well assay plates and grown until 2.5 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM20504(1-(2-bromophenyl)-3-[(3R)-1-[5-(trifluoromethyl)py...)
Affinity DataEC50:  32nMpH: 7.2 T: 2°CAssay Description:One day before the assay was performed, human TRPV1 expressed in 1321N1 astrocytoma cells were plated onto 96-well assay plates and grown until 2.5 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM20505(1-(2-bromophenyl)-3-[(3R)-1-[6-(trifluoromethyl)py...)
Affinity DataEC50:  63nMpH: 7.2 T: 2°CAssay Description:One day before the assay was performed, human TRPV1 expressed in 1321N1 astrocytoma cells were plated onto 96-well assay plates and grown until 2.5 h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM20506(1-(2-bromophenyl)-3-[(3R)-1-(5-bromopyridin-2-yl)p...)
Affinity DataEC50:  63nMpH: 7.2 T: 2°CAssay Description:One day before the assay was performed, human TRPV1 expressed in 1321N1 astrocytoma cells were plated onto 96-well assay plates and grown until 2.5 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM20507(1-(2-bromophenyl)-3-[(3R)-1-(5-chloropyridin-2-yl)...)
Affinity DataEC50:  50nMpH: 7.2 T: 2°CAssay Description:One day before the assay was performed, human TRPV1 expressed in 1321N1 astrocytoma cells were plated onto 96-well assay plates and grown until 2.5 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM20508(1-(2-bromophenyl)-3-[(3R)-1-(5-cyanopyridin-2-yl)p...)
Affinity DataEC50:  200nMpH: 7.2 T: 2°CAssay Description:One day before the assay was performed, human TRPV1 expressed in 1321N1 astrocytoma cells were plated onto 96-well assay plates and grown until 2.5 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM20491(1-(2-bromophenyl)-3-[2-(4-methyl-2,3-dihydro-1H-in...)
Affinity DataEC50:  40nMpH: 7.2 T: 2°CAssay Description:One day before the assay was performed, human TRPV1 expressed in 1321N1 astrocytoma cells were plated onto 96-well assay plates and grown until 2.5 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed