Compile Data Set for Download or QSAR
maximum 50k data
Found 13 Enz. Inhib. hit(s) with all data for entry = 50017734
TargetProtein kinase C eta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50185931(8-Octyl-benzolactam-V9 | CHEMBL206866)
Affinity DataKi:  144nMAssay Description:Displacement of [3H]phorbol 12,13-dibutyrate from PKC eta-C1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50185931(8-Octyl-benzolactam-V9 | CHEMBL206866)
Affinity DataKi:  216nMAssay Description:Displacement of [3H]phorbol 12,13-dibutyrate from PKC delta-C1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50185931(8-Octyl-benzolactam-V9 | CHEMBL206866)
Affinity DataKi:  290nMAssay Description:Displacement of [3H]phorbol 12,13-dibutyrate from PKC theta-C1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50185931(8-Octyl-benzolactam-V9 | CHEMBL206866)
Affinity DataKi:  510nMAssay Description:Displacement of [3H]phorbol 12,13-dibutyrate from PKC epsilon-C1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50185931(8-Octyl-benzolactam-V9 | CHEMBL206866)
Affinity DataKi:  5.20E+3nMAssay Description:Displacement of [3H]phorbol 12,13-dibutyrate from PKC gamma-C1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50185931(8-Octyl-benzolactam-V9 | CHEMBL206866)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]phorbol 12,13-dibutyrate from PKC beta-C1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50185931(8-Octyl-benzolactam-V9 | CHEMBL206866)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]phorbol 12,13-dibutyrate from PKC beta-C1AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50185931(8-Octyl-benzolactam-V9 | CHEMBL206866)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]phorbol 12,13-dibutyrate from PKC alpha-C1AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50185931(8-Octyl-benzolactam-V9 | CHEMBL206866)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]phorbol 12,13-dibutyrate from PKC delta-C1AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50185931(8-Octyl-benzolactam-V9 | CHEMBL206866)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]phorbol 12,13-dibutyrate from PKC gamma-C1AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50185931(8-Octyl-benzolactam-V9 | CHEMBL206866)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]phorbol 12,13-dibutyrate from PKC alpha-C1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50185931(8-Octyl-benzolactam-V9 | CHEMBL206866)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]phorbol 12,13-dibutyrate from PKC epsilon-C1AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50185931(8-Octyl-benzolactam-V9 | CHEMBL206866)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]phorbol 12,13-dibutyrate from PKC eta-C1AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed