Compile Data Set for Download or QSAR
maximum 50k data
Found 17 Enz. Inhib. hit(s) with all data for entry = 50017809
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186863(CHEMBL379497 | N-((R)-3-(4-chlorophenyl)-1-(4-(1-c...)
Affinity DataKi:  5nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human MC4 receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186868(CHEMBL213340 | N-{(R)-1-(4-chloro-benzyl)-2-[4-(4-...)
Affinity DataKi:  6.80nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human MC4 receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186874(CHEMBL376999 | N-{(R)-1-(4-chloro-benzyl)-2-[4-(4-...)
Affinity DataKi:  13nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human MC4 receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186862(CHEMBL211260 | N-{(R)-1-(4-chloro-benzyl)-2-[4-(4-...)
Affinity DataKi:  13nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human MC4 receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186865(CHEMBL211202 | N-{(R)-1-(4-chloro-benzyl)-2-[4-(1-...)
Affinity DataKi:  16nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human MC4 receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186869(CHEMBL375388 | N-{(R)-1-(4-chloro-benzyl)-2-[4-(4-...)
Affinity DataKi:  27nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human MC4 receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186861(CHEMBL213940 | N-{(R)-1-(4-chloro-benzyl)-2-[4-(4-...)
Affinity DataKi:  31nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human MC4 receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186864(CHEMBL373735 | N-[(R)-2-[4-(1-acetyl-4-isobutyl-pi...)
Affinity DataKi:  38nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human MC4 receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186871(CHEMBL211032 | N-{(R)-1-(4-chloro-benzyl)-2-[4-(4-...)
Affinity DataKi:  42nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human MC4 receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186867(CHEMBL378415 | N-[(R)-2-[4-(4-benzyl-1-methyl-pipe...)
Affinity DataKi:  44nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human MC4 receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186875(CHEMBL375389 | N-{(R)-1-(4-chloro-benzyl)-2-[4-(1-...)
Affinity DataKi:  47nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human MC4 receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186859(CHEMBL211475 | N-{(R)-1-(4-chloro-benzyl)-2-[4-(4-...)
Affinity DataKi:  68nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human MC4 receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186860(CHEMBL210922 | N-{(R)-1-(4-chloro-benzyl)-2-[4-(4-...)
Affinity DataKi:  70nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human MC4 receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186866(CHEMBL211792 | N-{(R)-1-(4-chloro-benzyl)-2-[4-(4-...)
Affinity DataKi:  76nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human MC4 receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186873(CHEMBL209417 | N-{(R)-1-(4-chloro-benzyl)-2-[4-(4-...)
Affinity DataKi:  101nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human MC4 receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186872(CHEMBL376936 | N-{(R)-1-(4-chloro-benzyl)-2-[4-(1-...)
Affinity DataKi:  215nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human MC4 receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50186870(CHEMBL208953 | N-{(R)-1-(4-chloro-benzyl)-2-[4-(4-...)
Affinity DataKi:  370nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human MC4 receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed