TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Novartis Research Foundation
Curated by ChEMBL
Novartis Research Foundation
Curated by ChEMBL
Affinity DataKi: 37nMAssay Description:Inhibition of unphosporylated AblMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Novartis Research Foundation
Curated by ChEMBL
Novartis Research Foundation
Curated by ChEMBL
Affinity DataKi: 7.00E+3nMAssay Description:Inhibition of phosporylated AblMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Novartis Research Foundation
Curated by ChEMBL
Novartis Research Foundation
Curated by ChEMBL
Affinity DataIC50: 0.900nMAssay Description:Inhibition of VEGFR-2 kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: <1nMAssay Description:Inhibition of Aurora A kinaseMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Novartis Research Foundation
Curated by ChEMBL
Novartis Research Foundation
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of VEGFR-2 kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of Aurora B kinaseMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Novartis Research Foundation
Curated by ChEMBL
Novartis Research Foundation
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of Tie2 kinaseMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Novartis Research Foundation
Curated by ChEMBL
Novartis Research Foundation
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of VEGFR-3 kinaseMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Novartis Research Foundation
Curated by ChEMBL
Novartis Research Foundation
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of B-Raf kinaseMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Novartis Research Foundation
Curated by ChEMBL
Novartis Research Foundation
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Inhibition of VEGFR-2 kinaseMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Novartis Research Foundation
Curated by ChEMBL
Novartis Research Foundation
Curated by ChEMBL
Affinity DataIC50: 39nMAssay Description:Inhibition of p38alpha kinaseMore data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Novartis Research Foundation
Curated by ChEMBL
Novartis Research Foundation
Curated by ChEMBL
Affinity DataIC50: 57nMAssay Description:Inhibition of PDGFRbeta kinaseMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Novartis Research Foundation
Curated by ChEMBL
Novartis Research Foundation
Curated by ChEMBL
Affinity DataIC50: 58nMAssay Description:Inhibition of Flt3 kinaseMore data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
Novartis Research Foundation
Curated by ChEMBL
Novartis Research Foundation
Curated by ChEMBL
Affinity DataIC50: 67nMAssay Description:Inhibition of PDGFRalpha kinaseMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Novartis Research Foundation
Curated by ChEMBL
Novartis Research Foundation
Curated by ChEMBL
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Novartis Research Foundation
Curated by ChEMBL
Novartis Research Foundation
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Inhibition of c-Raf kinaseMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Novartis Research Foundation
Curated by ChEMBL
Novartis Research Foundation
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Inhibition of VEGFR-2 kinaseMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
Novartis Research Foundation
Curated by ChEMBL
Novartis Research Foundation
Curated by ChEMBL
Affinity DataIC50: 98nMAssay Description:Inhibition of JNK2alpha2 kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibition of Tie2 kinaseMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Novartis Research Foundation
Curated by ChEMBL
Novartis Research Foundation
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of VEGFR-1 kinaseMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Novartis Research Foundation
Curated by ChEMBL
Novartis Research Foundation
Curated by ChEMBL
Affinity DataIC50: 188nMAssay Description:Inhibition of Abl kinaseMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Novartis Research Foundation
Curated by ChEMBL
Novartis Research Foundation
Curated by ChEMBL
Affinity DataIC50: 340nMAssay Description:Inhibition of p38alpha kinaseMore data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Novartis Research Foundation
Curated by ChEMBL
Novartis Research Foundation
Curated by ChEMBL
Affinity DataIC50: 386nMAssay Description:Inhibition of PDGFRbeta kinaseMore data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Novartis Research Foundation
Curated by ChEMBL
Novartis Research Foundation
Curated by ChEMBL
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Novartis Research Foundation
Curated by ChEMBL
Novartis Research Foundation
Curated by ChEMBL
Affinity DataIC50: 580nMAssay Description:Inhibition of FGFR-1 kinaseMore data for this Ligand-Target Pair
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Novartis Research Foundation
Curated by ChEMBL
Novartis Research Foundation
Curated by ChEMBL
Affinity DataIC50: 695nMAssay Description:Inhibition of c-Raf kinaseMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Novartis Research Foundation
Curated by ChEMBL
Novartis Research Foundation
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of EGFR kinaseMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Novartis Research Foundation
Curated by ChEMBL
Novartis Research Foundation
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of p38alpha kinaseMore data for this Ligand-Target Pair
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Novartis Research Foundation
Curated by ChEMBL
Novartis Research Foundation
Curated by ChEMBL
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of c-Raf kinaseMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Novartis Research Foundation
Curated by ChEMBL
Novartis Research Foundation
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Syk kinaseMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
Novartis Research Foundation
Curated by ChEMBL
Novartis Research Foundation
Curated by ChEMBL
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of Fyn kinaseMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Novartis Research Foundation
Curated by ChEMBL
Novartis Research Foundation
Curated by ChEMBL
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of Lck kinaseMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Novartis Research Foundation
Curated by ChEMBL
Novartis Research Foundation
Curated by ChEMBL
Affinity DataKd: 1.16E+3nMAssay Description:Inhibition of p38alpha kinaseMore data for this Ligand-Target Pair