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Found 31 Enz. Inhib. hit(s) with all data for entry = 50018002
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189833((S)-N-butyl-3-((S)-2-(4-fluorophenylsulfonamido)-3...)
Affinity DataIC50:  21nMAssay Description:Inhibition of human erythrocyte mu calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-2 catalytic subunit(Sus scrofa)
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189833((S)-N-butyl-3-((S)-2-(4-fluorophenylsulfonamido)-3...)
Affinity DataIC50:  21nMAssay Description:Inhibition of porcein kidney m calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114340((S)-2-(4-Fluoro-benzenesulfonylamino)-N-((S)-1-for...)
Affinity DataIC50:  22nMAssay Description:Inhibition of human erythrocyte mu calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-2 catalytic subunit(Sus scrofa)
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114340((S)-2-(4-Fluoro-benzenesulfonylamino)-N-((S)-1-for...)
Affinity DataIC50:  49nMAssay Description:Inhibition of porcein kidney m calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189828(1-((S)-1-((3S)-2-hydroxy-tetrahydrofuran-3-ylamino...)
Affinity DataIC50:  86nMAssay Description:Inhibition of human erythrocyte mu calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-2 catalytic subunit(Sus scrofa)
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189825((2S)-2-((((4-cyanophenyl)amino)thioxomethyl)amino)...)
Affinity DataIC50:  120nMAssay Description:Inhibition of porcein kidney m calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189825((2S)-2-((((4-cyanophenyl)amino)thioxomethyl)amino)...)
Affinity DataIC50:  140nMAssay Description:Inhibition of human erythrocyte mu calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189822((2S)-2-((benzylamino)thioxomethyl)amino)-4-methyl-...)
Affinity DataIC50:  150nMAssay Description:Inhibition of human erythrocyte mu calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189835((2S)-2-((((4-fluorophenyl)amino)thioxomethyl)amino...)
Affinity DataIC50:  150nMAssay Description:Inhibition of human erythrocyte mu calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-2 catalytic subunit(Sus scrofa)
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189832((2S)-4-methyl-2-((((4-methylphenyl)amino)thioxomet...)
Affinity DataIC50:  170nMAssay Description:Inhibition of porcein kidney m calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-2 catalytic subunit(Sus scrofa)
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189834((2S)-2-((((3-cyanophenyl)amino)thioxomethyl)amino)...)
Affinity DataIC50:  170nMAssay Description:Inhibition of porcein kidney m calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189831((2S)-4-methyl-2-((((3-methylphenyl)amino)thioxomet...)
Affinity DataIC50:  180nMAssay Description:Inhibition of human erythrocyte mu calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-2 catalytic subunit(Sus scrofa)
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189835((2S)-2-((((4-fluorophenyl)amino)thioxomethyl)amino...)
Affinity DataIC50:  190nMAssay Description:Inhibition of porcein kidney m calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-2 catalytic subunit(Sus scrofa)
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189828(1-((S)-1-((3S)-2-hydroxy-tetrahydrofuran-3-ylamino...)
Affinity DataIC50:  190nMAssay Description:Inhibition of porcein kidney m calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-2 catalytic subunit(Sus scrofa)
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189827((2S)-2-((((4-methoxyphenyl)amino)thioxomethyl)amin...)
Affinity DataIC50:  200nMAssay Description:Inhibition of porcein kidney m calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189827((2S)-2-((((4-methoxyphenyl)amino)thioxomethyl)amin...)
Affinity DataIC50:  220nMAssay Description:Inhibition of human erythrocyte mu calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-2 catalytic subunit(Sus scrofa)
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189822((2S)-2-((benzylamino)thioxomethyl)amino)-4-methyl-...)
Affinity DataIC50:  240nMAssay Description:Inhibition of porcein kidney m calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189830((2S)-4-methyl-2-((((2-methylphenyl)amino)thioxomet...)
Affinity DataIC50:  240nMAssay Description:Inhibition of human erythrocyte mu calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-2 catalytic subunit(Sus scrofa)
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189830((2S)-4-methyl-2-((((2-methylphenyl)amino)thioxomet...)
Affinity DataIC50:  250nMAssay Description:Inhibition of porcein kidney m calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189834((2S)-2-((((3-cyanophenyl)amino)thioxomethyl)amino)...)
Affinity DataIC50:  260nMAssay Description:Inhibition of human erythrocyte mu calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-2 catalytic subunit(Sus scrofa)
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189831((2S)-4-methyl-2-((((3-methylphenyl)amino)thioxomet...)
Affinity DataIC50:  340nMAssay Description:Inhibition of porcein kidney m calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114342((E)-2-(dimethylamino)-N'-((S)-2-((S)-2-(4-fluoroph...)
Affinity DataIC50:  370nMAssay Description:Inhibition of human erythrocyte mu calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189823((2S,3S)-3-methyl-2-(((phenylamino)thioxomethyl)ami...)
Affinity DataIC50:  600nMAssay Description:Inhibition of human erythrocyte mu calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189829((2S)-3-methyl-2-(((phenylamino)thioxomethyl)amino)...)
Affinity DataIC50:  630nMAssay Description:Inhibition of human erythrocyte mu calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189826((S)-2-(4-fluorophenylsulfonamido)-N-((3S)-2-hydrox...)
Affinity DataIC50:  880nMAssay Description:Inhibition of human erythrocyte mu calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189832((2S)-4-methyl-2-((((4-methylphenyl)amino)thioxomet...)
Affinity DataIC50:  910nMAssay Description:Inhibition of human erythrocyte mu calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-2 catalytic subunit(Sus scrofa)
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189823((2S,3S)-3-methyl-2-(((phenylamino)thioxomethyl)ami...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of porcein kidney m calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-2 catalytic subunit(Sus scrofa)
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189829((2S)-3-methyl-2-(((phenylamino)thioxomethyl)amino)...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of porcein kidney m calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-2 catalytic subunit(Sus scrofa)
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189826((S)-2-(4-fluorophenylsulfonamido)-N-((3S)-2-hydrox...)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of porcein kidney m calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189824(CHEMBL206737 | N-(1-cyano-3-methylbutyl)-2-((4-flu...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human erythrocyte mu calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-2 catalytic subunit(Sus scrofa)
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189824(CHEMBL206737 | N-(1-cyano-3-methylbutyl)-2-((4-flu...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of porcein kidney m calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed