Compile Data Set for Download or QSAR
maximum 50k data
Found 30 Enz. Inhib. hit(s) with all data for entry = 50018101
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50191271((4R,7S,10S,13R,16S,19R)-13-((1H-indol-3-yl)methyl)...)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of [125I](Leu8,DTrp22,Tyr25)-SRIF28 binding to human sst2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50191271((4R,7S,10S,13R,16S,19R)-13-((1H-indol-3-yl)methyl)...)
Affinity DataIC50:  2.70nMAssay Description:Inhibition of [125I](Leu8,DTrp22,Tyr25)-SRIF28 binding to human sst5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50191270(CHEMBL436892 | H2N-CO-DPhe-c[Cys-Aph(CONHOCH3)-DTr...)
Affinity DataIC50:  3.10nMAssay Description:Inhibition of [125I](Leu8,DTrp22,Tyr25)-SRIF28 binding to human sst2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50191267(CHEMBL376703 | H-D-Phe-c[Cys-Ala-D-Trp-Lys-Thr-Cys...)
Affinity DataIC50:  3.60nMAssay Description:Inhibition of [125I](Leu8,DTrp22,Tyr25)-SRIF28 binding to human sst2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50191268(CHEMBL219201 | H2N-CO-DPhe-c[Cys-Aph(CONH2)-DTrp-L...)
Affinity DataIC50:  6.20nMAssay Description:Inhibition of [125I](Leu8,DTrp22,Tyr25)-SRIF28 binding to human sst2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50191269(CHEMBL412029 | H2N-CO-Phe-c[Cys-Aph(CONH2) -DTrp-L...)
Affinity DataIC50:  7.5nMAssay Description:Inhibition of [125I](Leu8,DTrp22,Tyr25)-SRIF28 binding to human sst2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50191271((4R,7S,10S,13R,16S,19R)-13-((1H-indol-3-yl)methyl)...)
Affinity DataIC50:  38nMAssay Description:Inhibition of [125I](Leu8,DTrp22,Tyr25)-SRIF28 binding to human sst3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50191268(CHEMBL219201 | H2N-CO-DPhe-c[Cys-Aph(CONH2)-DTrp-L...)
Affinity DataIC50:  77nMAssay Description:Inhibition of [125I](Leu8,DTrp22,Tyr25)-SRIF28 binding to human sst5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50191269(CHEMBL412029 | H2N-CO-Phe-c[Cys-Aph(CONH2) -DTrp-L...)
Affinity DataIC50:  109nMAssay Description:Inhibition of [125I](Leu8,DTrp22,Tyr25)-SRIF28 binding to human sst5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50191267(CHEMBL376703 | H-D-Phe-c[Cys-Ala-D-Trp-Lys-Thr-Cys...)
Affinity DataIC50:  158nMAssay Description:Inhibition of [125I](Leu8,DTrp22,Tyr25)-SRIF28 binding to human sst5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50191268(CHEMBL219201 | H2N-CO-DPhe-c[Cys-Aph(CONH2)-DTrp-L...)
Affinity DataIC50:  210nMAssay Description:Inhibition of [125I](Leu8,DTrp22,Tyr25)-SRIF28 binding to human sst3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50191272(CHEMBL438247 | H-c[Cys-Phe-DTrp-Lys-Thr-Cys]-OH)
Affinity DataIC50:  378nMAssay Description:Inhibition of [125I](Leu8,DTrp22,Tyr25)-SRIF28 binding to human sst2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50191268(CHEMBL219201 | H2N-CO-DPhe-c[Cys-Aph(CONH2)-DTrp-L...)
Affinity DataIC50:  494nMAssay Description:Inhibition of [125I](Leu8,DTrp22,Tyr25)-SRIF28 binding to human sst4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50191270(CHEMBL436892 | H2N-CO-DPhe-c[Cys-Aph(CONHOCH3)-DTr...)
Affinity DataIC50:  539nMAssay Description:Inhibition of [125I](Leu8,DTrp22,Tyr25)-SRIF28 binding to human sst5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50191267(CHEMBL376703 | H-D-Phe-c[Cys-Ala-D-Trp-Lys-Thr-Cys...)
Affinity DataIC50:  543nMAssay Description:Inhibition of [125I](Leu8,DTrp22,Tyr25)-SRIF28 binding to human sst3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50191269(CHEMBL412029 | H2N-CO-Phe-c[Cys-Aph(CONH2) -DTrp-L...)
Affinity DataIC50:  872nMAssay Description:Inhibition of [125I](Leu8,DTrp22,Tyr25)-SRIF28 binding to human sst4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50191269(CHEMBL412029 | H2N-CO-Phe-c[Cys-Aph(CONH2) -DTrp-L...)
Affinity DataIC50:  942nMAssay Description:Inhibition of [125I](Leu8,DTrp22,Tyr25)-SRIF28 binding to human sst3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50191270(CHEMBL436892 | H2N-CO-DPhe-c[Cys-Aph(CONHOCH3)-DTr...)
Affinity DataIC50:  958nMAssay Description:Inhibition of [125I](Leu8,DTrp22,Tyr25)-SRIF28 binding to human sst3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50191272(CHEMBL438247 | H-c[Cys-Phe-DTrp-Lys-Thr-Cys]-OH)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of [125I](Leu8,DTrp22,Tyr25)-SRIF28 binding to human sst3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50191272(CHEMBL438247 | H-c[Cys-Phe-DTrp-Lys-Thr-Cys]-OH)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of [125I](Leu8,DTrp22,Tyr25)-SRIF28 binding to human sst5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50191269(CHEMBL412029 | H2N-CO-Phe-c[Cys-Aph(CONH2) -DTrp-L...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of [125I](Leu8,DTrp22,Tyr25)-SRIF28 binding to human sst1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50191270(CHEMBL436892 | H2N-CO-DPhe-c[Cys-Aph(CONHOCH3)-DTr...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of [125I](Leu8,DTrp22,Tyr25)-SRIF28 binding to human sst1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50191272(CHEMBL438247 | H-c[Cys-Phe-DTrp-Lys-Thr-Cys]-OH)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of [125I](Leu8,DTrp22,Tyr25)-SRIF28 binding to human sst1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50191267(CHEMBL376703 | H-D-Phe-c[Cys-Ala-D-Trp-Lys-Thr-Cys...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of [125I](Leu8,DTrp22,Tyr25)-SRIF28 binding to human sst1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50191271((4R,7S,10S,13R,16S,19R)-13-((1H-indol-3-yl)methyl)...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of [125I](Leu8,DTrp22,Tyr25)-SRIF28 binding to human sst1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50191267(CHEMBL376703 | H-D-Phe-c[Cys-Ala-D-Trp-Lys-Thr-Cys...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of [125I](Leu8,DTrp22,Tyr25)-SRIF28 binding to human sst4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50191268(CHEMBL219201 | H2N-CO-DPhe-c[Cys-Aph(CONH2)-DTrp-L...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of [125I](Leu8,DTrp22,Tyr25)-SRIF28 binding to human sst1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50191272(CHEMBL438247 | H-c[Cys-Phe-DTrp-Lys-Thr-Cys]-OH)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of [125I](Leu8,DTrp22,Tyr25)-SRIF28 binding to human sst4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50191270(CHEMBL436892 | H2N-CO-DPhe-c[Cys-Aph(CONHOCH3)-DTr...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of [125I](Leu8,DTrp22,Tyr25)-SRIF28 binding to human sst4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50191271((4R,7S,10S,13R,16S,19R)-13-((1H-indol-3-yl)methyl)...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of [125I](Leu8,DTrp22,Tyr25)-SRIF28 binding to human sst4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed