Compile Data Set for Download or QSAR
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Found 372 Enz. Inhib. hit(s) with all data for entry = 50018237
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193321((Z)-1-(3,5-difluorophenyl)-3-(4-pyridin-2-ylpipera...)
Affinity DataKi:  6.30nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193331((E)-1-(3,4-dichlorophenyl)-3-(4-pyridin-2-ylpipera...)
Affinity DataKi:  6.40nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193296((Z)-1-(3-fluorophenyl)-3-(4-pyridin-2-ylpiperazin-...)
Affinity DataKi:  6.40nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193330((E)-3-(4-pyridin-2-ylpiperazin-1-yl)-1-(m-tolyl)pr...)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193290((E)-3-(4-pyridin-2-ylpiperazin-1-yl)-1-(o-tolyl)pr...)
Affinity DataKi:  11.4nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193361((Z)-1-(4-chloro-3-methylphenyl)-3-(4-pyridin-2-ylp...)
Affinity DataKi:  11.6nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193307((E)-1-(3-chlorophenyl)-3-(4-pyridin-2-ylpiperazin-...)
Affinity DataKi:  13.5nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193350((E)-1-(3-fluorophenyl)-3-(4-pyridin-2-ylpiperazin-...)
Affinity DataKi:  13.9nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193378((E)-1-(4-fluorophenyl)-3-(4-pyridin-2-ylpiperazin-...)
Affinity DataKi:  14.2nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193311((Z)-1-(4-chlorophenyl)-3-(3',4',5',6'-tetrahydro-2...)
Affinity DataKi:  19.4nMAssay Description:Displacement of [3H]PIPAT from human recombinant D2L receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193357((Z)-4-[1-methoxyimino-3-(4-pyridin-2-ylpiperazin-1...)
Affinity DataKi:  20.1nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193306((E)-1-phenyl-3-(4-pyridin-2-ylpiperazin-1-yl)propa...)
Affinity DataKi:  22.8nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193315((E)-1-(4-chlorophenyl)-3-(3',4',5',6'-tetrahydro-2...)
Affinity DataKi:  25.3nMAssay Description:Displacement of [3H]PIPAT from human recombinant D2L receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193312((E)-1-phenyl-3-(4-pyridin-2-ylpiperazin-1-yl)propa...)
Affinity DataKi:  25.4nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193289((E)-1-(3,4-dimethylphenyl)-3-(4-pyridin-2-ylpipera...)
Affinity DataKi:  27.5nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193317((Z)-3-(4-pyridin-2-ylpiperazin-1-yl)-1-(m-tolyl)pr...)
Affinity DataKi:  32.1nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193323((E)-1-phenyl-3-(4-pyridin-2-ylpiperazin-1-yl)propa...)
Affinity DataKi:  38nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193303((E)-1-(4-chlorophenyl)-3-(4-pyridin-2-ylpiperazin-...)
Affinity DataKi:  38.2nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193296((Z)-1-(3-fluorophenyl)-3-(4-pyridin-2-ylpiperazin-...)
Affinity DataKi:  46.6nMAssay Description:Displacement of [3H]PIPAT from human recombinant D2L receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193334((Z)-1-(4-fluorophenyl)-3-(4-pyridin-2-ylpiperazin-...)
Affinity DataKi:  53.3nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193361((Z)-1-(4-chloro-3-methylphenyl)-3-(4-pyridin-2-ylp...)
Affinity DataKi:  60.9nMAssay Description:Displacement of [3H]PIPAT from human recombinant D2L receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193303((E)-1-(4-chlorophenyl)-3-(4-pyridin-2-ylpiperazin-...)
Affinity DataKi:  63.8nMAssay Description:Displacement of [3H]PIPAT from human recombinant D2L receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193331((E)-1-(3,4-dichlorophenyl)-3-(4-pyridin-2-ylpipera...)
Affinity DataKi:  64.5nMAssay Description:Displacement of [3H]PIPAT from human recombinant D2L receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193375((E)-1-(4-chlorophenyl)-3-(2-methyl-4-pyridin-2-ylp...)
Affinity DataKi:  67.1nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193317((Z)-3-(4-pyridin-2-ylpiperazin-1-yl)-1-(m-tolyl)pr...)
Affinity DataKi:  68nMAssay Description:Displacement of [3H]PIPAT from human recombinant D2L receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193330((E)-3-(4-pyridin-2-ylpiperazin-1-yl)-1-(m-tolyl)pr...)
Affinity DataKi:  68.4nMAssay Description:Displacement of [3H]PIPAT from human recombinant D2L receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193372((E)-1-(3-chloro-4-fluorophenyl)-3-(4-pyridin-2-ylp...)
Affinity DataKi:  71.2nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193375((E)-1-(4-chlorophenyl)-3-(2-methyl-4-pyridin-2-ylp...)
Affinity DataKi:  76.5nMAssay Description:Displacement of [3H]PIPAT from human recombinant D2L receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193316(CHEMBL376955 | [1-phenyl-3-(4-pyridin-2-ylpiperazi...)
Affinity DataKi:  88nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193311((Z)-1-(4-chlorophenyl)-3-(3',4',5',6'-tetrahydro-2...)
Affinity DataKi:  90nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193307((E)-1-(3-chlorophenyl)-3-(4-pyridin-2-ylpiperazin-...)
Affinity DataKi:  98.7nMAssay Description:Displacement of [3H]PIPAT from human recombinant D2L receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193350((E)-1-(3-fluorophenyl)-3-(4-pyridin-2-ylpiperazin-...)
Affinity DataKi:  101nMAssay Description:Displacement of [3H]PIPAT from human recombinant D2L receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193360((E)-1-(3,5-difluorophenyl)-3-(4-pyridin-2-ylpipera...)
Affinity DataKi:  110nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193290((E)-3-(4-pyridin-2-ylpiperazin-1-yl)-1-(o-tolyl)pr...)
Affinity DataKi:  112nMAssay Description:Displacement of [3H]PIPAT from human recombinant D2L receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193336((E)-1-(4-chlorophenyl)-2-hydroxy-3-(4-pyridin-2-yl...)
Affinity DataKi:  113nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193320(1-(4-chlorophenyl)-2-(methoxyaminomethyl)-3-(4-pyr...)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193357((Z)-4-[1-methoxyimino-3-(4-pyridin-2-ylpiperazin-1...)
Affinity DataKi:  125nMAssay Description:Displacement of [3H]PIPAT from human recombinant D2L receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193323((E)-1-phenyl-3-(4-pyridin-2-ylpiperazin-1-yl)propa...)
Affinity DataKi:  128nMAssay Description:Displacement of [3H]PIPAT from human recombinant D2L receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193322(1-pyridin-3-yl-3-(4-pyridin-2-ylpiperazin-1-yl)pro...)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193360((E)-1-(3,5-difluorophenyl)-3-(4-pyridin-2-ylpipera...)
Affinity DataKi:  132nMAssay Description:Displacement of [3H]PIPAT from human recombinant D2L receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193315((E)-1-(4-chlorophenyl)-3-(3',4',5',6'-tetrahydro-2...)
Affinity DataKi:  134nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193289((E)-1-(3,4-dimethylphenyl)-3-(4-pyridin-2-ylpipera...)
Affinity DataKi:  137nMAssay Description:Displacement of [3H]PIPAT from human recombinant D2L receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193316(CHEMBL376955 | [1-phenyl-3-(4-pyridin-2-ylpiperazi...)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]PIPAT from human recombinant D2L receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193335(1-(4-chlorophenyl)-2-methyl-3-(4-pyridin-2-ylpiper...)
Affinity DataKi:  146nMAssay Description:Displacement of [3H]PIPAT from human recombinant D2L receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193313((Z)-1-(4-chlorophenyl)-2-hydroxy-3-(4-pyridin-2-yl...)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193320(1-(4-chlorophenyl)-2-(methoxyaminomethyl)-3-(4-pyr...)
Affinity DataKi:  164nMAssay Description:Displacement of [3H]PIPAT from human recombinant D2L receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193364((E)-1-phenyl-3-(4-thiazol-2-ylpiperazin-1-yl)propa...)
Affinity DataKi:  168nMAssay Description:Displacement of [3H]A-369508 from human recombinant D4.4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193378((E)-1-(4-fluorophenyl)-3-(4-pyridin-2-ylpiperazin-...)
Affinity DataKi:  168nMAssay Description:Displacement of [3H]PIPAT from human recombinant D2L receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193372((E)-1-(3-chloro-4-fluorophenyl)-3-(4-pyridin-2-ylp...)
Affinity DataKi:  171nMAssay Description:Displacement of [3H]PIPAT from human recombinant D2L receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50193306((E)-1-phenyl-3-(4-pyridin-2-ylpiperazin-1-yl)propa...)
Affinity DataKi:  172nMAssay Description:Displacement of [3H]PIPAT from human recombinant D2L receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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