Compile Data Set for Download or QSAR
maximum 50k data
Found 74 Enz. Inhib. hit(s) with all data for entry = 50018357
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194745(CHEMBL385900 | diphenyl 1-[(N-2-thiophenesulfonyl-...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194741(CHEMBL385158 | diphenyl 1-[(N-benzenesulfonyl-D-se...)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194743(CHEMBL214814 | diphenyl 1-[(N-alpha-toluenesulfony...)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50145689(CHEMBL80844 | [1-[(S)-2-((R)-2-Benzyloxycarbonylam...)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194737(CHEMBL384263 | diphenyl 1-[(N-o-methylbenzoyl-D-se...)
Affinity DataIC50:  4.40nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194746(CHEMBL405546 | diphenyl 1-[(N-o-methylbenzoyl-D-se...)
Affinity DataIC50:  5nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194742(CHEMBL263977 | diphenyl 1-[(N-benzyl-D-seryl)-L-al...)
Affinity DataIC50:  5nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194744(CHEMBL385897 | diphenyl 1-[(N-naphthalenesulfonyl-...)
Affinity DataIC50:  5.80nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194734(CHEMBL386275 | diphenyl 1-[(N-p-methoxybenzenesulf...)
Affinity DataIC50:  5.80nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194736(CHEMBL189823 | diphenyl 1-[(N-o,o-dimethylbenzoyl-...)
Affinity DataIC50:  6nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194735(CHEMBL215961 | diphenyl 1-[(N-p-cyanobenzenesulfon...)
Affinity DataIC50:  6.20nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194738(CHEMBL386249 | diphenyl 1-[(N-p-bromobenzenesulfon...)
Affinity DataIC50:  6.60nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194732(CHEMBL214539 | di-(4-acetamidophenyl) 1-[(N-benzyl...)
Affinity DataIC50:  6.70nMAssay Description:Inhibition of [3H]-FPP incorporation into biotin-linked K-ras decapeptide (CVIM) by bovine farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194739(CHEMBL213216 | diphenyl 1-[(N-2-thienyl-D-seryl)-L...)
Affinity DataIC50:  6.90nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194740(CHEMBL404226 | diphenyl 1-[(N-p-methylbenzoyl-D-se...)
Affinity DataIC50:  7nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194733(CHEMBL411215 | diphenyl 1-[(N-1-adamantanyl-D-sery...)
Affinity DataIC50:  8nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194743(CHEMBL214814 | diphenyl 1-[(N-alpha-toluenesulfony...)
Affinity DataIC50:  37nMAssay Description:Inhibition of human plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50145688(CHEMBL311067 | benzyl (R)-1-((S)-1-(1-(diphenoxyph...)
Affinity DataIC50:  61nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194743(CHEMBL214814 | diphenyl 1-[(N-alpha-toluenesulfony...)
Affinity DataIC50:  280nMAssay Description:Inhibition of recombinant tPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194732(CHEMBL214539 | di-(4-acetamidophenyl) 1-[(N-benzyl...)
Affinity DataIC50:  410nMAssay Description:Inhibition of mouse uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50145688(CHEMBL311067 | benzyl (R)-1-((S)-1-(1-(diphenoxyph...)
Affinity DataIC50:  500nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194743(CHEMBL214814 | diphenyl 1-[(N-alpha-toluenesulfony...)
Affinity DataIC50:  770nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194732(CHEMBL214539 | di-(4-acetamidophenyl) 1-[(N-benzyl...)
Affinity DataIC50:  900nMAssay Description:Inhibition of human plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194735(CHEMBL215961 | diphenyl 1-[(N-p-cyanobenzenesulfon...)
Affinity DataIC50:  900nMAssay Description:Inhibition of human plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194738(CHEMBL386249 | diphenyl 1-[(N-p-bromobenzenesulfon...)
Affinity DataIC50:  900nMAssay Description:Inhibition of human plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194744(CHEMBL385897 | diphenyl 1-[(N-naphthalenesulfonyl-...)
Affinity DataIC50:  990nMAssay Description:Inhibition of human plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194732(CHEMBL214539 | di-(4-acetamidophenyl) 1-[(N-benzyl...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194745(CHEMBL385900 | diphenyl 1-[(N-2-thiophenesulfonyl-...)
Affinity DataIC50:  1.54E+3nMAssay Description:Inhibition of human plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194734(CHEMBL386275 | diphenyl 1-[(N-p-methoxybenzenesulf...)
Affinity DataIC50:  1.67E+3nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194734(CHEMBL386275 | diphenyl 1-[(N-p-methoxybenzenesulf...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of human plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194741(CHEMBL385158 | diphenyl 1-[(N-benzenesulfonyl-D-se...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of human plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50145689(CHEMBL80844 | [1-[(S)-2-((R)-2-Benzyloxycarbonylam...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of human plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194738(CHEMBL386249 | diphenyl 1-[(N-p-bromobenzenesulfon...)
Affinity DataIC50:  2.98E+3nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194741(CHEMBL385158 | diphenyl 1-[(N-benzenesulfonyl-D-se...)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of recombinant tPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194745(CHEMBL385900 | diphenyl 1-[(N-2-thiophenesulfonyl-...)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of recombinant tPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194736(CHEMBL189823 | diphenyl 1-[(N-o,o-dimethylbenzoyl-...)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of recombinant tPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194738(CHEMBL386249 | diphenyl 1-[(N-p-bromobenzenesulfon...)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of recombinant tPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194736(CHEMBL189823 | diphenyl 1-[(N-o,o-dimethylbenzoyl-...)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of human plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194734(CHEMBL386275 | diphenyl 1-[(N-p-methoxybenzenesulf...)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of recombinant tPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194745(CHEMBL385900 | diphenyl 1-[(N-2-thiophenesulfonyl-...)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194744(CHEMBL385897 | diphenyl 1-[(N-naphthalenesulfonyl-...)
Affinity DataIC50:  4.40E+3nMAssay Description:Inhibition of recombinant tPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50145689(CHEMBL80844 | [1-[(S)-2-((R)-2-Benzyloxycarbonylam...)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of recombinant tPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194741(CHEMBL385158 | diphenyl 1-[(N-benzenesulfonyl-D-se...)
Affinity DataIC50:  4.90E+3nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194740(CHEMBL404226 | diphenyl 1-[(N-p-methylbenzoyl-D-se...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of human plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194733(CHEMBL411215 | diphenyl 1-[(N-1-adamantanyl-D-sery...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of human plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194746(CHEMBL405546 | diphenyl 1-[(N-o-methylbenzoyl-D-se...)
Affinity DataIC50:  5.50E+3nMAssay Description:Inhibition of recombinant tPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194744(CHEMBL385897 | diphenyl 1-[(N-naphthalenesulfonyl-...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194733(CHEMBL411215 | diphenyl 1-[(N-1-adamantanyl-D-sery...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194736(CHEMBL189823 | diphenyl 1-[(N-o,o-dimethylbenzoyl-...)
Affinity DataIC50:  6.30E+3nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50194732(CHEMBL214539 | di-(4-acetamidophenyl) 1-[(N-benzyl...)
Affinity DataIC50:  6.40E+3nMAssay Description:Inhibition of recombinant tPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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