Compile Data Set for Download or QSAR
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Found 12 Enz. Inhib. hit(s) with all data for entry = 50018386
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Ildong Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50195190(6-chloro-5-(4-ethoxyphenylamino)-1H-indazole-4,7-d...)
Affinity DataIC50:  4.90E+3nMAssay Description:Inhibition of Akt1 activity assessed as decrease in GSK3 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Ildong Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50195189(6-chloro-5-(3-fluorophenylamino)-1H-indazole-4,7-d...)
Affinity DataIC50:  1.18E+4nMAssay Description:Inhibition of Akt1 activity assessed as decrease in GSK3 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Ildong Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50195193(6-chloro-5-(3,4-dichlorophenylthio)-1H-indazole-4,...)
Affinity DataIC50:  1.23E+4nMAssay Description:Inhibition of Akt1 activity assessed as decrease in GSK3 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Ildong Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50195186(6-chloro-5-(4-(trifluoromethyl)phenylamino)-1H-ind...)
Affinity DataIC50:  1.24E+4nMAssay Description:Inhibition of Akt1 activity assessed as decrease in GSK3 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Ildong Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50195195(5-(3-bromophenylamino)-6-chloro-1H-indazole-4,7-di...)
Affinity DataIC50:  1.39E+4nMAssay Description:Inhibition of Akt1 activity assessed as decrease in GSK3 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Ildong Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50195187(6-chloro-5-(2-fluorophenylamino)-1H-indazole-4,7-d...)
Affinity DataIC50:  1.58E+4nMAssay Description:Inhibition of Akt1 activity assessed as decrease in GSK3 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Ildong Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50195192(6-chloro-5-(2,4-difluorophenylamino)-1H-indazole-4...)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of Akt1 activity assessed as decrease in GSK3 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Ildong Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50195188(2-thioxo-(1,3)ditholo[4,5-beta][1,4-dithine-5,6-di...)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of Akt1 activity assessed as decrease in GSK3 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Ildong Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50195185(6-chloro-5-(3,5-difluorophenylamino)-1H-indazole-4...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Akt1 activity assessed as decrease in GSK3 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Ildong Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50195191(6-chloro-5-(4-fluorophenylamino)-1H-indazole-4,7-d...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Akt1 activity assessed as decrease in GSK3 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Ildong Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50195184(6-chloro-5-(3,5-dimethylphenylthio)-1H-indazole-4,...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Akt1 activity assessed as decrease in GSK3 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Ildong Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50195194(1H-indazole-4,7-diamine | CHEMBL376871)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Akt1 activity assessed as decrease in GSK3 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed