Compile Data Set for Download or QSAR
maximum 50k data
Found 10 Enz. Inhib. hit(s) with all data for entry = 50037831
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50204623(CHEMBL223747 | [2-(hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  5.20nMAssay Description:Displacement of [3H]PDBu from PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50204626((2-(hydroxymethyl)-5-oxo-4-(propan-2-ylidene)-tetr...)
Affinity DataKi:  5.90nMAssay Description:Displacement of [3H]PDBu from PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50204628(CHEMBL223570 | [2-(hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]PDBu from PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50204629(CHEMBL221289 | methyl 2-{4-[2-(4-{2-[4-({[2-(hydro...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]PDBu from PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50204630(CHEMBL413585 | [2-(hydroxymethyl)-4-(methylethylid...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]PDBu from PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50370871(CHEMBL1162941)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]PDBu from PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50204625(CHEMBL220962 | methyl 16-{4-[2-(4-{2-[4-({[2-(Hydr...)
Affinity DataKi:  53nMAssay Description:Displacement of [3H]PDBu from PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50204624(CHEMBL220099 | tert-butyl 2-({[(tert-Butyl)oxycarb...)
Affinity DataKi:  111nMAssay Description:Displacement of [3H]PDBu from PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50204622(CHEMBL221290 | methyl 2-[4-(2-{4-[2-(4-{2-[4-({[2-...)
Affinity DataKi:  127nMAssay Description:Displacement of [3H]PDBu from PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50204627(2-(N-(carboxymethyl){2-[2-(2-{4-[2-(4-{2-[4-({[2-(...)
Affinity DataKi:  1.39E+3nMAssay Description:Displacement of [3H]PDBu from PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed