Affinity DataKi: 0.570nMAssay Description:Binding affinity to human DP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.840nMAssay Description:Binding affinity to human TP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Binding affinity to human DP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Binding affinity to human DP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Binding affinity to human DP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Binding affinity to human DP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Binding affinity to human TP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8.90nMAssay Description:Binding affinity to human DP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 9.60nMAssay Description:Binding affinity to human DP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding affinity to human TP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Merck Frosst Canada
Curated by ChEMBL
Merck Frosst Canada
Curated by ChEMBL
Affinity DataKi: 136nMAssay Description:Binding affinity to human EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Merck Frosst Canada
Curated by ChEMBL
Merck Frosst Canada
Curated by ChEMBL
Affinity DataKi: 230nMAssay Description:Binding affinity to human EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Merck Frosst Canada
Curated by ChEMBL
Merck Frosst Canada
Curated by ChEMBL
Affinity DataKi: 310nMAssay Description:Binding affinity to human EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Merck Frosst Canada
Curated by ChEMBL
Merck Frosst Canada
Curated by ChEMBL
Affinity DataKi: 390nMAssay Description:Binding affinity to human EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 400nMAssay Description:Binding affinity to human IP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Merck Frosst Canada
Curated by ChEMBL
Merck Frosst Canada
Curated by ChEMBL
Affinity DataKi: 410nMAssay Description:Binding affinity to human EP2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP3 subtype(Homo sapiens (Human))
Merck Frosst Canada
Curated by ChEMBL
Merck Frosst Canada
Curated by ChEMBL
Affinity DataKi: 470nMAssay Description:Binding affinity to human EP3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 745nMAssay Description:Activity at CRTH2 receptorMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP3 subtype(Homo sapiens (Human))
Merck Frosst Canada
Curated by ChEMBL
Merck Frosst Canada
Curated by ChEMBL
Affinity DataKi: 892nMAssay Description:Binding affinity to human EP3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.05E+3nMAssay Description:Binding affinity to human TP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP1 subtype(Homo sapiens (Human))
Merck Frosst Canada
Curated by ChEMBL
Merck Frosst Canada
Curated by ChEMBL
Affinity DataKi: 1.16E+3nMAssay Description:Binding affinity to human EP1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP3 subtype(Homo sapiens (Human))
Merck Frosst Canada
Curated by ChEMBL
Merck Frosst Canada
Curated by ChEMBL
Affinity DataKi: 1.20E+3nMAssay Description:Binding affinity to human EP3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.20E+3nMAssay Description:Binding affinity to human TP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Merck Frosst Canada
Curated by ChEMBL
Merck Frosst Canada
Curated by ChEMBL
Affinity DataKi: 4.40E+3nMAssay Description:Binding affinity to human EP4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP1 subtype(Homo sapiens (Human))
Merck Frosst Canada
Curated by ChEMBL
Merck Frosst Canada
Curated by ChEMBL
Affinity DataKi: 4.40E+3nMAssay Description:Binding affinity to human EP1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.63E+3nMAssay Description:Binding affinity to human IP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.10E+3nMAssay Description:Binding affinity to human TP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP1 subtype(Homo sapiens (Human))
Merck Frosst Canada
Curated by ChEMBL
Merck Frosst Canada
Curated by ChEMBL
Affinity DataKi: >9.00E+3nMAssay Description:Binding affinity to human EP1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 9.99E+3nMAssay Description:Binding affinity to human FP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+4nMAssay Description:Binding affinity to human FP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+4nMAssay Description:Binding affinity to human IP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Merck Frosst Canada
Curated by ChEMBL
Merck Frosst Canada
Curated by ChEMBL
Affinity DataKi: >1.52E+4nMAssay Description:Binding affinity to human EP4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP3 subtype(Homo sapiens (Human))
Merck Frosst Canada
Curated by ChEMBL
Merck Frosst Canada
Curated by ChEMBL
Affinity DataKi: >2.00E+4nMAssay Description:Binding affinity to human EP3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+4nMAssay Description:Binding affinity to human FP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+4nMAssay Description:Binding affinity to human IP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP1 subtype(Homo sapiens (Human))
Merck Frosst Canada
Curated by ChEMBL
Merck Frosst Canada
Curated by ChEMBL
Affinity DataKi: >2.00E+4nMAssay Description:Binding affinity to human EP1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+4nMAssay Description:Binding affinity to human FP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+4nMAssay Description:Binding affinity to human IP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Merck Frosst Canada
Curated by ChEMBL
Merck Frosst Canada
Curated by ChEMBL
Affinity DataKi: >2.00E+4nMAssay Description:Binding affinity to human EP4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Merck Frosst Canada
Curated by ChEMBL
Merck Frosst Canada
Curated by ChEMBL
Affinity DataKi: >2.00E+4nMAssay Description:Binding affinity to human EP4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP3 subtype(Homo sapiens (Human))
Merck Frosst Canada
Curated by ChEMBL
Merck Frosst Canada
Curated by ChEMBL
Affinity DataKi: >2.00E+4nMAssay Description:Binding affinity to human EP3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Merck Frosst Canada
Curated by ChEMBL
Merck Frosst Canada
Curated by ChEMBL
Affinity DataKi: >2.00E+4nMAssay Description:Binding affinity to human EP4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+4nMAssay Description:Binding affinity to human FP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP1 subtype(Homo sapiens (Human))
Merck Frosst Canada
Curated by ChEMBL
Merck Frosst Canada
Curated by ChEMBL
Affinity DataKi: >2.00E+4nMAssay Description:Binding affinity to human EP1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0900nMAssay Description:Activity at human DP receptor in washed platelets assessed as inhibition of PGD2-induced cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.260nMAssay Description:Activity at human DP receptor in washed platelets assessed as inhibition of PGD2-induced cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.290nMAssay Description:Activity at human DP receptor in washed platelets assessed as inhibition of PGD2-induced cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Activity at sheep DP receptor by PRP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Activity at human DP receptor in washed platelets assessed as inhibition of PGD2-induced cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Activity at human DP receptor in washed platelets assessed as inhibition of PGD2-induced cAMP accumulationMore data for this Ligand-Target Pair