Affinity DataKi: 0.75nMAssay Description:Displacement of [3H]U69,593 from rat cloned KORMore data for this Ligand-Target Pair
Affinity DataKi: 54.5nMAssay Description:Displacement of [3H]U69,593 from rat cloned KORMore data for this Ligand-Target Pair
Affinity DataKi: 151nMAssay Description:Displacement of [3H]U69,593 from rat cloned KORMore data for this Ligand-Target Pair
Affinity DataKi: 546nMAssay Description:Displacement of [3H]U69,593 from rat cloned KORMore data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+3nMAssay Description:Activity at human kappa opioid receptor expressed in HEK293 cells as intracellular calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 2.82nMAssay Description:Activity at human kappa opioid receptor expressed in HEK293 cells as intracellular calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 287nMAssay Description:Activity at human kappa opioid receptor expressed in HEK293 cells as intracellular calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 123nMAssay Description:Activity at human kappa opioid receptor expressed in HEK293 cells as intracellular calcium mobilizationMore data for this Ligand-Target Pair