Compile Data Set for Download or QSAR
maximum 50k data
Found 53 Enz. Inhib. hit(s) with all data for entry = 50019682
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206687((S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimi...)
Affinity DataKi:  1nMAssay Description:Binding affinity to human MCHR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206675((S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimi...)
Affinity DataKi:  2nMAssay Description:Binding affinity to human MCHR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206679((S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimi...)
Affinity DataKi:  3nMAssay Description:Binding affinity to human MCHR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206666((S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimi...)
Affinity DataKi:  3nMAssay Description:Binding affinity to human MCHR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206681((S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimi...)
Affinity DataKi:  4nMAssay Description:Binding affinity to human MCHR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206677((S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimi...)
Affinity DataKi:  4nMAssay Description:Binding affinity to human MCHR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206690((S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimi...)
Affinity DataKi:  4nMAssay Description:Binding affinity to human MCHR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206689((S)-3-(6-(4-ethylphenyl)-4-oxothieno[3,2-d]pyrimid...)
Affinity DataKi:  5nMAssay Description:Binding affinity to human MCHR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206673((S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimi...)
Affinity DataKi:  5nMAssay Description:Binding affinity to human MCHR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206669((S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimi...)
Affinity DataKi:  6nMAssay Description:Binding affinity to human MCHR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206663((S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimi...)
Affinity DataKi:  7nMAssay Description:Binding affinity to human MCHR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206662((S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimi...)
Affinity DataKi:  7nMAssay Description:Binding affinity to human MCHR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206665((S)-3-(6-(4-ethylphenyl)-4-oxothieno[3,2-d]pyrimid...)
Affinity DataKi:  8nMAssay Description:Binding affinity to human MCHR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206670((S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimi...)
Affinity DataKi:  10nMAssay Description:Binding affinity to human MCHR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206693((S)-N-methyl-3-(4-oxo-6-p-tolylthieno[3,2-d]pyrimi...)
Affinity DataKi:  14nMAssay Description:Binding affinity to human MCHR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206686((S)-3-(6-(2-chloro-4-ethoxyphenyl)-4-oxothieno[3,2...)
Affinity DataKi:  14nMAssay Description:Binding affinity to human MCHR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206678((S)-N-methyl-N-((S)-1-methylpyrrolidin-3-yl)-3-(4-...)
Affinity DataKi:  15nMAssay Description:Binding affinity to human MCHR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206692((S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimi...)
Affinity DataKi:  17nMAssay Description:Binding affinity to human MCHR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206684((S)-N-methyl-N-((S)-1-methylpyrrolidin-3-yl)-3-(4-...)
Affinity DataKi:  17nMAssay Description:Binding affinity to human MCHR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206676((S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimi...)
Affinity DataKi:  17nMAssay Description:Binding affinity to human MCHR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206685((S)-N-methyl-3-(4-oxo-6-(4-(trifluoromethoxy)pheny...)
Affinity DataKi:  18nMAssay Description:Binding affinity to human MCHR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206688((S)-N-methyl-3-(4-oxo-6-(4-(trifluoromethyl)phenyl...)
Affinity DataKi:  19nMAssay Description:Binding affinity to human MCHR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206680((S)-3-(6-(4-methoxyphenyl)-4-oxothieno[3,2-d]pyrim...)
Affinity DataKi:  21nMAssay Description:Binding affinity to human MCHR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206667((S)-3-(6-(2-chloro-4-ethoxyphenyl)-4-oxothieno[3,2...)
Affinity DataKi:  26nMAssay Description:Binding affinity to human MCHR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206672((S)-3-(6-(4-methoxy-2-methylphenyl)-4-oxothieno[3,...)
Affinity DataKi:  28nMAssay Description:Binding affinity to human MCHR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206671((S)-N-methyl-N-((S)-1-methylpyrrolidin-3-yl)-3-(4-...)
Affinity DataKi:  39nMAssay Description:Binding affinity to human MCHR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206674((S)-3-(6-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-4-o...)
Affinity DataKi:  45nMAssay Description:Binding affinity to human MCHR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206694((S)-3-(6-(4-methoxy-2-methylphenyl)-4-oxothieno[3,...)
Affinity DataKi:  46nMAssay Description:Binding affinity to human MCHR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206661((S)-3-(6-(2,4-dimethylphenyl)-4-oxothieno[3,2-d]py...)
Affinity DataKi:  49nMAssay Description:Binding affinity to human MCHR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206664((S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimi...)
Affinity DataKi:  50nMAssay Description:Binding affinity to human MCHR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206668((R)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimi...)
Affinity DataKi:  69nMAssay Description:Binding affinity to human MCHR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206682((S)-3-(6-(2,4-dimethylphenyl)-4-oxothieno[3,2-d]py...)
Affinity DataKi:  70nMAssay Description:Binding affinity to human MCHR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206691((S)-3-[6-(4-chloro-phenyl)-4-oxo-4H-thieno[3,2-d]p...)
Affinity DataKi:  80nMAssay Description:Binding affinity to human MCHR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206695((S)-3-(6-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-4-o...)
Affinity DataKi:  143nMAssay Description:Binding affinity to human MCHR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206683((R)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimi...)
Affinity DataKi:  154nMAssay Description:Binding affinity to human MCHR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206687((S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimi...)
Affinity DataIC50:  9nMAssay Description:Antagonist activity at human MCHR1 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206675((S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimi...)
Affinity DataIC50:  10nMAssay Description:Antagonist activity at human MCHR1 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206690((S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimi...)
Affinity DataIC50:  10nMAssay Description:Antagonist activity at human MCHR1 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206679((S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimi...)
Affinity DataIC50:  10nMAssay Description:Antagonist activity at human MCHR1 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206663((S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimi...)
Affinity DataIC50:  11nMAssay Description:Antagonist activity at human MCHR1 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206662((S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimi...)
Affinity DataIC50:  11nMAssay Description:Antagonist activity at human MCHR1 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206677((S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimi...)
Affinity DataIC50:  13nMAssay Description:Antagonist activity at human MCHR1 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206681((S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimi...)
Affinity DataIC50:  15nMAssay Description:Antagonist activity at human MCHR1 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206670((S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimi...)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at human MCHR1 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206673((S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimi...)
Affinity DataIC50:  23nMAssay Description:Antagonist activity at human MCHR1 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206666((S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimi...)
Affinity DataIC50:  23nMAssay Description:Antagonist activity at human MCHR1 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206692((S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimi...)
Affinity DataIC50:  29nMAssay Description:Antagonist activity at human MCHR1 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206669((S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimi...)
Affinity DataIC50:  31nMAssay Description:Antagonist activity at human MCHR1 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206676((S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimi...)
Affinity DataIC50:  44nMAssay Description:Antagonist activity at human MCHR1 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50206664((S)-3-(6-(4-chlorophenyl)-4-oxothieno[3,2-d]pyrimi...)
Affinity DataIC50:  53nMAssay Description:Antagonist activity at human MCHR1 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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