Compile Data Set for Download or QSAR
maximum 50k data
Found 100 Enz. Inhib. hit(s) with all data for entry = 50019960
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209158(2-(4-methyl-piperazin-1-yl)-N-{3-[5-(3-phenoxy-pro...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Flt1 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209158(2-(4-methyl-piperazin-1-yl)-N-{3-[5-(3-phenoxy-pro...)
Affinity DataIC50:  10nMAssay Description:Inhibition of KDR by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209148(CHEMBL246166 | N-{3-[5-(3-phenoxy-prop-1-ynyl)-thi...)
Affinity DataIC50:  20nMAssay Description:Inhibition of Flt1 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209158(2-(4-methyl-piperazin-1-yl)-N-{3-[5-(3-phenoxy-pro...)
Affinity DataIC50:  22nMAssay Description:Inhibition of Flt3 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209143(2-methoxy-N-(3-thiophen-3-yl-2,4-dihydro-indeno[1,...)
Affinity DataIC50:  30nMAssay Description:Inhibition of Flt1 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209148(CHEMBL246166 | N-{3-[5-(3-phenoxy-prop-1-ynyl)-thi...)
Affinity DataIC50:  36nMAssay Description:Inhibition of KDR by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209158(2-(4-methyl-piperazin-1-yl)-N-{3-[5-(3-phenoxy-pro...)
Affinity DataIC50:  45nMAssay Description:Inhibition of CSF1R by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209158(2-(4-methyl-piperazin-1-yl)-N-{3-[5-(3-phenoxy-pro...)
Affinity DataIC50:  49nMAssay Description:Inhibition of c-Kit by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209151(CHEMBL247388 | N-(3-thiophen-3-yl-2,4-dihydro-inde...)
Affinity DataIC50:  50nMAssay Description:Inhibition of KDR by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209146(CHEMBL247585 | N-(3-thiophen-3-yl-2,4-dihydro-inde...)
Affinity DataIC50:  50nMAssay Description:Inhibition of Flt1 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209150(2-methoxy-N-{3-[5-(3-phenoxy-prop-1-ynyl)-thiophen...)
Affinity DataIC50:  53nMAssay Description:Inhibition of KDR by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209154(5-methyl-isoxazole-3-carboxylic acid (3-thiophen-3...)
Affinity DataIC50:  60nMAssay Description:Inhibition of KDR by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209148(CHEMBL246166 | N-{3-[5-(3-phenoxy-prop-1-ynyl)-thi...)
Affinity DataIC50:  65nMAssay Description:Inhibition of Flt3 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209143(2-methoxy-N-(3-thiophen-3-yl-2,4-dihydro-indeno[1,...)
Affinity DataIC50:  70nMAssay Description:Inhibition of KDR by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209154(5-methyl-isoxazole-3-carboxylic acid (3-thiophen-3...)
Affinity DataIC50:  70nMAssay Description:Inhibition of Flt1 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209151(CHEMBL247388 | N-(3-thiophen-3-yl-2,4-dihydro-inde...)
Affinity DataIC50:  80nMAssay Description:Inhibition of Flt1 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209153(CHEMBL247389 | furan-2-carboxylic acid (3-thiophen...)
Affinity DataIC50:  90nMAssay Description:Inhibition of Flt1 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209146(CHEMBL247585 | N-(3-thiophen-3-yl-2,4-dihydro-inde...)
Affinity DataIC50:  100nMAssay Description:Inhibition of KDR by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209153(CHEMBL247389 | furan-2-carboxylic acid (3-thiophen...)
Affinity DataIC50:  110nMAssay Description:Inhibition of KDR by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209150(2-methoxy-N-{3-[5-(3-phenoxy-prop-1-ynyl)-thiophen...)
Affinity DataIC50:  113nMAssay Description:Inhibition of CSF1R by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209148(CHEMBL246166 | N-{3-[5-(3-phenoxy-prop-1-ynyl)-thi...)
Affinity DataIC50:  127nMAssay Description:Inhibition of c-Kit by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209144(2-(2-methoxy-ethoxy)-N-{3-[5-(3-phenoxy-prop-1-yny...)
Affinity DataIC50:  136nMAssay Description:Inhibition of Flt1 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209156(CHEMBL395427 | N-{3-[5-(3-phenoxy-prop-1-ynyl)-thi...)
Affinity DataIC50:  153nMAssay Description:Inhibition of Flt1 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209150(2-methoxy-N-{3-[5-(3-phenoxy-prop-1-ynyl)-thiophen...)
Affinity DataIC50:  153nMAssay Description:Inhibition of Flt3 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209150(2-methoxy-N-{3-[5-(3-phenoxy-prop-1-ynyl)-thiophen...)
Affinity DataIC50:  175nMAssay Description:Inhibition of c-Kit by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209146(CHEMBL247585 | N-(3-thiophen-3-yl-2,4-dihydro-inde...)
Affinity DataIC50:  180nMAssay Description:Inhibition of c-Kit by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209148(CHEMBL246166 | N-{3-[5-(3-phenoxy-prop-1-ynyl)-thi...)
Affinity DataIC50:  190nMAssay Description:Inhibition of CSF1R by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209159(CHEMBL246343 | [(3-thiophen-3-yl-2,4-dihydro-inden...)
Affinity DataIC50:  240nMAssay Description:Inhibition of Flt1 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209156(CHEMBL395427 | N-{3-[5-(3-phenoxy-prop-1-ynyl)-thi...)
Affinity DataIC50:  263nMAssay Description:Inhibition of KDR by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209144(2-(2-methoxy-ethoxy)-N-{3-[5-(3-phenoxy-prop-1-yny...)
Affinity DataIC50:  270nMAssay Description:Inhibition of KDR by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209160(2-[(3-thiophen-3-yl-2,4-dihydro-indeno[1,2-c]pyraz...)
Affinity DataIC50:  270nMAssay Description:Inhibition of Flt1 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209145(CHEMBL245362 | N-(3-thiophen-3-yl-2,4-dihydro-inde...)
Affinity DataIC50:  290nMAssay Description:Inhibition of Flt1 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209161(CHEMBL395694 | ethanesulfonic acid (3-thiophen-3-y...)
Affinity DataIC50:  290nMAssay Description:Inhibition of Flt1 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209161(CHEMBL395694 | ethanesulfonic acid (3-thiophen-3-y...)
Affinity DataIC50:  310nMAssay Description:Inhibition of KDR by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209147(3-[(3-thiophen-3-yl-2,4-dihydro-indeno[1,2-c]pyraz...)
Affinity DataIC50:  370nMAssay Description:Inhibition of Flt1 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209159(CHEMBL246343 | [(3-thiophen-3-yl-2,4-dihydro-inden...)
Affinity DataIC50:  410nMAssay Description:Inhibition of KDR by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209160(2-[(3-thiophen-3-yl-2,4-dihydro-indeno[1,2-c]pyraz...)
Affinity DataIC50:  440nMAssay Description:Inhibition of KDR by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209157((3-thiophen-3-yl-2,4-dihydro-indeno[1,2-c]pyrazol-...)
Affinity DataIC50:  450nMAssay Description:Inhibition of Flt1 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209145(CHEMBL245362 | N-(3-thiophen-3-yl-2,4-dihydro-inde...)
Affinity DataIC50:  560nMAssay Description:Inhibition of KDR by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209147(3-[(3-thiophen-3-yl-2,4-dihydro-indeno[1,2-c]pyraz...)
Affinity DataIC50:  580nMAssay Description:Inhibition of KDR by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209156(CHEMBL395427 | N-{3-[5-(3-phenoxy-prop-1-ynyl)-thi...)
Affinity DataIC50:  619nMAssay Description:Inhibition of c-Kit by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209144(2-(2-methoxy-ethoxy)-N-{3-[5-(3-phenoxy-prop-1-yny...)
Affinity DataIC50:  624nMAssay Description:Inhibition of Flt3 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209157((3-thiophen-3-yl-2,4-dihydro-indeno[1,2-c]pyrazol-...)
Affinity DataIC50:  650nMAssay Description:Inhibition of KDR by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209162(2-(4-methyl-piperazin-1-yl)-N-(3-thiophen-3-yl-2,4...)
Affinity DataIC50:  710nMAssay Description:Inhibition of Flt1 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209150(2-methoxy-N-{3-[5-(3-phenoxy-prop-1-ynyl)-thiophen...)
Affinity DataIC50:  710nMAssay Description:Inhibition of Flt1 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209154(5-methyl-isoxazole-3-carboxylic acid (3-thiophen-3...)
Affinity DataIC50:  900nMAssay Description:Inhibition of c-Kit by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209162(2-(4-methyl-piperazin-1-yl)-N-(3-thiophen-3-yl-2,4...)
Affinity DataIC50:  920nMAssay Description:Inhibition of KDR by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209153(CHEMBL247389 | furan-2-carboxylic acid (3-thiophen...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of c-Kit by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209156(CHEMBL395427 | N-{3-[5-(3-phenoxy-prop-1-ynyl)-thi...)
Affinity DataIC50:  1.11E+3nMAssay Description:Inhibition of Flt3 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209151(CHEMBL247388 | N-(3-thiophen-3-yl-2,4-dihydro-inde...)
Affinity DataIC50:  1.12E+3nMAssay Description:Inhibition of c-Kit by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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