Compile Data Set for Download or QSAR
maximum 50k data
Found 99 Enz. Inhib. hit(s) with all data for entry = 50020141
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM11162((1R)-3-oxo-3-[3-(trifluoroethyl)-5,6-dihydro[1,2,4...)
Affinity DataIC50:  18nMAssay Description:Inhibition of DPP4 activityMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM15561((3R)-3-amino-4-(5-chloro-2-fluorophenyl)-1-[3-(tri...)
Affinity DataIC50:  21nMAssay Description:Inhibition of DPP4 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210657((R)-3-amino-4-(2,4-dichlorophenyl)-1-(3-(trifluoro...)
Affinity DataIC50:  23nMAssay Description:Inhibition of DPP4 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM11160((3R)-3-amino-4-(2,5-difluorophenyl)-1-[3-(trifluor...)
Affinity DataIC50:  27nMAssay Description:Inhibition of DPP4 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210649((R)-3-amino-1-(3-(difluoromethyl)-5,6-dihydro-[1,2...)
Affinity DataIC50:  29nMAssay Description:Inhibition of DPP4 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210647((R)-3-amino-1-(3-cyclopropyl-5,6-dihydro-[1,2,4]tr...)
Affinity DataIC50:  30nMAssay Description:Inhibition of DPP4 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210668((3R)-3-amino-4-(2,5-difluorophenyl)-1-(3-(2,4-difl...)
Affinity DataIC50:  30nMAssay Description:Inhibition of DPP4 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210652((R)-3-amino-1-(3-ethyl-5,6-dihydro-[1,2,4]triazolo...)
Affinity DataIC50:  37nMAssay Description:Inhibition of DPP4 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210650((R)-3-amino-4-(3-chlorophenyl)-1-(3-(trifluorometh...)
Affinity DataIC50:  59nMAssay Description:Inhibition of DPP4 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210672((R)-3-amino-4-(2,5-difluorophenyl)-1-(3-(4-fluorop...)
Affinity DataIC50:  60nMAssay Description:Inhibition of DPP4 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210648((R)-3-amino-4-(2,5-difluorophenyl)-1-(3-(pyridin-4...)
Affinity DataIC50:  65nMAssay Description:Inhibition of DPP4 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210670((R)-3-amino-4-(2,5-difluorophenyl)-1-(3-(hydroxyme...)
Affinity DataIC50:  69nMAssay Description:Inhibition of DPP4 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210669((R)-3-amino-4-(4-chloro-2,5-difluorophenyl)-1-(3-(...)
Affinity DataIC50:  76nMAssay Description:Inhibition of DPP4 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210665((R)-3-amino-4-(2,4-difluorophenyl)-1-(3-(trifluoro...)
Affinity DataIC50:  82nMAssay Description:Inhibition of DPP4 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210643((R)-3-amino-4-(2-chloro-4,5-difluorophenyl)-1-(3-(...)
Affinity DataIC50:  84nMAssay Description:Inhibition of DPP4 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210658((R)-3-amino-1-(3-(trifluoromethyl)-5,6-dihydro-[1,...)
Affinity DataIC50:  87nMAssay Description:Inhibition of DPP4 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210663((R)-3-amino-4-(2-fluorophenyl)-1-(3-(trifluorometh...)
Affinity DataIC50:  98nMAssay Description:Inhibition of DPP4 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM11159((1R)-1-(3,4-difluorobenzyl)-3-oxo-3-[3-(trifluorom...)
Affinity DataIC50:  128nMAssay Description:Inhibition of DPP4 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210662((R)-3-amino-4-(3-fluorophenyl)-1-(3-(trifluorometh...)
Affinity DataIC50:  135nMAssay Description:Inhibition of DPP4 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210661((R)-3-amino-4-(2-chlorophenyl)-1-(3-(trifluorometh...)
Affinity DataIC50:  145nMAssay Description:Inhibition of DPP4 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210653((R)-3-amino-1-(3-(trifluoromethyl)-5,6-dihydro-[1,...)
Affinity DataIC50:  151nMAssay Description:Inhibition of DPP4 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210664((R)-3-amino-4-(2,5-dichlorophenyl)-1-(3-(trifluoro...)
Affinity DataIC50:  180nMAssay Description:Inhibition of DPP4 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210651((R)-ethyl 7-(3-amino-4-(2,5-difluorophenyl)butanoy...)
Affinity DataIC50:  190nMAssay Description:Inhibition of DPP4 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210666((R)-ethyl 7-(3-amino-4-(2,4,5-trifluorophenyl)buta...)
Affinity DataIC50:  219nMAssay Description:Inhibition of DPP4 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210671((R)-7-(3-amino-4-(2,4,5-trifluorophenyl)butanoyl)-...)
Affinity DataIC50:  234nMAssay Description:Inhibition of DPP4 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210660((R)-3-amino-4-(4-chlorophenyl)-1-(3-(trifluorometh...)
Affinity DataIC50:  264nMAssay Description:Inhibition of DPP4 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210645((R)-3-amino-4-(4-fluorophenyl)-1-(3-(trifluorometh...)
Affinity DataIC50:  272nMAssay Description:Inhibition of DPP4 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210659((R)-3-amino-1-(3-(trifluoromethyl)-5,6-dihydro-[1,...)
Affinity DataIC50:  366nMAssay Description:Inhibition of DPP4 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210644((R)-3-amino-1-(3-(trifluoromethyl)-5,6-dihydro-[1,...)
Affinity DataIC50:  486nMAssay Description:Inhibition of DPP4 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210667((R)-3-amino-1-(3-(trifluoromethyl)-5,6-dihydro-[1,...)
Affinity DataIC50:  511nMAssay Description:Inhibition of DPP4 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210655((R)-3-amino-1-(3-(trifluoromethyl)-5,6-dihydro-[1,...)
Affinity DataIC50:  805nMAssay Description:Inhibition of DPP4 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210672((R)-3-amino-4-(2,5-difluorophenyl)-1-(3-(4-fluorop...)
Affinity DataIC50:  979nMAssay Description:Inhibition of DPP8 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210668((3R)-3-amino-4-(2,5-difluorophenyl)-1-(3-(2,4-difl...)
Affinity DataIC50:  1.01E+3nMAssay Description:Inhibition of DPP8 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210654((R)-3-amino-4-(perfluorophenyl)-1-(3-(trifluoromet...)
Affinity DataIC50:  1.02E+3nMAssay Description:Inhibition of DPP4 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210656((R)-3-amino-4-(3,4-dichlorophenyl)-1-(3-(trifluoro...)
Affinity DataIC50:  1.58E+3nMAssay Description:Inhibition of DPP4 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210648((R)-3-amino-4-(2,5-difluorophenyl)-1-(3-(pyridin-4...)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of DPP8 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210658((R)-3-amino-1-(3-(trifluoromethyl)-5,6-dihydro-[1,...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of DPP8 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210653((R)-3-amino-1-(3-(trifluoromethyl)-5,6-dihydro-[1,...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of DPP8 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210655((R)-3-amino-1-(3-(trifluoromethyl)-5,6-dihydro-[1,...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of DPP8 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210666((R)-ethyl 7-(3-amino-4-(2,4,5-trifluorophenyl)buta...)
Affinity DataIC50: >2.20E+4nMAssay Description:Inhibition of DPP8 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210660((R)-3-amino-4-(4-chlorophenyl)-1-(3-(trifluorometh...)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of DPP8 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210657((R)-3-amino-4-(2,4-dichlorophenyl)-1-(3-(trifluoro...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of DPP8 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210651((R)-ethyl 7-(3-amino-4-(2,5-difluorophenyl)butanoy...)
Affinity DataIC50:  3.70E+4nMAssay Description:Inhibition of DPP8 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210652((R)-3-amino-1-(3-ethyl-5,6-dihydro-[1,2,4]triazolo...)
Affinity DataIC50:  3.90E+4nMAssay Description:Inhibition of DPP8 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM11159((1R)-1-(3,4-difluorobenzyl)-3-oxo-3-[3-(trifluorom...)
Affinity DataIC50:  4.60E+4nMAssay Description:Inhibition of DPP8 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM11162((1R)-3-oxo-3-[3-(trifluoroethyl)-5,6-dihydro[1,2,4...)
Affinity DataIC50:  4.80E+4nMAssay Description:Inhibition of DPP8 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210657((R)-3-amino-4-(2,4-dichlorophenyl)-1-(3-(trifluoro...)
Affinity DataIC50:  4.90E+4nMAssay Description:Inhibition of DPP9 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210669((R)-3-amino-4-(4-chloro-2,5-difluorophenyl)-1-(3-(...)
Affinity DataIC50:  4.90E+4nMAssay Description:Inhibition of DPP8 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210647((R)-3-amino-1-(3-cyclopropyl-5,6-dihydro-[1,2,4]tr...)
Affinity DataIC50:  5.40E+4nMAssay Description:Inhibition of DPP8 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50210668((3R)-3-amino-4-(2,5-difluorophenyl)-1-(3-(2,4-difl...)
Affinity DataIC50: >5.80E+4nMAssay Description:Inhibition of DPP9 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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