Compile Data Set for Download or QSAR
maximum 50k data
Found 12 Enz. Inhib. hit(s) with all data for entry = 50038201
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM50373059(CHEMBL429317)
Affinity DataKi:  4.5nMAssay Description:Displacement of [125I]alpha-bungarotoxin from alpha-7 nAChR in rat hipocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM50373059(CHEMBL429317)
Affinity DataKi:  4.5nMAssay Description:Displacement of [125I]alpha-bungarotoxin from alpha-7 nAChR in rat amygdalaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM50373059(CHEMBL429317)
Affinity DataKi:  10nMAssay Description:Displacement of [125I]alpha-bungarotoxin from alpha-7 nAChR in rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM50373059(CHEMBL429317)
Affinity DataIC50:  12nMAssay Description:Displacement of [125I]alpha-bungarotoxin from alpha-7 nAChR in rat hipocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM50373059(CHEMBL429317)
Affinity DataIC50:  12nMAssay Description:Displacement of [125I]alpha-bungarotoxin from alpha-7 nAChR in rat amygdalaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM50373059(CHEMBL429317)
Affinity DataIC50:  28nMAssay Description:Displacement of [125I]alpha-bungarotoxin from alpha-7 nAChR in rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50373059(CHEMBL429317)
Affinity DataEC50:  600nMAssay Description:Activation of human alpha-7 nAChR expressed in Xenopus oocytes assessed as modulation of choline-induced current by two-electrode voltage-clamp metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50373059(CHEMBL429317)
Affinity DataEC50:  6.30E+3nMAssay Description:Activation of human GABAA alpha-2-beta-3-gamma-2L receptor expressed in Xenopus oocytes assessed as modulation of GABA-induced current by two-electro...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50373059(CHEMBL429317)
Affinity DataEC50:  700nMAssay Description:Activation of human alpha-7 nAChR expressed in Xenopus oocytes assessed as modulation of acetyl choline -induced current by two-electrode voltage-cla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50373060(CHEMBL257155)
Affinity DataEC50:  1.80E+3nMAssay Description:Activation of human alpha-7 nAChR expressed in Xenopus oocytes assessed as modulation of nicotine-induced current by two-electrode voltage-clamp meth...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50373059(CHEMBL429317)
Affinity DataEC50:  500nMAssay Description:Activation of human alpha-7 nAChR expressed in Xenopus oocytes assessed as modulation of nicotine-induced current by two-electrode voltage-clamp meth...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGABA-A receptor; alpha-2/beta-3/gamma-2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50373060(CHEMBL257155)
Affinity DataEC50:  200nMAssay Description:Activation of human GABAA alpha-2-beta-3-gamma-2L receptor expressed in Xenopus oocytes assessed as modulation of nicotine-induced current by two-ele...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed