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Found 24 Enz. Inhib. hit(s) with all data for entry = 50042267
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50115998(3-[(Benzyl-methyl-amino)-methyl]-8-(2,6-difluoro-b...)
Affinity DataIC50:  71nMAssay Description:Antagonist activity at human GnRHR expressed in CHO cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50423185(CHEMBL392008)
Affinity DataIC50:  309nMAssay Description:Antagonist activity at human GnRHR expressed in CHO cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50423173(CHEMBL392434)
Affinity DataIC50:  355nMAssay Description:Antagonist activity at human GnRHR expressed in CHO cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50423174(CHEMBL235132)
Affinity DataIC50:  468nMAssay Description:Antagonist activity at human GnRHR expressed in CHO cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50423180(CHEMBL392435)
Affinity DataIC50:  525nMAssay Description:Antagonist activity at human GnRHR expressed in CHO cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50423188(CHEMBL237734)
Affinity DataIC50:  676nMAssay Description:Antagonist activity at human GnRHR expressed in CHO cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50423168(CHEMBL238177)
Affinity DataIC50:  676nMAssay Description:Antagonist activity at human GnRHR expressed in CHO cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50423184(CHEMBL236221)
Affinity DataIC50:  724nMAssay Description:Antagonist activity at human GnRHR expressed in CHO cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50423187(CHEMBL235180)
Affinity DataIC50:  724nMAssay Description:Antagonist activity at human GnRHR expressed in CHO cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50423178(CHEMBL395825)
Affinity DataIC50:  832nMAssay Description:Antagonist activity at human GnRHR expressed in CHO cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50423179(CHEMBL236222)
Affinity DataIC50:  832nMAssay Description:Antagonist activity at human GnRHR expressed in CHO cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50423166(CHEMBL427981)
Affinity DataIC50:  955nMAssay Description:Antagonist activity at human GnRHR expressed in CHO cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50423175(CHEMBL235179)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity at human GnRHR expressed in CHO cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50423171(CHEMBL395826)
Affinity DataIC50:  1.32E+3nMAssay Description:Antagonist activity at human GnRHR expressed in CHO cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50423182(CHEMBL414045)
Affinity DataIC50:  1.35E+3nMAssay Description:Antagonist activity at human GnRHR expressed in CHO cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50423183(CHEMBL235361)
Affinity DataIC50:  1.55E+3nMAssay Description:Antagonist activity at human GnRHR expressed in CHO cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50423169(CHEMBL393486)
Affinity DataIC50:  1.91E+3nMAssay Description:Antagonist activity at human GnRHR expressed in CHO cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50423176(CHEMBL439200)
Affinity DataIC50:  1.91E+3nMAssay Description:Antagonist activity at human GnRHR expressed in CHO cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50423172(CHEMBL438504)
Affinity DataIC50:  2.40E+3nMAssay Description:Antagonist activity at human GnRHR expressed in CHO cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50423186(CHEMBL397360)
Affinity DataIC50:  2.57E+3nMAssay Description:Antagonist activity at human GnRHR expressed in CHO cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50423167(CHEMBL396385)
Affinity DataIC50:  3.02E+3nMAssay Description:Antagonist activity at human GnRHR expressed in CHO cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50423181(CHEMBL392433)
Affinity DataIC50:  3.16E+3nMAssay Description:Antagonist activity at human GnRHR expressed in CHO cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50423177(CHEMBL237729)
Affinity DataIC50:  3.63E+3nMAssay Description:Antagonist activity at human GnRHR expressed in CHO cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50423170(CHEMBL238160)
Affinity DataIC50:  7.08E+3nMAssay Description:Antagonist activity at human GnRHR expressed in CHO cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed