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Found 14 Enz. Inhib. hit(s) with all data for entry = 50020436
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50213768(3-(4-(2-((4-(trifluoromethyl)benzyl)(benzo[d]thiaz...)
Affinity DataEC50:  4.46E+3nMAssay Description:Agonist activity at human PPARalpha receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50213769(3-(4-(2-(benzo[d]thiazol-2-yl(thiophen-2-ylmethyl)...)
Affinity DataEC50:  1.74E+3nMAssay Description:Agonist activity at human PPARdelta receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50213768(3-(4-(2-((4-(trifluoromethyl)benzyl)(benzo[d]thiaz...)
Affinity DataEC50:  3.69E+3nMAssay Description:Agonist activity at human PPARgamma receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50213771(3-(4-(2-((4-tert-butylbenzyl)(benzo[d]thiazol-2-yl...)
Affinity DataEC50:  6.34E+3nMAssay Description:Agonist activity at human PPARgamma receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50213770(3-(4-(2-(benzyl(6-chlorobenzo[d]thiazol-2-yl)amino...)
Affinity DataEC50:  1.36E+3nMAssay Description:Agonist activity at human PPARdelta receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50213772(3-(4-(2-(benzo[d]thiazol-2-yl(benzyl)amino)ethoxy)...)
Affinity DataEC50:  1.17E+3nMAssay Description:Agonist activity at human PPARdelta receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50213768(3-(4-(2-((4-(trifluoromethyl)benzyl)(benzo[d]thiaz...)
Affinity DataEC50:  940nMAssay Description:Agonist activity at human PPARdelta receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50213774(3-(4-(3-((6-chlorobenzo[d]thiazol-2-yl)(thiophen-2...)
Affinity DataEC50:  390nMAssay Description:Agonist activity at human PPARdelta receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM28661(2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)ph...)
Affinity DataEC50:  85nMAssay Description:Agonist activity at human PPARdelta receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50213775(3-(4-(3-(benzo[d]thiazol-2-yl(benzyl)amino)propoxy...)
Affinity DataEC50:  2.55E+3nMAssay Description:Agonist activity at human PPARdelta receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50213771(3-(4-(2-((4-tert-butylbenzyl)(benzo[d]thiazol-2-yl...)
Affinity DataEC50:  4.88E+3nMAssay Description:Agonist activity at human PPARdelta receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50213777(3-(4-(2-(benzo[d]thiazol-2-yl(benzyl)amino)ethoxy)...)
Affinity DataEC50:  2.97E+3nMAssay Description:Agonist activity at human PPARdelta receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50213776(3-(4-(2-(benzyl(6-methylbenzo[d]thiazol-2-yl)amino...)
Affinity DataEC50:  2.61E+3nMAssay Description:Agonist activity at human PPARdelta receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50213773(3-(4-(2-(benzo[d]thiazol-2-yl(benzyl)amino)ethoxy)...)
Affinity DataEC50:  2.81E+3nMAssay Description:Agonist activity at human PPARdelta receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed