Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with all data for entry = 50025309
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50270042((2-hydroxy-4-morpholinophenyl)(phenyl)methanone | ...)
Affinity DataIC50:  270nMAssay Description:Inhibition of DNA-PKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50159620(2-Morpholin-4-yl-pyrimido[2,1-a]isoquinolin-4-one ...)
Affinity DataIC50:  280nMAssay Description:Inhibition of DNA-PKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM12915(2-(4-Morpholinyl)-8-phenyl-4H-1-benzopyran-4-one |...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50159620(2-Morpholin-4-yl-pyrimido[2,1-a]isoquinolin-4-one ...)
Affinity DataIC50:  5.30E+3nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50270042((2-hydroxy-4-morpholinophenyl)(phenyl)methanone | ...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50159620(2-Morpholin-4-yl-pyrimido[2,1-a]isoquinolin-4-one ...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of p110alpha/p85-alpha PI3KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed