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Found 24 Enz. Inhib. hit(s) with all data for entry = 50020728
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50216982(CHEMBL235239 | UMB-97 | UMB97)
Affinity DataKi:  4.30nMAssay Description:Displacement of [3H]DAMGO from cloned mu opioid receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50216981(CHEMBL238017 | UMB-95 | UMB95)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]DAMGO from cloned mu opioid receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50216980(CHEMBL401245 | UMB-94 | UMB94)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]DAMGO from cloned mu opioid receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50216980(CHEMBL401245 | UMB-94 | UMB94)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]DPDPE from cloned delta opioid receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50216980(CHEMBL401245 | UMB-94 | UMB94)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]U-69593 from cloned kappa opioid receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50216981(CHEMBL238017 | UMB-95 | UMB95)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]DPDPE from cloned delta opioid receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50216983(CHEMBL392269 | UMB-96 | UMB96)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]DAMGO from cloned mu opioid receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50216981(CHEMBL238017 | UMB-95 | UMB95)
Affinity DataKi:  64nMAssay Description:Displacement of [3H]U-69593 from cloned kappa opioid receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50216983(CHEMBL392269 | UMB-96 | UMB96)
Affinity DataKi:  110nMAssay Description:Displacement of [3H]DPDPE from cloned delta opioid receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50216982(CHEMBL235239 | UMB-97 | UMB97)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]DPDPE from cloned delta opioid receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50216983(CHEMBL392269 | UMB-96 | UMB96)
Affinity DataKi:  170nMAssay Description:Displacement of [3H]U-69593 from cloned kappa opioid receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50216982(CHEMBL235239 | UMB-97 | UMB97)
Affinity DataKi:  230nMAssay Description:Displacement of [3H]U-69593 from cloned kappa opioid receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50216983(CHEMBL392269 | UMB-96 | UMB96)
Affinity DataEC50:  520nMAssay Description:Agonist activity at human kappa opioid receptor expressed in CHO membrane by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50216981(CHEMBL238017 | UMB-95 | UMB95)
Affinity DataEC50:  210nMAssay Description:Agonist activity at human kappa opioid receptor expressed in CHO membrane by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50216982(CHEMBL235239 | UMB-97 | UMB97)
Affinity DataEC50:  12nMAssay Description:Agonist activity at human mu opioid receptor expressed in CHO membrane by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50216982(CHEMBL235239 | UMB-97 | UMB97)
Affinity DataEC50:  720nMAssay Description:Agonist activity at human kappa opioid receptor expressed in CHO membrane by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50216983(CHEMBL392269 | UMB-96 | UMB96)
Affinity DataEC50:  89nMAssay Description:Agonist activity at human mu opioid receptor expressed in CHO membrane by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50216980(CHEMBL401245 | UMB-94 | UMB94)
Affinity DataEC50:  240nMAssay Description:Agonist activity at human kappa opioid receptor expressed in CHO membrane by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50216981(CHEMBL238017 | UMB-95 | UMB95)
Affinity DataEC50:  15nMAssay Description:Agonist activity at human mu opioid receptor expressed in CHO membrane by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50216981(CHEMBL238017 | UMB-95 | UMB95)
Affinity DataEC50:  21nMAssay Description:Agonist activity at human delta opioid receptor expressed in CHO membrane by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50216980(CHEMBL401245 | UMB-94 | UMB94)
Affinity DataEC50:  88nMAssay Description:Agonist activity at human delta opioid receptor expressed in CHO membrane by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50216980(CHEMBL401245 | UMB-94 | UMB94)
Affinity DataEC50:  43nMAssay Description:Agonist activity at human mu opioid receptor expressed in CHO membrane by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50216982(CHEMBL235239 | UMB-97 | UMB97)
Affinity DataEC50:  57nMAssay Description:Agonist activity at human delta opioid receptor expressed in CHO membrane by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50216983(CHEMBL392269 | UMB-96 | UMB96)
Affinity DataEC50:  210nMAssay Description:Agonist activity at human delta opioid receptor expressed in CHO membrane by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed