Found 4 Enz. Inhib. hit(s) with all data for entry = 50025407 TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Of Bern
Curated by ChEMBL
University Of Bern
Curated by ChEMBL
Affinity DataEC50: 191nMAssay Description:Activity at rat wild type GABAA alpha1beta2gamma2 receptor expressed in xenopus oocytes assessed as GABA-elicited response by two electrode voltage c...More data for this Ligand-Target Pair
3D Structure (crystal)TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Of Bern
Curated by ChEMBL
University Of Bern
Curated by ChEMBL
Affinity DataKd: 878nMAssay Description:Displacement of [3H]Ro15-1788 from rat GABAA alpha1beta2gamma2 receptor expressed in HEK293 cells after 1 hr assessed as residual binding by liquid s...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Of Bern
Curated by ChEMBL
University Of Bern
Curated by ChEMBL
Affinity DataEC50: 1.10nMAssay Description:Activity at rat wild type GABAA alpha1beta2gamma2 receptor expressed in xenopus oocytes assessed as GABA-elicited response by two electrode voltage c...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
University Of Bern
Curated by ChEMBL
University Of Bern
Curated by ChEMBL
Affinity DataEC50: 250nMAssay Description:Activity at rat wild type GABAA alpha1beta2gamma2 receptor expressed in xenopus oocytes assessed as GABA-elicited response by two electrode voltage c...More data for this Ligand-Target Pair
